Patil, Rameshwar, Elz, Sigurd and Reiser, Oliver (2006) Side-chain modified analogues of histaprodifen: Asymmetric synthesis and histamine H₁-receptor activity. Bioorg. Med. Chem. Lett. 16 (3), pp. 672-676.
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Other URL: http://dx.doi.org/10.1016/j.bmcl.2005.10.030
Abstract
New analogues of histaprodifen with polar side chains have been stereoselectively synthesized and evaluated as histamine H₁-receptor agonists. As a key transformation the asymmetric aminohydroxylation has been used, which was successfully realized for the first time on an imidazolyl derivative. While all chiral analogues proved to be weak H₁-receptor antagonists, an achiral keto derivative of ...
Export bibliographical data
| Item type: | Article | ||||
|---|---|---|---|---|---|
| Date: | 1 February 2006 | ||||
| Institutions: | Chemistry and Pharmacy > Institut für Organische Chemie > Lehrstuhl Prof. Dr. Oliver Reiser | ||||
| Identification Number: |
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| Dewey Decimal Classification: | 500 Science > 540 Chemistry & allied sciences | ||||
| Status: | Published | ||||
| Refereed: | Yes, this version has been refereed | ||||
| Created at the University of Regensburg: | Yes | ||||
| Item ID: | 359 |
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