Influence of the N-terminus and the E2-loop onto the binding kinetics of the antagonist mepyramine and the partial agonist phenoprodifen to H1R
Wittmann, Hans-Joachim, Seifert, Roland and Strasser, Andrea (2011) Influence of the N-terminus and the E2-loop onto the binding kinetics of the antagonist mepyramine and the partial agonist phenoprodifen to H1R. Biochemical Pharmacology 12, pp. 1910-1918.Date of publication of this fulltext: 25 Jan 2012 08:47
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| Item type | Article | ||||
| Journal or Publication Title | Biochemical Pharmacology | ||||
| Publisher: | PERGAMON-ELSEVIER SCIENCE LTD | ||||
|---|---|---|---|---|---|
| Place of Publication: | OXFORD | ||||
| Volume: | 12 | ||||
| Page Range: | pp. 1910-1918 | ||||
| Date | 2011 | ||||
| Institutions | Chemistry and Pharmacy > Institute of Pharmacy | ||||
| Identification Number |
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| Keywords | PROTEIN-COUPLED RECEPTOR; HISTAMINE H-1 RECEPTOR; IN-VITRO EVALUATION; H-1-RECEPTOR AGONISTS; INTERNATIONAL UNION; CRYSTAL-STRUCTURE; HISTAPRODIFENS; PHARMACOLOGY; COMPLEX; POCKET; Histamine H-1 receptor; Binding kinetics; Gibbs energy; Extracellular surface; Molecular modelling; Molecular dynamics | ||||
| Dewey Decimal Classification | 600 Technology > 615 Pharmacy | ||||
| Status | Published | ||||
| Refereed | Yes, this version has been refereed | ||||
| Created at the University of Regensburg | Yes | ||||
| Item ID | 23277 |
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