Bibliography of the Universität Regensburg

University of Regensburg (2629)
- Chemistry and Pharmacy (2629)
  - Institute of Pharmacy (2629)
    - Group Clinical Pharmacy (Dr. Dorn) (61)
    - Pharmaceutical Biology (Prof. Heilmann) (275)
    - Pharmaceutical Technology (Prof. Göpferich) (464)
    - Pharmaceutical/Medicinal Chemistry I (Prof. Elz) (166)
    - Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer) (629)
    - Pharmacology and Toxicology (Prof. Schlossmann, formerly Prof. Seifert) (333)
    - Alumni or Retired Professors (726)

Group by: Date | Creators | Item type | No Grouping

Jump to: 2025 | 2024 | 2023 | 2022 | 2021 | 2020 | 2019 | 2018 | 2017 | 2016 | 2015 | 2014 | 2013 | 2012 | 2011 | 2010 | 2009 | 2008 | 2007 | 2006 | 2005 | 2004 | 2003 | 2002 | 2001 | 2000

Number of items at this level: 270.

2025

Schettler, Franziska, Gattor, Albert O., Koch, Pierre

and Keller, Max

(2025) Characterization of [3H]Propionylated Human Peptide YY-A New Probe for Neuropeptide Y Y2 Receptor Binding Studies. ACS Pharmacology & Translational Science 8 (3), pp. 785-799.

Zimmer, Oliver (2025) Contributions to the Fundamental Understanding of Nanoparticle Cell Interactions and Target-Specific Biodistribution. PhD, Universität Regensburg.

Brunner, Julia (2025) Phytochemische und pharmakologische in vitro Untersuchungen von Hypericum tetrapterum Fr. PhD, Universität Regensburg.

2024

Müller, Christoph

(2024) Structure-based development of nonpeptidic fluorescent probes, PET tracers and homobivalent neuropeptide Y Y1 receptor ligands with picomolar binding affinities. PhD, Universität Regensburg.

Rosier, Niklas (2024) Synthesis and pharmacological characterization of bivalent ligands for the D1-H3 receptor heteromer and fluorescent ligands for the D1 and H3 receptors. PhD, Universität Regensburg.

Gonzalez-Valerio, Carlos, Peregrina-Lucano, Alejandro A.

, Manríquez-González, Ricardo, Pérez-Fonseca, Aida A., Robledo-Ortíz, Jorge R., Shenderovich, Ilya G.

and Gómez-Salazar, Sergio (2024) Color Compounds Removal from Tequila Vinasses Using Silica Gel Adsorbents Functionalized with Thiol Moieties: Equilibrium and Kinetics Studies. Molecules 29 (24), p. 5910.

Becker, Jasmin, Ellerkmann, Clara S., Schmelzer, Hannah, Hermann, Christian, Lützel, Kyra, Gudermann, Thomas, Konrad, David B., Trauner, Dirk, Storch, Ursula

and Mederos y Schnitzler, Michael (2024) Optical Control of TRPM8 Channels with Photoswitchable Menthol. Angewandte Chemie International Edition.

Ferrando Plo, Lucas

, Nitsopoulos, Athanasios, Friedle, Albrecht, Schmidberger, Andreas and Heilmann, Jörg (2024) Anthraquinone Residues in Dried Walnut (Juglans regia) Leaves for Herbal Infusions: Proof of Endogenous Origin via a Sampling-Driven and GC-MS/MS-Based Strategy. Journal of Agricultural and Food Chemistry 72 (48), pp. 26915-26925.

Ertl, Fabian J., Kopanchuk, Sergei

, Dijon, Nicola C., Veikšina, Santa, Tahk, Maris-Johanna

, Laasfeld, Tõnis, Schettler, Franziska, Gattor, Albert O., Hübner, Harald, Archipowa, Nataliya

, Köckenberger, Johannes, Heinrich, Markus R., Gmeiner, Peter

, Kutta, Roger Jan

, Holliday, Nicholas D.

, Rinken, Ago

and Keller, Max

(2024) Dually Labeled Neurotensin NTS1R Ligands for Probing Radiochemical and Fluorescence-Based Binding Assays. Journal of Medicinal Chemistry 67 (18), pp. 16664-16691.

2023

Stahl, Monika (2023) Polymeric Nanoparticles for Antigen Delivery to Dendritic Cells. PhD, Universität Regensburg.

Höring, Carina

(2023) Split-Luciferase Complementation and Molecular Dynamics Studies for the Mini-G Protein-Based Functional Characterization of GPCRs. PhD, Universität Regensburg.

Geiben, Ann-Kathrin Christine Maria (2023) Analyse von Sedierung als unerwünschte Arzneimittelwirkung und Entwicklung eines Risikoscores für die Gerontopsychiatrie. PhD, Universität Regensburg.

Bresinsky, Merlin, Shahraki, Aida

, Kolb, Peter

, Pockes, Steffen

and Schihada, Hannes (2023) Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3. Journal of Medicinal Chemistry 66 (21), pp. 15025-15041. Fulltext not available.

Mönnich, Denise, Nagl, Martin, Forster, Lisa, Rosier, Niklas, Igel, Patrick and Pockes, Steffen (2023) Discovery of a Tritiated Radioligand with High Affinity and Selectivity for the Histamine H3 Receptor. ACS Medicinal Chemistry Letters 14 (11), pp. 1589-1595. Fulltext not available.

Szczepańska, Katarzyna, Karcz, Tadeusz, Dichiara, Maria, Mogilski, Szczepan, Kalinowska-Tłuścik, Justyna, Pilarski, Bogusław, Leniak, Arkadiusz, Pietruś, Wojciech

, Podlewska, Sabina

, Popiołek-Barczyk, Katarzyna, Humphrys, Laura J.

, Ruiz-Cantero, M. Carmen, Reiner-Link, David

, Leitzbach, Luisa, Łażewska, Dorota, Pockes, Steffen

, Górka, Michał, Zmysłowski, Adam, Calmels, Thierry, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Bojarski, Andrzej J., Amata, Emanuele and Kieć-Kononowicz, Katarzyna (2023) Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain. Journal of Medicinal Chemistry 66 (14), pp. 9658-9683. Fulltext not available.

Plut, Eva

, Calderón, Jacqueline C., Stanojlović, Vesna, Gattor, Albert O., Höring, Carina, Humphrys, Laura J., Konieczny, Adam, Kerres, Sabine, Schubert, Mario

, Keller, Max, Cabrele, Chiara, Clark, Timothy and Reiser, Oliver (2023) Stereochemistry-Driven Interactions of α,γ-Peptide Ligands with the Neuropeptide Y Y4-Receptor. Journal of Medicinal Chemistry 66 (14), pp. 9642-9657. Fulltext not available.

Gleixner, Jakob, Gattor, Albert O., Humphrys, Laura J., Brunner, Thomas and Keller, Max (2023) [3H]UR-JG102–A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y4 Receptor. Journal of Medicinal Chemistry 66 (19), pp. 13788-13808. Fulltext not available.

2022

Bohley, Marilena (2022) Targeted Lipid Nanoparticles for Retinal Drug Delivery. PhD, Universität Regensburg.

Forster, Lisa and Pockes, Steffen

(2022) Investigating the ligand agonism and antagonism at the D2long receptor by dynamic mass redistribution. Scientific Reports 12 (1).

Bresinsky, Merlin, Strasser, Jessica M., Hubmann, Alexander, Vallaster, Bernadette, McCue, William M., Fuller, Jessica, Singh, Gurpreet, Nelson, Kathryn M., Cuellar, Matthew E., Finzel, Barry C., Ashe, Karen H., Walters, Michael A. and Pockes, Steffen

(2022) Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis. Archiv der Pharmazie 355 (9), p. 2200095.

Endres, Katharina Walburga Maria

(2022) Wirkstoffkonzentrationsbestimmungen zur Therapieleitung der medikamentösen Behandlung kardiovaskulärer Erkrankungen bei psychiatrischen Patienten. PhD, Universität Regensburg.

Tahk, Maris-Johanna

, Torp, Jane

, Ali, Mohammed A. S.

, Fishman, Dmytro, Parts, Leopold

, Grätz, Lukas

, Müller, Christoph

, Keller, Max

, Veiksina, Santa

, Laasfeld, Tõnis

and Rinken, Ago

(2022) Live-cell microscopy or fluorescence anisotropy with budded baculoviruses—which way to go with measuring ligand binding to M 4 muscarinic receptors? Open Biology 12 (6). Fulltext not available.

Lier, Svenja, Sellmer, Andreas, Orben, Felix

, Heinzlmeir, Stephanie, Krauß, Lukas

, Schneeweis, Christian, Hassan, Zonera

, Schneider, Carolin

, Patricia Gloria Schäfer, Arlett, Pongratz, Herwig, Engleitner, Thomas, Öllinger, Rupert, Kuisl, Anna, Bassermann, Florian, Schlag, Christoph, Kong, Bo, Dove, Stefan, Kuster, Bernhard, Rad, Roland, Reichert, Maximilian, Wirth, Matthias

, Saur, Dieter

, Mahboobi, Siavosh and Schneider, Günter

(2022) A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer. Bioorganic Chemistry 119, p. 105505. Fulltext not available.

Schihada, Hannes, Klompstra, Thomas M.

, Humphrys, Laura J.

, Cervenka, Igor, Dadvar, Shamim

, Kolb, Peter

, Ruas, Jorge L.

and Schulte, Gunnar

(2022) Isoforms of GPR35 have distinct extracellular N-termini that allosterically modify receptor-transducer coupling and mediate intracellular pathway bias. Journal of Biological Chemistry 298 (9), p. 102328. Fulltext not available.

Shcherbina, Nadezhda A., Kazakov, Igor V., Lisovenko, Anna S., Kryukova, Mariya A., Krasnova, Irina S.

, Bodensteiner, Michael and Timoshkin, Alexey Y. (2022) Molecular complexes of non-chelating polydentate Lewis bases with group 13 Lewis acids: crystal structure and computed energy of stepwise donor–acceptor bond formation. Mendeleev Communications 32 (1), pp. 74-77. Fulltext not available.

Schindler, Lisa, Wohlfahrt, Katrin, Gluhacevic von Krüchten, Lara, Prante, Olaf, Keller, Max and Maschauer, Simone (2022) Neurotensin analogs by fluoroglycosylation at Nω-carbamoylated arginines for PET imaging of NTS1-positive tumors. Scientific Reports 12 (1). Fulltext not available.

Tang, Tingting, Tan, Qiuxiang, Han, Shuo, Diemar, Anne, Löbner, Kristin, Wang, Hongyu, Schüß, Corinna, Behr, Victoria, Mörl, Karin, Wang, Mu, Chu, Xiaojing, Yi, Cuiying, Keller, Max, Kofoed, Jacob, Reedtz-Runge, Steffen, Kaiser, Anette, Beck-Sickinger, Annette G., Zhao, Qiang and Wu, Beili (2022) Receptor-specific recognition of NPY peptides revealed by structures of NPY receptors. Science Advances 8 (18). Fulltext not available.

Müller, Christoph, Gleixner, Jakob

, Tahk, Maris-Johanna

, Kopanchuk, Sergei

, Laasfeld, Tõnis, Weinhart, Michael, Schollmeyer, Dieter, Betschart, Martin U., Lüdeke, Steffen, Koch, Pierre, Rinken, Ago

and Keller, Max (2022) Structure-Based Design of High-Affinity Fluorescent Probes for the Neuropeptide Y Y1 Receptor. Journal of Medicinal Chemistry 65 (6), pp. 4832-4853. Fulltext not available.

Rösch, G., El Bagdadi, K., Muschter, D., Taheri, S.

, Dorn, C., Meurer, A., Straub, R.H., Zaucke, F.

, Schilling, A.F., Grässel, S. and Jenei-Lanzl, Z.

(2022) Sympathectomy aggravates subchondral bone changes during osteoarthritis progression in mice without affecting cartilage degeneration or synovial inflammation. Osteoarthritis and Cartilage 30 (3), pp. 461-474. Fulltext not available.

2021

Lawrowska, Alexandra (2021) Nanoparticles for drug delivery to ocular neovascularizations. PhD, Universität Regensburg.

Seibel-Ehlert, Ulla

, Plank, Nicole, Inoue, Asuka, Bernhardt, Guenther

and Strasser, Andrea (2021) Label-Free Investigations on the G Protein Dependent Signaling Pathways of Histamine Receptors. International Journal of Molecular Sciences 22 (18), pp. 1-33.

Antoni, Frauke

(2021) Design, Synthesis and Characterization of ABCG2 Inhibitors with a Focus on Water Solubility and Stability in Plasma. PhD, Universität Regensburg.

Wolfgarten, Eva Maria (2021) HPTLC, HPLC-UV und HPLC-MS Untersuchungen zur Isolierung, zum Fingerprint und zur Quantifizierung von Iridoid- und Phenylethanoidglykosiden in den Blättern von Plantago lanceolata L. PhD, Universität Regensburg.

Rosier, Niklas, Grätz, Lukas, Schihada, Hannes

, Möller, Jan, Işbilir, Ali

, Humphrys, Laura J.

, Nagl, Martin, Seibel, Ulla, Lohse, Martin J.

and Pockes, Steffen

(2021) A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor. Journal of Medicinal Chemistry 64 (15), pp. 11695-11708. Fulltext not available.

Endres, Katharina, Schiller, Ernst and Haen, Ekkehard (2021) Antihypertensiva in der Psychiatrie. Der Nervenarzt 92, pp. 487-792.

Antoni, Frauke

and Bernhardt, Günther (2021) Derivatives of nitrogen mustard anticancer agents with improved cytotoxicity. Archiv der Pharmazie 354, e2000366.

Tropmann, Katharina, Seibel-Ehlert, Ulla, Littmann, Timo and Strasser, Andrea (2021) Shining light on the histamine H2 receptor: Synthesis of carbamoylguanidine-type agonists as a pharmacological tool to study internalization. Bioorganic & Medicinal Chemistry Letters 52, p. 128388. Fulltext not available.

Eap, C. B.

, Gründer, G.

, Baumann, P.

, Ansermot, N., Conca, A., Corruble, E., Crettol, S., Dahl, M. L., de Leon, J.

, Greiner, C., Howes, O., Kim, E., Lanzenberger, R., Meyer, J. H., Moessner, R., Mulder, H., Müller, D. J., Reis, M., Riederer, P., Ruhe, H. G., Spigset, O., Spina, E., Stegman, B., Steimer, W., Stingl, J.

, Suzen, S., Uchida, H., Unterecker, S., Vandenberghe, F.

and Hiemke, C.

(2021) Tools for optimising pharmacotherapy in psychiatry (therapeutic drug monitoring, molecular brain imaging and pharmacogenetic tests): focus on antidepressants. The World Journal of Biological Psychiatry 22 (8), pp. 561-628. Fulltext not available.

2020

Höring, Carina

, Seibel, Ulla

, Tropmann, Katharina, Grätz, Lukas

, Mönnich, Denise

, Pitzl, Sebastian, Bernhardt, Günther

, Pockes, Steffen

and Strasser, Andrea (2020) A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes. International Journal of Molecular Sciences 21 (22), p. 8440.

Grätz, Lukas, Tropmann, Katharina, Bresinsky, Merlin, Müller, Christoph, Bernhardt, Günther

and Pockes, Steffen (2020) NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells. Scientific Reports 10, p. 13288.

Schwarz, Mirjam (2020) Erstellung eines Hypotonie-Risikoscores und Validierung anhand einer retrospektiven Anwendungsbeobachtung an geriatrischen Patienten. PhD, Universität Regensburg.

Thalhauser, Stefanie and Breunig, Miriam

(2020) Considerations for efficient surface functionalization of nanoparticles with a high molecular weight protein as targeting ligand. European Journal of Pharmaceutical Sciences 155 (105520). Fulltext not available.

Bartole, Edith, Grätz, Lukas, Littmann, Timo, Wifling, David

, Seibel, Ulla, Buschauer, Armin

and Bernhardt, Günther (2020) UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors. Journal of Medicinal Chemistry 63 (10), pp. 5297-5311. Fulltext not available.

Maslanka Figueroa, Sara

, Fleischmann, Daniel, Beck, Sebastian, Tauber, Philipp, Witzgall, Ralph, Schweda, Frank and Goepferich, Achim (2020) Nanoparticles Mimicking Viral Cell Recognition Strategies Are Superior Transporters into Mesangial Cells. Advanced Science 7 (11), p. 1903204.

Dorn, Christoph

, Schießer, Selina, Wulkersdorfer, Beatrix, Hitzenbichler, Florian, Kees, Martin G.

and Zeitlinger, Markus (2020) Determination of free clindamycin, flucloxacillin or tedizolid in plasma: Keep attention to physiological conditions when using ultrafiltration. Biomedical Chromatography 34, e4820.

Abstiens, Kathrin

(2020) Heteromultivalent Nanoparticles for Selective Targeting of Renal Cells. PhD, Universität Regensburg.

Fleischmann, Daniel, Maslanka-Figueroa, Sara, Beck, Sebastian, Abstiens, Kathrin, Witzgall, Ralph, Schweda, Frank, Tauber, Philipp and Goepferich, Achim

(2020) Adenovirus-Mimetic Nanoparticles: Sequential Ligand-Receptor Interplay as a Universal Tool for Enhanced In Vitro/In Vivo Cell Identification. ACS Applied Materials & Interfaces 12 (31), pp. 34689-34702. Fulltext not available.

Spinnler, Katrin, von Krüchten, Lara, Konieczny, Adam, Schindler, Lisa, Bernhardt, Günther and Keller, Max (2020) An Alkyne-functionalized Arginine for Solid-Phase Synthesis Enabling “Bioorthogonal” Peptide Conjugation. ACS Medicinal Chemistry Letters 11 (3), pp. 334-339. Fulltext not available.

Weber, Laura, Kuck, Katrin, Jürgenliemk, Guido, Heilmann, Jörg, Lipowicz, Bartosz and Vissiennon, Cica

(2020) Anti-Inflammatory and Barrier-Stabilising Effects of Myrrh, Coffee Charcoal and Chamomile Flower Extract in a Co-Culture Cell Model of the Intestinal Mucosa. Biomolecules 10 (7), p. 1033. Fulltext not available.

Buschmann, Jonas, Seiler, Theresa, Bernhardt, Günther, Keller, Max and Wifling, David (2020) Argininamide-type neuropeptide Y Y1 receptor antagonists: the nature of Nω-carbamoyl substituents determines Y1R binding mode and affinity. RSC Medicinal Chemistry 11 (2), pp. 274-282. Fulltext not available.

Ullah, Sami, Beer, Ronny, Fuhr, Uwe, Taubert, Max

, Zeitlinger, Markus, Kratzer, Alexander, Dorn, Christoph, Arshad, Usman, Kofler, Mario and Helbok, Raimund (2020) Brain Exposure to Piperacillin in Acute Hemorrhagic Stroke Patients Assessed by Cerebral Microdialysis and Population Pharmacokinetics. Neurocritical Care.

Thalhauser, Stefanie and Breunig, Miriam

Bohley, Marilena S., Birch, Emily, Baumann, Felix J., Dillinger, Andrea E., Tamm, Ernst R. and Goepferich, Achim M. (2020) Design of dye and superparamagnetic iron oxide nanoparticle loaded lipid nanocapsules with dual detectability in vitro and in vivo. International Journal of Pharmaceutics 585, p. 119433. Fulltext not available.

Gruber, Corinna G., Pegoli, Andrea, Müller, Christoph, Grätz, Lukas, She, Xueke and Keller, Max (2020) Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity. RSC Medicinal Chemistry 11 (7), pp. 823-832. Fulltext not available.

Tropmann, Katharina, Höring, Carina

, Plank, Nicole and Pockes, Steffen

(2020) Discovery of a G Protein-Biased Radioligand for the Histamine H2 Receptor with Reversible Binding Properties. Journal of Medicinal Chemistry 63 (21), pp. 13090-13102. Fulltext not available.

Keller, Max, Mahuroof, Shahani A., Hong Yee, Vivyanne, Carpenter, Jessica, Schindler, Lisa, Littmann, Timo, Pegoli, Andrea, Hübner, Harald, Bernhardt, Günther, Gmeiner, Peter

and Holliday, Nicholas D.

(2020) Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity. ACS Medicinal Chemistry Letters 11 (1), pp. 16-22. Fulltext not available.

Biselli, Sabrina, Alencastre, Inês, Tropmann, Katharina, Erdmann, Daniela, Chen, Mengya, Littmann, Timo, Maia, André F.

, Gomez-Lazaro, Maria, Tanaka, Miho, Ozawa, Takeaki, Keller, Max, Lamghari, Meriem, Buschauer, Armin and Bernhardt, Günther (2020) Fluorescent H2 Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications. ACS Medicinal Chemistry Letters 11 (8), pp. 1521-1528. Fulltext not available.

Abdellatif, Ahmed

, Hennig, Robert, Pollinger, Klaus, Tawfeek, Hesham and Goepferich, Achim (2020) Fluorescent Nanoparticles Coated with a Somatostatin Analogue Target Blood Monocyte for Efficient Leukaemia Treatment. Pharmaceutical Research 37 (11), p. 2017.

Sommer, Judith, Dorn, Christoph

, Gäbele, Erwin, Bataille, Frauke, Freese, Kim, Seitz, Tatjana, Thasler, Wolfgang E., Büttner, Reinhard, Weiskirchen, Ralf

, Bosserhoff, Anja

and Hellerbrand, Claus (2020) Four-And-A-Half LIM-Domain Protein 2 (FHL2) Deficiency Aggravates Cholestatic Liver Injury. Cells 9 (1), p. 248.

Apaolaza, P.S.

, Busch, M., Asin-Prieto, E.

, Peynshaert, K.

, Rathod, R., Remaut, K., Dünker, N. and Göpferich, A. (2020) Hyaluronic acid coating of gold nanoparticles for intraocular drug delivery: Evaluation of the surface properties and effect on their distribution. Experimental Eye Research 198, p. 108151. Fulltext not available.

Biswas, Siladitta, Kojonazarov, Baktybek, Hadzic, Stefan, Majer, Michael, Bajraktari, Ganimete, Novoyatleva, Tatyana, Ghofrani, Hossein Ardeschir, Grimminger, Friedrich, Seeger, Werner, Weissmann, Norbert, Schlossmann, Jens and Schermuly, Ralph Theo (2020) IRAG1 Deficient Mice Develop PKG1β Dependent Pulmonary Hypertension. Cells 9 (10), p. 2280. Fulltext not available.

Yagati, Ajay Kumar

, Behrent, Arne, Beck, Sebastian, Rink, Simone, Goepferich, Achim M., Min, Junhong

, Lee, Min-Ho

and Baeumner, Antje J.

(2020) Laser-induced graphene interdigitated electrodes for label-free or nanolabel-enhanced highly sensitive capacitive aptamer-based biosensors. Biosensors and Bioelectronics 164, p. 112272. Fulltext not available.

Pontes de Sousa, Ingrid, Ferreira, Antônio Gilberto

, Miller Crotti, Antônio Eduardo, Alves dos Santos, Raquel, Kiermaier, Josef, Kraus, Birgit, Heilmann, Jörg and Jacometti Cardoso Furtado, Niege Araçari (2020) New antifungal ent-labdane diterpenes against Candida glabrata produced by microbial transformation of ent-polyalthic acid. Bioorganic Chemistry 95, p. 103560. Fulltext not available.

Konieczny, Adam, Braun, Diana, Wifling, David

, Bernhardt, Günther and Keller, Max (2020) Oligopeptides as Neuropeptide Y Y4 Receptor Ligands: Identification of a High-Affinity Tetrapeptide Agonist and a Hexapeptide Antagonist. Journal of Medicinal Chemistry 63 (15), pp. 8198-8215. Fulltext not available.

Thalhauser, Stefanie, Peterhoff, David, Wagner, Ralf and Breunig, Miriam

(2020) Presentation of HIV-1 Envelope Trimers on the Surface of Silicia Nanoparticles. Journal of Pharmaceutical Sciences 109, pp. 911-921. Fulltext not available.

Ehmann, L., Simon, P., Busse, D., Petroff, D., Dorn, Christoph

, Huisinga, W., Dietrich, A., Zeitlinger, M., Wrigge, H. and Kloft, C. (2020) Risk of target non-attainment In obese compared to non-obese patients In Calculated linezolid therapy. Clinical Microbiology and Infection. Fulltext not available.

Thalhauser, Stefanie, Peterhoff, David, Wagner, Ralf and Breunig, Miriam

(2020) Silica particles incorporated into PLGA-based in situ-forming implants exploit the dual advantage of sustained release and particulate delivery. European Journal of Pharmaceutics and Biopharmaceutics (156), pp. 1-10. Fulltext not available.

Stolwijk, Judith A., Mildner, Anne-Kathrin, Kade, Christian, Skiba, Michael, Bernhardt, Guenther, Buschauer, Armin, Huebner, Harald, Gmeiner, Peter and Wegener, Joachim (2020) Stepwise Dosing Protocol for Increased Throughput in Label-Free Impedance-Based GPCR Assays. Journal of Visualized Experiments (156). Fulltext not available.

2019

Silva Gracia, Margarete (2019) Verbesserung der Arzneimitteltherapiesicherheit von Antipsychotika und Beta-Adrenozeptor-Antagonisten durch Therapeutisches Drug Monitoring und Untersuchungen zu pharmakokinetischen Interaktionen. PhD, Universität Regensburg.

Maschauer, Simone, Ott, Julian J.

, Bernhardt, Günther, Kuwert, Torsten, Keller, Max and Prante, Olaf (2019) 18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET Imaging of mammary carcinoma. Scientific Reports 9, p. 12990.

Schramm, Andrea, Schweda, Frank, Sequeira-Lopez, Maria Luisa S., Hofmann, Franz, Sandner, Peter and Schlossmann, Jens (2019) Protein Kinase G Is Involved in Acute but Not in Long-Term Regulation of Renin Secretion. Frontiers in Pharmacology 2019 (10), p. 800.

Dorn, Christoph, Petroff, David, Neumann, Nancy, Kratzer, Alexander, El-Najjar, Nahed

, Dietrich, Arne, Kloft, Charlotte, Zeitlinger, Markus

, Kees, Martin, Kees, Frieder, Wrigge, Hermann and Simon, Philipp (2019) Plasma and tissue pharmacokinetics of fosfomycin in morbidly obese and non-obese surgical patients: a controlled clinical trial. Journal of Antimicrobial Chemotherapy. Fulltext not available.

Pegoli, Andrea, Wifling, David

, Gruber, Corinna G., Xueke, She, Hübner, Harald, Bernhardt, Günther, Gmeiner, Peter

and Keller, Max (2019) Conjugation of Short Peptides to Dibenzodiazepinone-Type
Muscarinic Acetylcholine Receptor Ligands Determines M2R
Selectivity. Journal of Medicinal Chemistry 62, pp. 5358-5369. Fulltext not available.

Schindler, Lisa, Bernhardt, Günther

and Keller, Max

(2019) Modifications at Arg and Ile Give Neurotensin(8−13) Derivatives with High Stability and Retained NTS1 Receptor Affinity. ACS Medicinal Chemistry Letters 10 (6), pp. 960-965. Fulltext not available.

Pockes, Steffen, Wifling, David

, Buschauer, Armin

and Elz, Sigurd (2019) Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands †. ChemistryOpen 8 (3), pp. 285-297.

Schramm, Simon, Agnetta, Luca, Bermudez, Marcel, Gerwe, Hubert, Irmen, Matthias, Holze, Janine, Littmann, Timo, Wolber, Gerhard

, Tränkle, Christian and Decker, Michael (2019) Novel BQCA‐ and TBPB‐Derived M 1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism. ChemMedChem 14 (14), pp. 1349-1358. Fulltext not available.

Wiegrebe, Wolfgang (2019) Adam and Eve's Origin According to Islam: A Response to Daud Abdul-Fattah Batchelor. Theology and Science 17 (4), pp. 455-468. Fulltext not available.

Łażewska, Dorota

, Mogilski, Szczepan, Hagenow, Stefanie

, Kuder, Kamil, Głuch-Lutwin, Monika

, Siwek, Agata

, Więcek, Małgorzata, Kaleta, Maria, Seibel, Ulla, Buschauer, Armin, Filipek, Barbara, Stark, Holger

and Kieć-Kononowicz, Katarzyna (2019) Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands. Bioorganic & Medicinal Chemistry 27 (7), pp. 1254-1262. Fulltext not available.

Polykandriotis, Elias, Horch, Raymund E., Jost, Matthias, Arkudas, Andreas, Kees, Frieder and Schmitz, Marweh (2019) Can systemically administered antibiotics be detected in wound tissues and surfaces under negative pressure wound therapy? International Wound Journal 16 (2), pp. 503-510. Fulltext not available.

Kowalewski, Christoph, Haen, Ekkehard, Hiemke, Christoph, Ridders, Florian, Endres, Katharina, Gründer, Gerhard, Paulzen, Michael and Schoretsanitis, Georgios (2019) Cytochrome P450-mediated inhibition of venlafaxine metabolism by trimipramine. International Clinical Psychopharmacology 34 (5), pp. 241-246. Fulltext not available.

Dorn, Christoph

, Kratzer, Alexander Ludwig, Schießer, Selina, Kees, Frieder

, Wrigge, Hermann and Simon, Philipp (2019) Determination of total or free cefazolin and metronidazole in human plasma or interstitial fluid by HPLC-UV for pharmacokinetic studies in man. Journal of Chromatography B. Fulltext not available.

Agnetta, Luca, Bermudez, Marcel

, Riefolo, Fabio

, Matera, Carlo

, Claro, Enrique

, Messerer, Regina, Littmann, Timo, Wolber, Gerhard

, Holzgrabe, Ulrike and Decker, Michael (2019) Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties. Journal of Medicinal Chemistry 62 (6), pp. 3009-3020. Fulltext not available.

Graf, Moritz, Ziegler, Christian, Gregoritza, Manuel

and Goepferich, Achim

(2019) Hydrogel microspheres evading alveolar macrophages for sustained pulmonary protein delivery. nternational Journal of Pharmaceutics 566, pp. 652-661. Fulltext not available.

Scharrenbroich, Jessica, Kaever, Volkhard, Dove, Stefan, Seifert, Roland and Schneider, Erich H. (2019) Hydrolysis of the non-canonical cyclic nucleotide cUMP by PDE9A: kinetics and binding mode. Naunyn-Schmiedeberg's Archives of Pharmacology 392 (2), pp. 199-208. Fulltext not available.

Walz, Johanna M., Wecker, Thomas

, Zhang, Pei Pei, Cakir, Bertan, Gruening, Bjoern, Agostini, Hansjuergen, Reuer, Tristan, Ludwig, Franziska, Boneva, Stefaniya

, Faerber, Lothar, Lange, Clemens, Schlunck, Guenther R. and Stahl, Andreas (2019) Impact of angiogenic activation and inhibition on miRNA profiles of human retinal endothelial cells. Experimental Eye Research 181, pp. 98-104. Fulltext not available.

Stolwijk, J. A., Skiba, M., Kade, C., Bernhardt, G., Buschauer, Armin

, Hübner, H., Gmeiner, P. and Wegener, Joachim

(2019) Increasing the throughput of label-free cell assays to study the activation of G-protein-coupled receptors by using a serial agonist exposure protocol. Integrative Biology 11 (3), pp. 99-108. Fulltext not available.

Maslanka-Figueroa, Sara, Veser, Anika, Abstiens, Kathrin, Fleischmann, Daniel and Göpferich, Achim (2019) Influenza A virus mimetic nanoparticles trigger selective cell uptake. PNAS 116 (20), pp. 9831-9836. Fulltext not available.

Gergs, U.

, Bernhardt, Günther, Buchwalow, I. B., Edler, H., Fröba, J., Keller, Max, Kirchhefer, U., Köhler, F., Mißlinger, N., Wache, H. and Neumann, J. (2019) Initial Characterization of Transgenic Mice Overexpressing Human Histamine H2 Receptors. Journal of Pharmacology and Experimental Therapeutics 369 (1), pp. 129-141. Fulltext not available.

Abstiens, Kathrin

, Maslanka Figueroa, Sara

, Gregoritza, Manuel

and Göpferich, Achim (2019) Interaction of funtionalized nanoparticles with serum proteins and its impact on colloidal stability and cargo leaching. Soft Matter 15 (4), pp. 709-720. Fulltext not available.

Bohley, Marilena, Haunberger, Alexandra and Göpferich, Achim

(2019) Intracellular availability of poorly soluble drugs from lipid nanocapsules. European Journal of Pharmaceutics and Biopharmaceutics 139, pp. 23-32. Fulltext not available.

Abstiens, Kathrin

and Göpferich, Achim (2019) Microfluidic manufacturing improves polydispersity of multicomponent polymeric nanoparticles. Journal of Drug Delivery Science and Technology 49, pp. 433-439. Fulltext not available.

Schoretsanitis, Georgios

, Haen, Ekkehard, Hiemke, Christoph, Endres, Katharina, Ridders, Florian, Veselinovic, Tanja, Gründer, Gerhard and Paulzen, Michael (2019) Pharmacokinetic correlates of venlafaxine: associated adverse reactions. European Archives of Psychiatry and Clinical Neuroscience 269 (7), pp. 851-857. Fulltext not available.

Heider, Fabian

, Ansideri, Francesco, Tesch, Roberta, Pantsar, Tatu, Haun, Urs, Döring, Eva, Kudolo, Mark, Poso, Antti

, Albrecht, Wolfgang, Laufer, Stefan A.

and Koch, Pierre (2019) Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors. European Journal of Medicinal Chemistry 175, pp. 309-329. Fulltext not available.

Nowak, Hartmuth, Weidemann, Caroline, Martini, Stefan, Oesterreicher, Zoe Anne, Dorn, Christoph, Adamzik, Michael, Kees, Frieder, Zeitlinger, Markus

and Rahmel, Tim

(2019) Repeated determination of moxifloxacin concentrations in interstitial space fluid of muscle and subcutis in septic patients. Journal of Antimicrobial Chemotherapy. Fulltext not available.

Schwindl, Sebastian, Kraus, Birgit and Heilmann, Jörg (2019) Secondary metabolites from the leaves of Juglans regia L. Biochemical Systematics and Ecology 83, pp. 130-136. Fulltext not available.

Kerres, Sabine, Plut, Eva, Malcherek, Simon, Rehbein, Julia and Reiser, Oliver

(2019) Visible Light‐Mediated Synthesis of Enantiopure γ‐Cyclobutane Amino and 3‐(Aminomethyl)‐5‐phenylpentanoic Acids. Advanced Synthesis & Catalysis 361 (6), pp. 1400-1407. Fulltext not available.

2018

Abstiens, Kathrin

, Gregoritza, Manuel

and Goepferich, Achim (2018) Ligand Density and Linker Length are Critical Factors for Multivalent Nanoparticle−Receptor Interactions. ACS Applied Materials & Interfaces 11 (1), pp. 1311-1320. Fulltext not available.

Kratzer, Alexander, Schießer, Selina, Matzneller, Peter, Wulkersdorfer, Beatrix, Zeitlinger, Markus

, Schlossmann, Jens

, Kees, Frieder

and Dorn, Christoph (2018) Determination of Total and Free Ceftolozane and Tazobactam in Human Plasma and Interstitial Fluid by HPLC-UV. Journal of Pharmaceutical and Biomedical Analysis. Fulltext not available.

Walz, Johanna Madeleine (2018) VEGF-Inhibition bei der Frühgeborenenretinopathie
- Präklinische und klinische Aspekte -. PhD, Universität Regensburg.

Böhr, Sebastian (2018) Therapeutisches Drug Monitoring der direkten oralen Antikoagulanzien. PhD, Universität Regensburg.

Dukorn, Stefanie (2018) Pharmacological tools for the NPY receptors: [³⁵S]GTPγS binding assays, luciferase gene reporter assays and labeled peptides. PhD, Universität Regensburg.

Dietrich, Peter, Kuphal, Silke, Spruss, Thilo, Hellerbrand, Claus and Bosserhoff, Anja K.

(2018) Micro RNA ‐622 is a novel mediator of tumorigenicity in melanoma by targeting Kirsten rat sarcoma. Pigment Cell & Melanoma Research 31 (5), pp. 614-629. Fulltext not available.

Walz, J. M., Bemme, S., Reichl, S., Akman, S., Breuß, H., Süsskind, D., Glitz, B., Müller, V. C., Wagenfeld, L., Gabel-Pfisterer, A., Aisenbrey, S., Engelmann, K., Koutsonas, A., Krohne, T. U. and Stahl, A.

(2018) Behandelte Frühgeborenenretinopathie in Deutschland. Der Ophthalmologe 115 (6), pp. 476-488. Fulltext not available.

Leonhardt, Michel, Sellmer, Andreas

, Krämer, Oliver H., Dove, Stefan, Elz, Sigurd, Kraus, Birgit, Beyer, Mandy and Mahboobi, Siavosh (2018) Design and biological evaluation of tetrahydro-β-carboline derivatives as highly potent histone deacetylase 6 (HDAC6) inhibitors. European Journal of Medicinal Chemistry 152, pp. 329-357. Fulltext not available.

Ridinger, Johannes, Koeneke, Emily, Kolbinger, Fiona R., Koerholz, Katharina, Mahboobi, Siavosh, Hellweg, Lars, Gunkel, Nikolas, Miller, Aubry K., Peterziel, Heike, Schmezer, Peter, Hamacher-Brady, Anne

, Witt, Olaf and Oehme, Ina (2018) Dual role of HDAC10 in lysosomal exocytosis and DNA repair promotes neuroblastoma chemoresistance. Scientific Reports 8 (1). Fulltext not available.

Gregoritza, Manuel, Abstiens, Kathrin

, Graf, Moritz and Göpferich, Achim (2018) Fabrication of antibody-loaded microgels using microfluidics and thiol-ene photoclick chemistry. European Journal of Pharmaceutics and Biopharmaceutics 127, pp. 194-203. Fulltext not available.

Dorn, Christoph, Kratzer, Alexander, Liebchen, Uwe, Schleibinger, Michael, Murschhauser, Alexandra, Schlossmann, Jens

, Kees, Frieder, Simon, Philipp and Kees, Martin G. (2018) Impact of Experimental Variables on the Protein Binding of Tigecycline in Human Plasma as Determined by Ultrafiltration. Journal of Pharmaceutical Sciences 107 (2), pp. 739-744. Fulltext not available.

Wiesneth, Stefan, Aas, Gregor, Heilmann, Jörg and Jürgenliemk, Guido (2018) Investigation of the flavan-3-ol patterns in willow species during one growing-season. Phytochemistry 145, pp. 26-39. Fulltext not available.

Sellmer, Andreas, Stangl, Hubert, Beyer, Mandy, Grünstein, Elisabeth, Leonhardt, Michel, Pongratz, Herwig, Eichhorn, Emerich, Elz, Sigurd, Striegl, Birgit, Jenei-Lanzl, Zsuzsa, Dove, Stefan, Straub, Rainer H., Krämer, Oliver H. and Mahboobi, Siavosh (2018) Marbostat-100 Defines a New Class of Potent and Selective Antiinflammatory and Antirheumatic Histone Deacetylase 6 Inhibitors. Journal of Medicinal Chemistry 61 (8), pp. 3454-3477. Fulltext not available.

Schoretsanitis, Georgios, de Leon, Jose, Haen, Ekkehard, Stegmann, Benedikt, Hiemke, Christoph, Gründer, Gerhard and Paulzen, Michael (2018) Pharmacokinetics of risperidone in different application forms – Comparing long-acting injectable and oral formulations. European Neuropsychopharmacology 28 (1), pp. 130-137. Fulltext not available.

Mathioudaki, Angeliki, Berzesta, Ariola, Kypriotakis, Zacharias, Skaltsa, Helen and Heilmann, Jörg (2018) Phenolic metabolites from Hypericum kelleri Bald., an endemic species of Crete (Greece). Phytochemistry 146, pp. 1-7. Fulltext not available.

Peña-Solórzano, Diana, Scholler, Matthias, Bernhardt, Günther, Buschauer, Armin

, König, Burkhard

and Ochoa-Puentes, Cristian (2018) Tariquidar-Related Chalcones and Ketones as ABCG2 Modulators. ACS Medicinal Chemistry Letters 9, pp. 854-859. Fulltext not available.

Dietrich, P., Kuphal, S., Spruss, T., Hellerbrand, C. and Bosserhoff, A. K.

(2018) Wild-type KRAS is a novel therapeutic target for melanoma contributing to primary and acquired resistance to BRAF inhibition. Oncogene 37 (7), pp. 897-911. Fulltext not available.

2017

Chen, Kang, Berg, Nele, Gschwind, Ruth Maria

and König, Burkhard

(2017) Selective Single C(sp3)−F Bond Cleavage in Trifluoromethylarenes: Merging Visible-Light Catalysis with Lewis Acid Activation. Journal of the American Chemical Society 139, pp. 18444-18447. Fulltext not available.

She, Xueke, Pegoli, Andrea, Mayr, Judith, Hübner, Harald, Bernhardt, Günther

, Gmeiner, Peter and Keller, Max

(2017) Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity. ACS Omega 2 (10), pp. 6741-6754.

Dukorn, Stefanie, Littmann, Timo, Keller, Max, Kuhn, Kilian K., Cabrele, Chiara

, Baumeister, Paul, Bernhardt, Günther and Buschauer, Armin (2017) Fluorescence- and radio-labeling of Lys4,Nle17,30hPP yields molecular tools for the NPY Y4 receptor. Bioconjugate Chemistry. Fulltext not available.

Noack, Katrin, Mahendrarajah, Nisintha, Hennig, Dorle, Schmidt, Luisa, Grebien, Florian

, Hildebrand, Dagmar, Christmann, Markus, Kaina, Bernd, Sellmer, Andreas, Mahboobi, Siavosh, Kubatzky, Katharina, Heinzel, Thorsten and Krämer, Oliver H. (2017) Analysis of the interplay between all-trans retinoic acid and histone deacetylase inhibitors in leukemic cells. Archives of Toxicology 91 (5), pp. 2191-2208. Fulltext not available.

Mayr, Judith, Bachl, Jürgen, Schlossmann, Jens and Díaz Díaz, David

(2017) Antimicrobial and Hemolytic Studies of a Series of Polycations Bearing Quaternary Ammonium Moieties: Structural and Topological Effects. International Journal of Molecular Sciences 18, p. 303.

Schäfer, Claudia, Göder, Anja, Beyer, Mandy, Kiweler, Nicole, Mahendrarajah, Nisintha, Rauch, Anke, Nikolova, Teodora, Stojanovic, Natasa, Wieczorek, Martin, Reich, Thomas R., Tomicic, Maja T., Linnebacher, Michael, Sonnemann, Jürgen, Dietrich, Sascha, Sellmer, Andreas, Mahboobi, Siavosh, Heinzel, Thorsten, Schneider, Günter and Krämer, Oliver H. (2017) Class I histone deacetylases regulate p53/NF-κB crosstalk in cancer cells. Cellular Signalling 29, pp. 218-225. Fulltext not available.

Wittmann, Hans-Joachim and Strasser, Andrea (2017) Competitive association binding kinetic assays: a new tool to detect two different binding orientations of a ligand to its target protein under distinct conditions? Naunyn-Schmiedeberg's Archives of Pharmacology 390 (6), pp. 595-612. Fulltext not available.

Gregoritza, Manuel

, Messmann, Viktoria, Abstiens, Kathrin, Brandl, Ferdinand and Göpferich, Achim

(2017) Controlled Antibody Release from Degradable Thermoresponsive
Hydrogels Cross-Linked by Diels−Alder Chemistry. Biomacromolecules 18, pp. 2410-2418. Fulltext not available.

Schoretsanitis, Georgios

, Haen, Ekkehard, Stegmann, Benedikt, Hiemke, Christoph, Gründer, Gerhard and Paulzen, Michael

(2017) Effect of smoking on risperidone pharmacokinetics – A multifactorial approach to better predict the influence on drug metabolism. Schizophrenia Research 185, pp. 51-57. Fulltext not available.

Mahendrarajah, Nisintha, Borisova, Marina E., Reichardt, Sigrid, Godmann, Maren, Sellmer, Andreas, Mahboobi, Siavosh, Haitel, Andrea, Schmid, Katharina, Kenner, Lukas

, Heinzel, Thorsten, Beli, Petra and Krämer, Oliver H. (2017) HSP90 is necessary for the ACK1-dependent phosphorylation of STAT1 and STAT3. Cellular Signalling 39, pp. 9-17. Fulltext not available.

Kuhn, Kilian K., Littmann, Timo, Dukorn, Stefanie, Tanaka, Miho, Keller, Max, Ozawa, Takeaki, Bernhardt, Günther and Buschauer, Armin

(2017) In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists. ACS Omega 2 (7), pp. 3616-3631.

Pegoli, Andrea

, She, Xueke, Wifling, David

, Hübner, Harald, Bernhardt, Günther, Gmeiner, Peter

and Keller, Max (2017) Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor. Journal of Medicinal Chemistry 60 (8), pp. 3314-3334. Fulltext not available.

2016

Onuoha, Mary Remigius Agatha (2016) Therapeutic Drug Monitoring of Antipsychotics - HPLC Analytical Method Development and Pharmaceutical Advices to the Ward Clinicians - For Successful Individualized Therapy. PhD, Universität Regensburg.

Lieb, Sebastian (2016) Investigations on histamine and neuropeptide Y receptors by label-free and label-dependent methods. PhD, Universität Regensburg.

Lieb, Sebastian, Littmann, Timo, Plank, Nicole, Felixberger, Johannes, Tanaka, Miho, Schäfer, Thorsten, Krief, Stéphane, Elz, Sigurd, Friedland, Kristina, Bernhardt, Günther, Wegener, Joachim, Ozawa, Takeaki and Buschauer, Armin (2016) Label-free versus conventional cellular assays: functional investigations on the human histamine H1 receptor. Pharmacological Research 114, pp. 13-26. Fulltext not available.

Töpper, Christoph, Steinbach, Cathérine Louise, Dorn, Christoph

, Kratzer, Alexander, Wicha, Sebastian G., Schleibinger, Michael, Liebchen, Uwe, Kees, Frieder, Salzberger, Bernd and Kees, Martin G. (2016) Variable linezolid exposure in ICU patients—possible role of drug-drug interactions. Therapeutic Drug Monitoring 38 (5), pp. 573-578. Fulltext not available.

Kunath, Julia (2016) Designermoleküle hemmen die Semaphorin 3F Wirkung in vitro, haben aber keinen Einfluss auf den Verlauf der experimentellen Arthritis. PhD, Universität Regensburg.

Schlossmann, Jens, Wetzl, Veronika, Schinner, Elisabeth, Kees, Frieder K., Hofmann, Franz and Faerber, Lothar

(2016) Involvement of cyclic guanosine monophosphate-dependent protein kinase I in renal antifibrotic effects of serelaxin. Frontiers in Pharmacology 7 (195), pp. 1-27.

Hennig, Robert (2016) Multivalent nanoparticles for the treatment of ocular diseases. PhD, Universität Regensburg.

Kuhn, Kilian K., Ertl, Thomas, Dukorn, Stefanie, Keller, Max, Bernhardt, Günther, Reiser, Oliver

and Buschauer, Armin (2016) High affinity agonists of the neuropeptide Y (NPY) Y4 receptor derived from the C-terminal pentapeptide of human pancreatic polypeptide (hPP): synthesis, stereochemical discrimination and radiolabeling. Journal of Medicinal Chemistry 59 (13), pp. 6045-6058. Fulltext not available.

Limmer, Franziska (2016) Funktionelle Analyse der cGMP-abhängigen Proteinkinase I in der Niere, insbesondere im dicken aufsteigenden Ast der Henle-Schleife. PhD, Universität Regensburg.

Stangl, Hubert Werner (2016) Arthritis and cholinergic transition of sympathetic nerve fibers. PhD, Universität Regensburg.

Vögeler, Jessica (2016) Pharmakotherapie und Humanpharmakologische Untersuchungen bei Patienten mit DME (Diabetisches Makulaödem) und PDR (Proliferative Diabetische Retinopathie) anhand klinischer Parameter und inflammatorischer Biomarker. PhD, Universität Regensburg.

Lorenz, Peter, Knittel, Diana N., Conrad, Jürgen, Lotter, Eva M., Heilmann, Jörg, Stintzing, Florian C. and Kammerer, Dietmar R. (2016) 1-Acetyl-3-[(3R)-hydroxyfatty acyl]glycerols: Lipid Compounds fromEuphrasia rostkovianaHayneandE. tetraquetra(Bréb.)Arrond. Chemistry & Biodiversity 13 (5), pp. 602-612. Fulltext not available.

Hammer, Sebastian, Gobleder, Susanne, Naporra, Franziska, Wittmann, Hans-Joachim, Elz, Sigurd, Heinrich, Markus

and Strasser, Andrea (2016) 2,4-Diaminopyrimidines as dual ligands at the histamine H1 and H4 receptor - H1/H4-receptor selectivity. Bioorganic & Medicinal Chemistry Letters 26, pp. 292-300. Fulltext not available.

Hennig, Robert, Kuespert, Sabrina, Haunberger, Alexandra, Goepferich, Achim

and Fuchshofer, Rudolf (2016) Cyclic RGD peptides target human trabecular meshwork cells while ameliorating connective tissue growth factor-induced fibrosis. Journal of Drug Targeting 24 (10), pp. 952-959. Fulltext not available.

Gregoritza, Manuel, Messmann, Viktoria, Goepferich, Achim M.

and Brandl, Ferdinand P. (2016) Design of hydrogels for delayed antibody release utilizing hydrophobic association and Diels–Alder chemistry in tandem. Journal of Materials Chemistry B 4 (19), pp. 3398-3408. Fulltext not available.

Sawatzky, Edgar, Wehle, Sarah, Kling, Beata, Wendrich, Jan, Bringmann, Gerhard, Sotriffer, Christoph A., Heilmann, Jörg and Decker, Michael (2016) Discovery of Highly Selective and Nanomolar Carbamate-Based Butyrylcholinesterase Inhibitors by Rational Investigation into Their Inhibition Mode. Journal of Medicinal Chemistry 59 (5), pp. 2067-2082. Fulltext not available.

Keller, Max, Kuhn, Kilian K., Einsiedel, Jürgen, Hübner, Harald, Biselli, Sabrina, Mollereau, Catherine

, Wifling, David, Svobodova, Jaroslava, Bernhardt, Günther, Cabrele, Chiara

, Vanderheyden, Patrick, Gmeiner, Peter

and Buschauer, Armin (2016) Mimicking of arginine by functionalized Nω-carbamoylated arginine as a new broadly applicable approach to labeled bioactive peptides: high affinity angiotensin, neuropeptide Y, neuropeptide FF and neurotensin receptor ligands as examples. Journal of Medicinal Chemistry 59 (5), pp. 1925-1945. Fulltext not available.

Khan, Nadia, Saad, Ali, Nurulain, Syed M., Darras, Fouad H., Decker, Michael and Sadek, Bassem (2016) The dual-acting H3 receptor antagonist and AChE inhibitor UW-MD-71 dose-dependently enhances memory retrieval and reverses dizocilpine-induced memory impairment in rats. Behavioural Brain Research 297, pp. 155-164. Fulltext not available.

Huang, Guozheng

, Schramm, Simon, Heilmann, Jörg, Biedermann, David, Křen, Vladimír and Decker, Michael (2016) Unconventional application of the Mitsunobu reaction: Selective flavonolignan dehydration yielding hydnocarpins. Beilstein Journal of Organic Chemistry 12, pp. 662-669. Fulltext not available.

2015

Rothenhöfer, Martin, Grundmann, Marco, Bernhardt, Günther, Matysik, Frank-Michael and Buschauer, Armin (2015) High performance anion exchange chromatography with pulsed amperometric detection (HPAEC–PAD) for the sensitive determination of hyaluronan oligosaccharides. Journal of Chromatography B 988 (C), pp. 106-115. Fulltext not available.

Mahli, Abdo (2015) Novel in vitro model for combined effects of alcohol and free fatty acids on hepatocellular lipid accumulation and inflammation. PhD, Universität Regensburg.

Dolles, Dominik, Nimczick, Martin, Scheiner, Matthias, Ramler, Jacqueline, Stadtmüller, Patricia, Sawatzky, Edgar, Drakopoulos, Antonios

, Sotriffer, Christoph, Wittmann, Hans-Joachim, Strasser, Andrea and Decker, Michael (2015) Aminobenzimidazoles and Structural Isomers as Templates for Dual-Acting Butyrylcholinesterase Inhibitors andhCB2R Ligands To Combat Neurodegenerative Disorders. ChemMedChem 11 (12), pp. 1270-1283. Fulltext not available.

Jenei-Lanzl, Zsuzsa, Capellino, Silvia

, Kees, Frieder, Fleck, Martin, Lowin, Torsten and Straub, Rainer H.

(2015) Anti-inflammatory effects of cell-based therapy with tyrosine hydroxylase-positive catecholaminergic cells in experimental arthritis. Annals of the Rheumatic Diseases 74, pp. 444-451.

Lübker, Carolin, Dove, Stefan, Tang, Wei-Jen

, Bieber Urbauer, Ramona J., Moskovitz, Jackob, Urbauer, Jeffrey L. and Seifert, Roland (2015) Different Roles of N-Terminal and C-Terminal Domains in Calmodulin for Activation of Bacillus anthracis Edema Factor. Toxins 7 (7), pp. 2598-2614.

Beermann, Silke, Bernhardt, Guenther, Seifert, Roland, Buschauer, Armin and Neumann, Detlef

(2015) Histamine H1- and H4-receptor signaling cooperatively regulate MAPK activation. Biochemical Pharmacology 98 (3), pp. 432-439. Fulltext not available.

Radons, Jürgen, Falk, Werner and Dove, Stefan (2015) Identification of critical regions within the TIR domain of IL-1 receptor type I. The international journal of biochemistry & cell biology 68, pp. 15-20. Fulltext not available.

Zenger, Katharina, Dutta, Subhajit, Wolff, Horst, Genton, Marc G.

and Kraus, Birgit (2015) In vitro structure-toxicity relationship of chalcones in human hepatic stellate cells. Toxicology 336, pp. 26-33. Fulltext not available.

Lübker, Carolin, Bieber-Urbauer, Ramona J., Moskovitz, Jackob, Dove, Stefan, Weisemann, Jasmin

, Fedorova, Maria, Urbauer, Jeffrey L. and Seifert, Roland (2015) Membranous adenylyl cyclase 1 activation is regulated by oxidation of N- and C-terminal methionine residues in calmodulin. Biochemical Pharmacology 93 (2), pp. 196-209. Fulltext not available.

Wifling, David

, Löffel, Karolin, Nordemann, Uwe, Strasser, Andrea, Bernhardt, Günther, Dove, Stefan, Seifert, Roland and Buschauer, Armin (2015) Molecular determinants for the high constitutive activity of the human histamine H4 receptor: Functional studies on orthologs and mutants. British Journal of Pharmacology 172, pp. 785-798. Fulltext not available.

Keller, Max, Weiss, Stefan, Hutzler, Christoph

, Kuhn, Kilian K., Mollereau, Catherine

, Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Günther, König, Burkhard and Buschauer, Armin (2015) N(omega)-carbamoylation of the argininamide moiety: an avenue to insurmountable NPY Y1 receptor antagonists and a radiolabeled selective high affinity molecular tool ([3H]UR-MK299) with extended residence time. Journal of Medicinal Chemistry 58 (22), pp. 8834-8849. Fulltext not available.

Kirchhof, Susanne, Strasser, Andrea, Wittmann, Hans-Joachim, Messmann, Viktoria, Hammer, Nadine, Goepferich, Achim M.

and Brandl, Ferdinand P. (2015) New insights into the cross-linking and degradation mechanism of Diels–Alder hydrogels. Journal of Materials Chemistry B 3 (3), pp. 449-457. Fulltext not available.

Chen, Xinyu, Klöckner, Jessika, Holze, Janine, Zimmermann, Cornelia, Seemann, Wiebke K., Schrage, Ramona, Bock, Andreas

, Mohr, Klaus, Tränkle, Christian, Holzgrabe, Ulrike

and Decker, Michael (2015) Rational Design of Partial Agonists for the Muscarinic M1 Acetylcholine Receptor. Journal of Medicinal Chemistry 58 (2), pp. 560-576. Fulltext not available.

2014

Cuboni, Serena, Devigny, Christian, Hoogeland, Bastiaan, Strasser, Andrea, Pomplun, Sebastian, Hauger, Barbara, Höfner, Georg, Wanner, Klaus, Eder, Matthias

, Buschauer, Armin, Holsboer, Florian and Hausch, Felix (2014) Loratadine and analogs: Discovery and preliminary SAR of inhibitors of the amino acid transporter B0AT2. Journal of Medicinal Chemistry 57 (22), pp. 9473-9479. Fulltext not available.

Thiele, Karinna Marie (2014) Charakterisierung Gαi3-gendefizienter Mauslinien. PhD, Universität Regensburg.

Darras, Fouad H., Wehle, Sarah, Huang, Guozheng

, Sotriffer, Christoph A. and Decker, Michael (2014) Amine substitution of quinazolinones leads to selective nanomolar AChE inhibitors with ‘inverted’ binding mode. Bioorganic & Medicinal Chemistry 22 (17), pp. 4867-4881. Fulltext not available.

Kremb, Stephan, Helfer, Markus, Kraus, Birgit, make_name_string expected hash reference, make_name_string expected hash reference, make_name_string expected hash reference, make_name_string expected hash reference

and make_name_string expected hash reference

(2014) Aqueous Extracts of the Marine Brown Alga Lobophora variegata Inhibit HIV-1 Infection at the Level of Virus Entry into Cells. PloS ONE 9, e103895.

Pollinger, Klaus, Hennig, Robert, Bauer, Stefanie, Breunig, Miriam, Tessmar, Joerg

, Buschauer, Armin, Witzgall, Ralph

and Göpferich, Achim

(2014) Biodistribution of quantum dots in the kidney after intravenous injection. Journal of Nanoscience and Nanotechnology 14 (5), pp. 3313-3319. Fulltext not available.

Darras, Fouad H., Kling, Beata, Sawatzky, Edgar, Heilmann, Jörg and Decker, Michael (2014) Cyclic acyl guanidines bearing carbamate moieties allow potent and dirigible cholinesterase inhibition of either acetyl- or butyrylcholinesterase. Bioorganic & Medicinal Chemistry 22 (17), pp. 5020-5034. Fulltext not available.

Kratzer, Alexander, Liebchen, Uwe, Schleibinger, Michael, Kees, Martin G. and Kees, Frieder (2014) Determination of free vancomycin, ceftriaxone, cefazolin and ertapenem in plasma by ultrafiltration: Impact of experimental conditions. Journal of Chromatography B 961, pp. 97-102. Fulltext not available.

2013

Brandl, Katharina (2013) Erratum: Untersuchungen zur pharmakologischen Beeinflussung der Toll-like Rezeptoren in der Sepsis.

Kees, Martin Georg, Schaeftlein, André, Haeberle, Helene Anna, Kees, Frieder K., Kloft, Charlotte and Heininger, Alexandra (2013) Population pharmacokinetics and pharmacodynamic evaluation of intravenous and enteral moxifloxacin in surgical intensive care unit patients. The Journal of antimicrobial chemotherapy. Fulltext not available.

Knuth, Susanne, Abdelsalam, Rania, Khayyal, Mohamed, Schweda, Frank, Heilmann, Jörg, Kees, Martin, Mair, Georg, Kees, Frieder and Jürgenliemk, Guido (2013) Catechol Conjugates Are In Vivo Metabolites of Salicis cortex. Planta Medica 79 (16), pp. 1489-1494. Fulltext not available.

Miller, Tobias, van Colen, G., Sander, B., Golas, M., Uezguen, Senta, Weigandt, Markus and Goepferich, Achim

(2013) Drug Loading of Polymerics Micelles. Pharmaceutical Research 30 (2), pp. 484-595. Fulltext not available.

Zenger, Katharina, Chen, Xinyu, Decker, Michael and Kraus, Birgit (2013) In-vitro stability and metabolism of a tacrine–silibinin codrug. Journal of Pharmacy and Pharmacology 65 (12), pp. 1765-1772. Fulltext not available.

Kirchhof, Susanne, Brandl, Ferdinand P., Hammer, Nadine and Goepferich, Achim M.

(2013) Investigation of the Diels–Alder reaction as a cross-linking mechanism for degradable poly(ethylene glycol) based hydrogels. Journal of Materials Chemistry B 1 (37), p. 4855. Fulltext not available.

Schweizer, Daniel, Vostiar, Igor, Heier, Annabelle, Serno, Tim, Schoenhammer, Karin, Jahn, Michael, Jones, Stewart, Piequet, Aline, Beerli, Christian, Gram, Hermann and Goepferich, Achim

(2013) Pharmacokinetics, biocompatibility and bioavailability of a controlled release monoclonal antibody formulation. Journal of Controlled Release 172 (3), pp. 975-982. Fulltext not available.

Miller, Tobias, Breyer, S., van Colen, G., Mier, W., Haberkorn, U., Geissler, S., Voss, S., Weigandt, Markus and Goepferich, Achim

(2013) Premature drug release of polymeric micelles and its effects on tumor targeting. International Journal of Pharmaceutics 445 (1-2), pp. 117-124. Fulltext not available.

Schweizer, Daniel, Schoenhammer, K., Jahn, M. and Goepferich, Achim

(2013) Protein-Polyanion Interactions for the Controlled Release of Monoclonal Antibodies. Biomacromolecules 14 (1), pp. 75-83. Fulltext not available.

Würtenberger, Irene, Angermaier, Bernhard, Kircher, Brigitte and Gust, Ronald (2013) Synthesis and In Vitro Pharmacological Behavior of Platinum(II) Complexes Containing 1,2-Diamino-1-(4-fluorophenyl)-2-alkanol Ligands. Journal of Medicinal Chemistry 56 (20), pp. 7951-7964. Fulltext not available.

Dorn, Christoph

, Massinger, Sabine, Wuzik, Andreas, Heilmann, Jörg and Hellerbrand, Claus (2013) Xanthohumol suppresses inflammatory response to warm ischemia–reperfusion induced liver injury. Experimental and Molecular Pathology 94 (1), pp. 10-16. Fulltext not available.

2012

Memminger, Martin, Keller, Max, Lopuch, Miroslaw, Pop, Nathalie, Bernhardt, Günther, von Angerer, Erwin and Buschauer, Armin (2012) The Neuropeptide Y Y1 receptor: a diagnostic marker? Expression in MCF-7 breast cancer cells is down-regulated by antiestrogens in vitro and in xenografts. PLoS ONE 7 (12), e51032.

Rothenhöfer, Martin, Scherübl, Rosmarie, Bernhardt, Günther, Heilmann, Jörg and Buschauer, Armin (2012) Qualitative and quantitative analysis of hyaluronan oligosaccharides with high performance thin layer chromatography using reagent-free derivatization on amino-modified silica and electrospray ionization-quadrupole time-of-flight mass spectrometry coupling on normal phase. Journal of chromatography. A 1248, pp. 169-77. Fulltext not available.

Bubik, Martin F., Willer, Elisabeth A., Bihari, Peter, Jürgenliemk, Guido, Ammer, Hermann

, Krombach, Fritz, Zahler, Stefan, Vollmar, Angelika M. and Fürst, Robert (2012) A novel approach to prevent endothelial hyperpermeability: The Crataegus extract WS® 1442 targets the cAMP/Rap1 pathway. Journal of Molecular and Cellular Cardiology 52 (1), pp. 196-205. Fulltext not available.

Freischmidt, A., Jürgenliemk, G., Kraus, B., Okpanyi, S.N., Müller, J., Kelber, O.

, Weiser, D. and Heilmann, J. (2012) Contribution of flavonoids and catechol to the reduction of ICAM-1 expression in endothelial cells by a standardised Willow bark extract. Phytomedicine 19 (3-4), pp. 245-252. Fulltext not available.

Vo, Hau T., Nguyen, Ngoc-Tuyet T., Nguyen, Hieu T., Do, Khoa Q.

, Connolly, Joseph D., Maas, Gerhard, Heilmann, Jörg, Werz, Udo R., Pham, Hung D. and Nguyen, Lien-Hoa D. (2012) Cytotoxic tetraoxygenated xanthones from the bark of Garcinia schomburgkiana. Phytochemistry Letters 5 (3), pp. 553-557. Fulltext not available.

Reher, Till M., Brunskole, Irena, Neumann, Detlef

and Seifert, Roland (2012) Evidence for ligand-specific conformations of the histamine H2-receptor in human eosinophils and neutrophils. Biochemical Pharmacology 84 (9), pp. 1174-1185. Fulltext not available.

Grundmann, Marco, Rothenhöfer, M., Bernhardt, Günther, Buschauer, Armin and Matysik, Frank-Michael (2012) Fast counter-electroosmotic capillary electrophoresis-time-of-flight mass spectrometry of hyaluronan oligosaccharides. Analytical and Bioanalytical Chemistry : Anal. Bioanal. Chem. 402, pp. 2617-2623. Fulltext not available.

Posavec, Damir, Zabel, Manfred, Bogner, Udo, Bernhardt, Günther and Knör, Günther (2012) Functionalized derivatives of 1,4-dimethylnaphthalene as precursors for biomedical applications: synthesis, structures, spectroscopy and photochemical activation in the presence of dioxygen. Organic & biomolecular chemistry 10 (35), pp. 7062-7069.

Zayed, Gamal M. S.

and Tessmar, Joerg K. V.

(2012) Heterobifunctional Poly(ethylene glycol) Derivatives for the Surface Modification of Gold Nanoparticles Toward Bone Mineral Targeting. Macromolecular Bioscience 12 (8), pp. 1124-1136. Fulltext not available.

Saugspier, Michael, Dorn, Christoph

, Czech, Barbara, Gehrig, Manfred, Heilmann, Jörg and Hellerbrand, Claus

(2012) Hop bitter acids inhibit tumorigenicity of hepatocellular carcinoma cells in vitro. Oncology Reports 28 (4), pp. 1423-1428. Fulltext not available.

Appl, Heidrun, Holzammer, Tobias, Dove, Stefan, Haen, Ekkehard, Strasser, Andrea and Seifert, Roland (2012) Interactions of recombinant human histamine H₁R, H₂R, H₃R, and H₄R receptors with 34 antidepressants and antipsychotics. Naunyn-Schmiedeberg's archives of pharmacology 385 (2), pp. 145-170. Fulltext not available.

Pollinger, Klaus, Hennig, Robert, Breunig, Miriam

, Teßmar, Jörg

, Ohlmann, Andreas

, Tamm, Ernst R.

, Witzgall, Ralph

and Goepferich, Achim

(2012) Kidney Podocytes as Specific Targets for cyclo(RGDfC)-Modified Nanoparticles. Small 8, pp. 3368-3375. Fulltext not available.

Elbakry, Asmaa Mohamed, Wurster, Eva-Christina, Zaky, Alaa, Liebl, Renate, Schindler, Edith, Bauer-Kreisel, Petra, Blunk, Torsten, Rachel, Reinhard, Goepferich, Achim

and Breunig, Miriam

(2012) Layer-by-Layer Coated Gold Nanoparticles: Size-Dependent Delivery of DNA into Cells. Small 8 (24), pp. 3847-3856. Fulltext not available.

Decker, Michael and Holzgrabe, Ulrike

(2012) M1 muscarinic cetylcholine receptor allosteric modulators as potential therapeutic opportunities for treating Alzheimer's disease. MedChemComm 3 (7), p. 752. Fulltext not available.

Darras, Fouad H., Kling, Beata, Heilmann, Jörg and Decker, Michael (2012) Neuroprotective Tri- and Tetracyclic BChE Inhibitors Releasing Reversible Inhibitors upon Carbamate Transfer. ACS Medicinal Chemistry Letters 3 (11), pp. 914-919. Fulltext not available.

Schmidt, Sebastian, Jürgenliemk, Guido, Skaltsa, Helen and Heilmann, Jörg (2012) Phloroglucinol derivatives from Hypericum empetrifolium with antiproliferative activity on endothelial cells. Phytochemistry 77, pp. 218-225. Fulltext not available.

Nguyen, Le-Thu T., Nguyen, Hieu T., Barbič, Matej, Brunner, Gabi, Heilmann, Jörg, Pham, Hung D., Nguyen, Duc M. and Nguyen, Lien-Hoa D. (2012) Polyisoprenylated acylphloroglucinols and a polyisoprenylated tetracyclic xanthone from the bark of Calophyllum thorelii. Tetrahedron Letters 53 (34), pp. 4487-4493. Fulltext not available.

Ulrich-Merzenich, G., Koptina, A.

, Kelber, O.

, Freischmidt, A., Heilmann, J., Müller, J., Sadeghlar, F., Zeitler, H. and Wagner, H. (2012) Prediction of adverse events by in vivo gene expression profiling exemplified for phytopharmaceuticals containing salicylates and the antidepressant imipramine. Phytomedicine 19 (3-4), pp. 322-329. Fulltext not available.

Wagner, Eva (2012) Synthese und pharmakologische Charakterisierung dualer Histamin-H1-/H4-Rezeptorliganden. PhD, Universität Regensburg.

Schmidt, Jennifer, Riechers, Alexander, Stoll, Raphael, Amann, Thomas, Fink, Florian, Spruss, Thilo, Gronwald, Wolfram, König, Burkhard

, Hellerbrand, Claus and Bosserhoff, Anja Katrin

(2012) Targeting melanoma metastasis and immunosuppression with a new mode of melanoma inhibitory activity (MIA) protein inhibition. PloS ONE 7 (5), e37941.

Jaumann, Mirko, Dettling, Juliane, Gubelt, Martin, Zimmermann, Ulrike, Gerling, Andrea, Paquet-Durand, François

, Feil, Susanne

, Wolpert, Stephan, Franz, Christoph, Varakina, Ksenya, Xiong, Hao, Brandt, Niels, Kuhn, Stephanie, Geisler, Hyun-Soon, Rohbock, Karin, Ruth, Peter, Schlossmann, Jens

, Hütter, Joachim, Sandner, Peter, Feil, Robert

, Engel, Jutta, Knipper, Marlies and Rüttiger, Lukas (2012) cGMP-Prkg1 signaling and Pde5 inhibition shelter cochlear hair cells and hearing function. Nature Medicine 18 (2), pp. 252-259. Fulltext not available.

2011

Pop, Nathalie, Igel, Patrick, Brennauer, Albert, Cabrele, Chiara

, Bernhardt, Günther, Seifert, Roland and Buschauer, Armin (2011) Functional reconstitution of human neuropeptide Y (NPY) Y2 and Y4 receptors in Sf9 insect cells. Journal of Receptors and Signal Transduction 31 (4), pp. 271-285. Fulltext not available.

Schaedlich, A., Rose, C., Kuntsche, J., Caysa, H., Mueller, T., Goepferich, Achim

and Maeder, K. (2011) How Stealthy are PEG-PLA Nanoparticles? An NIR In Vivo Study Combined with Detailed Size Measurements. Pharmaceutical Research 28 (8), pp. 1995-2007. Fulltext not available.

Decker, M. (2011) Hybrid Molecules Incorporating Natural Products: Applications in Cancer Therapy, Neurodegenerative Disorders and Beyond. Current Medicinal Chemistry 18 (10), pp. 1464-1475. Fulltext not available.

Sutor, Sarah, Heilmann, Jörg and Seifert, Roland (2011) Impact of fusion to Gαi2 and co-expression with RGS proteins on pharmacological properties of human cannabinoid receptors CB1R and CB2R. Journal of Pharmacy and Pharmacology 63 (8), pp. 1043-1055. Fulltext not available.

Wittmann, Hans-Joachim, Seifert, Roland and Strasser, Andrea (2011) Influence of the N-terminus and the E2-loop onto the binding kinetics of the antagonist mepyramine and the partial agonist phenoprodifen to H1R. Biochemical Pharmacology 12, pp. 1910-1918. Fulltext not available.

Chen, Xinyu, Tikhonova, Irina G. and Decker, Michael (2011) Probing the mid-gorge of cholinesterases with spacer-modified bivalent quinazolinimines leads to highly potent and selective butyrylcholinesterase inhibitors. Bioorganic & Medicinal Chemistry 19 (3), pp. 1222-1235. Fulltext not available.

Mannschreck, Albrecht and von Angerer, Erwin (2011) The Scent of Roses and Beyond: Molecular Structures, Analysis, and Practical Applications of Odorants. Journal of Chemical Education 88 (11), pp. 1501-1506. Fulltext not available.

2010

Dayoub, Rania

, Wagner, Hannah, Bataille, Frauke, Stöltzing, Oliver, Spruss, Thilo, Buechler, Christa, Schlitt, Hans-Jürgen and Weiss, Thomas S.

(2010) Liver Regeneration Associated Protein (ALR) Exhibits Antimetastatic Potential in Hepatocellular Carcinoma. Molecular Medicine 17, pp. 221-228.

Modrow, Susanne, Wenzel, J. J.

, Schimanski, S., Schwarzbeck, J., Rothe, U., Oldenburg, J., Jilg, W. and Eis-Hübinger, A. M. (2010) Prevalence of nucleic acid sequences specific for human parvoviruses, hepatitis A and hepatitis E viruses in coagulation factor concentrates. Vox sanguinis. Fulltext restricted.

Amann, Thomas, Bataille, Frauke, Spruss, Thilo, Dettmer, Katja

, Wild, Peter J., Liedtke, Christian

, Mühlbauer, Marcus, Kiefer, Paul, Oefner, Peter J.

, Trautwein, Christian, Bosserhoff, Anja-Katrin

and Hellerbrand, Claus (2010) Reduced expression of fibroblast growth factor receptor 2IIIb in hepatocellular carcinoma induces a more aggressive growth. The American journal of pathology 176 (3), pp. 1433-42. Fulltext not available.

Barbic, M, Willer, E, Fürst, R and Jürgenliemk, G (2010) Aesculin from Butcher's broom reduces the permeability of endothelial cells in vitro. Planta Medica 76 (12). Fulltext not available.

Fürst, R, Bubik, M, Bihari, P, Jürgenliemk, G, Ammer, H, Krombach, F, Zahler, S and Vollmar, A (2010) The hawthorn special extract WS® 1442 protects against endothelial barrier dysfunction – elucidation of the underlying molecular mechanisms. Planta Medica 76 (12). Fulltext not available.

2009

Silva, Maria Elena (2009) Theoretical study of the interaction of agonists with the 5-HT2A receptor. PhD, Universität Regensburg.

Sander, Kerstin, Kottke, Tim, Tanrikulu, Yusuf, Proschak, Ewgenij, Weizel, Lilia, Schneider, Erich H.

, Seifert, Roland, Schneider, Gisbert

and Stark, Holger

(2009) 2,4-Diaminopyrimidines as histamine H4 receptor ligands—Scaffold optimization and pharmacological characterization. Bioorganic & Medicinal Chemistry 17 (20), pp. 7186-7196. Fulltext not available.

Amann, Thomas, Bataille, Frauke, Spruss, Thilo, Mühlbauer, Marcus, Gäbele, Erwin, Schölmerich, Jürgen, Kiefer, Paul, Bosserhoff, Anja‐Katrin

and Hellerbrand, Claus (2009) Activated hepatic stellate cells promote tumorigenicity of hepatocellular carcinoma. Cancer Science 100 (4), pp. 646-653. Fulltext not available.

Weiser, Barbara, Sommer, Florian, Neubauer, M., Seitz, Anna Katharina, Teßmar, Jörg

, Göpferich, Achim

and Blunk, Torsten (2009) Ascorbic Acid Enhances Adipogenesis of Bone Marrow-Derived Mesenchymal Stromal Cells. Cells Tissues Organs 189 (6), pp. 373-381. Fulltext not available.

Göttle, Martin, Geduhn, Jens, König, Burkhard

, Gille, Andreas

, Höcherl, Klaus and Seifert, Roland (2009) Characterization of Mouse Heart Adenylyl Cyclase. Journal of Pharmacology and Experimental Therapeutics 329 (3), pp. 1156-1165. Fulltext not available.

Mahboobi, Siavosh, Dove, Stefan, Sellmer, Andreas, Winkler, Matthias, Eichhorn, Emerich, Pongratz, Herwig, Ciossek, Thomas, Baer, Thomas, Maier, Thomas and Beckers, Thomas (2009) Design of chimeric histone deacetylase- and tyrosine kinase-inhibitors: a series of imatinib hybrides as potent inhibitors of wild-type and mutant BCR-ABL, PDGF-Rbeta, and histone deacetylases. Journal of medicinal chemistry 52 (8), pp. 2265-79. Fulltext not available.

Massoumi, Ramin, Kuphal, Silke, Hellerbrand, Claus, Haas, Bodo

, Wild, Peter, Spruss, Thilo, Pfeifer, Alexander, Fässler, Reinhard and Bosserhoff, Anja K.

(2009) Down-regulation of CYLD expression by Snail promotes tumor progression in malignant melanoma. Journal of Experimental Medicine 206 (1), pp. 221-232. Fulltext not available.

Egger, Michael, Maity, Prantik, Hübner, Melanie, Seifert, Roland and König, Burkhard

(2009) Synthesis and pharmacological properties of new tetracyclic forskolin analogues. European Journal of Organic Chemistry 2009 (21), pp. 3613-3618. Fulltext not available.

2008

Weiss, Stefan, Keller, Max, Bernhardt, Günther, Buschauer, Armin and König, Burkhard

(2008) Modular synthesis of non-peptidic bivalent NPY Y(1) receptor antagonists. Bioorganic & Medicinal Chemistry 16 (22), pp. 9858-9866. Fulltext not available.

Strasser, Andrea, Striegl, Birgit, Wittmann, Hans-Joachim and Seifert, Roland (2008) Pharmacological Profile of Histaprodifens at Four Recombinant Histamine H1 Receptor Species Isoforms. Journal of Pharmacology and Experimental Therapeutics 324, pp. 60-71. Fulltext not available.

Vogel, Susanne, Kaufmann, Doris, Pojarová, Michaela, Müller, Christine, Pfaller, Tobias, Kühne, Sybille, Bednarski, Patrick J. and Angerer, Erwin von (2008) Aroyl hydrazones of 2-phenylindole-3-carbaldehydes as novel antimitotic agents. Bioorganic & Medicinal Chemistry 16 (12), pp. 6436-6447. Fulltext not available.

Kutta, Roger J., Hofinger, Edith S. A., Preuss, Hendrik, Bernhardt, Günther and Dick, Bernhard

(2008) Blue-light induced interaction of LOV domains from Chlamydomonas reinhardtii. Chembiochem : a European journal of chemical biology 9 (12), pp. 1931-1938. Fulltext not available.

Sommer, Florian, Pollinger, Klaus, Brandl, Ferdinand, Weiser, Barbara, Teßmar, Jörg

, Blunk, Torsten and Göpferich, Achim

(2008) Hyalocyte proliferation and ECM accumulation modulated by bFGF and TGF-β1. Graefe's Archive for Clinical and Experimental Ophthalmology 246 (9), pp. 1275-1284. Fulltext not available.

Weiser, Barbara, Prantl, Lukas, Schubert, Thomas E. O., Zellner, J.

, Fischbach-Teschl, Claudia, Spruss, Thilo, Seitz, Anna Katharina, Teßmar, Jörg

, Göpferich, Achim

and Blunk, Torsten (2008) In Vivo Development and Long-Term Survival of Engineered Adipose Tissue Depend on In Vitro Precultivation Strategy. Tissue Engineering Part A 14 (2), pp. 275-284. Fulltext not available.

Langgartner, Julia, Vasold, Antje, Glück, Thomas, Reng, Michel and Kees, Frieder (2008) Pharmacokinetics of meropenem during intermittent and continuous intravenous application in patients treated by continuous renal replacement therapy. Intensive Care Medicine 34 (6), pp. 1091-1096. Fulltext not available.

Egger, M., Pellett, P., Nickl, K., Geiger, S., Graetz, S., Seifert, R., Heilmann, J. and König, B.

(2008) Synthesis and Cannabinoid Receptor Activity of Ketoalkenes from Echinacea pallida and Non-natural Analogues. Chem. Eur. J. 14, 10978 - 10984. Fulltext not available.

Hellerbrand, C, Amann, T, Schlegel, J, Wild, P, Bataille, F, Spruss, T, Hartmann, A and Bosserhoff, A-K

(2008) The novel gene MIA2 acts as a tumour suppressor in hepatocellular carcinoma. Gut 57 (2), pp. 243-251. Fulltext not available.

2007

Matzdorf, Corina (2007) Untersuchungen zur Rolle von Cyclooxygenase-2-gebildeten Prostaglandinen für die Bildung und Freisetzung von Renin. PhD, Universität Regensburg.

Göttle, Martin, Dove, Stefan, Steindel, Phillip, Shen, Yuequan, Tang, Wei-Jen

, Geduhn, Jens, König, Burkhard

and Seifert, Roland (2007) Molecular Analysis of the Interaction of Bordetella pertussis Adenylyl Cyclase with Fluorescent Nucleotides. Molecular Pharmacology 72 (3), pp. 526-535.

Kaufmann, Doris, Pojarová, Michaela, Vogel, Susanne, Liebl, Renate, Gastpar, Robert, Gross, Dietmar, Nishino, Tsuyuki, Pfaller, Tobias and Angerer, Erwin von (2007) Antimitotic activities of 2-phenylindole-3-carbaldehydes in human breast cancer cells. Bioorganic & medicinal chemistry 15 (15), pp. 5122-36. Fulltext not available.

Matzdorf, Corina, Kurtz, A. and Höcherl, Klaus (2007) COX-2 activity determines the level of renin expression but is dispensable for acute upregulation of renin expression in rat kidneys. American Journal of Physiology-Renal Physiology 292 (6), F1782-F1790. Fulltext not available.

Koeber, R, Bader, W, Jahner, T, Melchner, D and Haen, E (2007) Determination of rivastigmine in serum using solid phase extraction and high perfomance liquid chromatography coupled to UV detection technique for routine medical analysis. Pharmacopsychiatry 40 (05). Fulltext not available.

Rothhammer, T, Bataille, F, Spruss, T, Eissner, G and Bosserhoff, A-K

(2007) Functional implication of BMP4 expression on angiogenesis in malignant melanoma. Oncogene 26 (28), pp. 4158-4170. Fulltext not available.

Bergmann, Antje, Teßmar, Jörg

and Owen, Anthony (2007) Influence of electron irradiation on the crystallisation, molecular weight and mechanical properties of poly-(R)-3-hydroxybutyrate. Journal of Materials Science 42 (11), pp. 3732-3738. Fulltext not available.

Zoriy, Myroslav, Matusch, Andreas, Spruss, Thilo and Becker, J. Sabine (2007) Laser ablation inductively coupled plasma mass spectrometry for imaging of copper, zinc, and platinum in thin sections of a kidney from a mouse treated with cis-platin. International Journal of Mass Spectrometry 260 (2-3), pp. 102-106. Fulltext not available.

Murphy, Matthew B., Hartgerink, Jeffrey D.

, Goepferich, Achim

and Mikos, Antonios G. (2007) Synthesis and in Vitro Hydroxyapatite Binding of Peptides Conjugated to Calcium-Binding Moieties. Biomacromolecules 8 (7), pp. 2237-2243. Fulltext not available.

Faerber, Lothar, Drechsler, Sabine, Ladenburger, Stephan, Gschaidmeier, Harald and Fischer, Wolfgang (2007) The neuronal 5-HT3 receptor network after 20 years of research — Evolving concepts in management of pain and inflammation. European Journal of Pharmacology 560 (1), pp. 1-8. Fulltext not available.

Mannschreck, Albrecht, Kiesswetter, Roland and von Angerer, Erwin (2007) Unequal Activities of Enantiomers via Biological Receptors: Examples of Chiral Drug, Pesticide, and Fragrance Molecules. Journal of Chemical Education 84 (12), p. 2012. Fulltext not available.

Amann, T., Spruss, T., Bataille, F., Liedtke, C., Muhlbauer, M., Trautwein, C., Bosserhoff, A.K. and Hellerbrand, C. (2007) [69] IDENTIFICATION OF FIBROBLAST GROWTH FACTOR RECEPTOR 2IIIB (FGFR2IIIB) AS TUMOR SUPPRESSOR IN HEPATOCANCEROGENESIS. Journal of Hepatology 46, S31. Fulltext not available.

2006

Lotter, Kristina (2006) Anti-inflammatorische Eigenschaften von Makrolid-Antibiotika bei akuter Lipopolysaccharid-induzierter Entzündung. PhD, Universität Regensburg.

Reithmeier-Rost, Dagmar (2006) Immunmodulation durch Interaktion des Yersinia enterocolitica V-Antigens mit Rezeptoren des angeborenen Immunsystems. PhD, Universität Regensburg.

Hellerbrand, C., Amann, T., Schlegel, J., Spruss, T., Bataille, F., Hartmann, A., Mühlbauer, M., Schölmerich, J. and Bosserhoff, A.K. (2006) 98 The novel gene MIA2 promotes progression of hepatocellular carcinoma. Journal of Hepatology 44, S43. Fulltext not available.

Fischer, Thomas, Bohmer, Frank D., Huber, Christoph, Dove, Stefan, Breitenbucher, Frank, Mirea, Fian K. and Heidel, Florian (2006) Bis(1H-indol-2yl)methanones Are Effective Inhibitors of Mutated FLT3 Tyrosine Kinase, Overcome Resistance to PKC412A In Vitro and Show Synergy with Chemotherapy. Blood 108 (11), p. 1369. Fulltext not available.

2005

Brandl, Katharina (2005) Untersuchungen zur pharmakologischen Beeinflussung der Toll-like Rezeptoren in der Sepsis. PhD, Universität Regensburg.

2004

Lyssenko, Alexei (2004) Synthese der Alkaloide Botryllazin B und (4-Hydroxyphenyl)-[4-(4-hydroxyphenyl)-1H-imidazol-2-yl]methanon sowie Synthese von Brevicollinderivaten. PhD, Universität Regensburg.

Walter, Georg, Liebl, Renate and Angerer, Erwin von (2004) 2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells. The Journal of Steroid Biochemistry and Molecular Biology 88 (4-5), pp. 409-420. Fulltext not available.

Bernhardt, Günther, Brunner, Henri, Gruber, Nick, Lottner, Christian, Pushpan, Simi K., Tsuno, Takashi

and Zabel, Manfred (2004) Carboplatin derivatives with superior antitumor activity compared to the parent compound. Inorganica Chimica Acta 357 (15), pp. 4452-4466. Fulltext not available.

Dittmar, Michael, Kiourkenidis, Georgios, Horn, Markus, Bollwein, Susanne and Bernhardt, Günther (2004) Cerebral Ischemia, Matrix Metalloproteinases, and TNF-α: MMP Inhibitors May Act Not Exclusively by Reducing MMP Activity. Stroke 35 (7). Fulltext not available.

Lottner, Christian, Knuechel, Ruth, Bernhardt, Guenther and Brunner, Henri (2004) Combined chemotherapeutic and photodynamic treatment on human bladder cells by hematoporphyrin–platinum(II) conjugates. Cancer Letters 203 (2), pp. 171-180. Fulltext not available.

Lottner, Christian, Knuechel, Ruth, Bernhardt, Günther and Brunner, Henri (2004) Distribution and subcellular localization of a water-soluble hematoporphyrin-platinum(II) complex in human bladder cancer cells. Cancer letters 215 (2), pp. 167-177. Fulltext not available.

Färber, L, Haus, U, Späth, M and Drechsler, S (2004) Physiology and pathophysiology of the 5‐HT3receptor. Scandinavian Journal of Rheumatology 33 (sup119), pp. 2-8. Fulltext not available.

Dove, Stefan (2004) Picolinic Acids as Inhibitors of Dopamine β‐Monooxygenase: QSAR and Putative Binding Site. Archiv der Pharmazie 337 (12), pp. 645-653. Fulltext not available.

Späth, M, Stratz, T, Färber, L, Haus, U and Pongratz, D (2004) Treatment of fibromyalgia with tropisetron – dose and efficacy correlations. Scandinavian Journal of Rheumatology 33 (sup119), pp. 63-66. Fulltext not available.

Schertl, Sabine, Hartmann, Rolf W., Batzl-Hartmann, Christine, Bernhardt, Günther, Spruß, Thilo, Beckenlehner, Karin, Koch, Marion, Krauser, Rudolf, Schlemmer, Richard, Gust, Ronald and Schönenberger, Helmut (2004) [1, 2-Bis(2, 6-difluoro-3-hydroxyphenyl)ethylene-diamine]platinum(II) complexes, compounds for the endocrine therapy of breast cancer - mode of action I: antitumor activity due to the reduction of the endogenous estrogen level. Archiv der Pharmazie 337 (6), pp. 335-348. Fulltext not available.

2003

Ladenburger, Stephan (2003) Relevanz der Galenik am Beispiel des Critical Dose Pharmakons Ciclosporin: Untersuchungen zur Pharmakokinetik und Pharmakodynamik verschiedener galenischer Formulierungen an gesunden Probanden und Ratten. PhD, Universität Regensburg.

Schneider, Dietmar (2003) Ringschluß- / Ringöffnungsreaktionen von Pyridinen: Synthese von N-Heterocyclen und Untersuchung auf Zytotoxizität. PhD, Universität Regensburg.

Jehkul, Andreas (2003) Klinisch-pharmakologische Untersuchungen zur Pharmakodynamik und Pharmakokinetik von Codein und Propyphenazon an Probanden und Patienten. PhD, Universität Regensburg.

Beckers, T., and Mahboobi, S., (2003) Natural, semisynthetic and synthetic microtubule inhibitors for cancer therapy. Drugs of the Future 28 (8), 0767. Fulltext not available.

Böhmer, Frank D., Karagyozov, Luchezar, Uecker, Andrea, Serve, Hubert, Botzki, Alexander

, Mahboobi, Siavosh and Dove, Stefan (2003) A Single Amino Acid Exchange Inverts Susceptibility of Related Receptor Tyrosine Kinases for the ATP Site Inhibitor STI-571. Journal of Biological Chemistry 278 (7), pp. 5148-5155. Fulltext not available.

Kaiser, Alexander, Mayer, Klaus K., Sellmer, Andreas and Wiegrebe, Wolfgang (2003) Electron Impact Induced Fragmentation of Aromatic Alkoxyimines II [5]. Formation and Transformation of Heterocyclic Radical Cations in the Gas Phase a. Monatshefte f�r Chemie / Chemical Monthly 134 (3), pp. 343-354. Fulltext not available.

Dittmar, Michael, Spruss, Thilo, Schuierer, Gerhard and Horn, Markus (2003) External Carotid Artery Territory Ischemia Impairs Outcome in the Endovascular Filament Model of Middle Cerebral Artery Occlusion in Rats. Stroke 34 (9), pp. 2252-2257. Fulltext not available.

2002

Dreher, Franziska (2002) Pharmakologische, molekularbiologische und biochemische Untersuchungen zur Beeinflussung des Renin-Angiotensin-Systems und der renalen Cyclooxygenase- und NO-Synthase-Isoenzyme in der Frühphase der primären, genetisch bedingten und sekundären, Immunsuppressivainduzierten Hypertonie. PhD, Universität Regensburg.

Bürgermeister, Jutta (2002) Wirkmechanistische Untersuchungen antiangiogener Galactansulfate. PhD, Universität Regensburg.

Köhler, Jens (2002) Untersuchungen zur Pharmakokinetik und Pharmakodynamik verschiedener galenischer Formulierungen des Immunsuppressivums Cyclosporin A vor und nach Nierentranplantation an Ratten. PhD, Universität Regensburg.

Apers, Sandra, Paper, Dietrich, Bürgermeister, Jutta, Baronikova, Slavka, Van Dyck, Stefaan, Lemière, Guy, Vlietinck, Arnold and Pieters, Luc

(2002) Antiangiogenic Activity of Synthetic Dihydrobenzofuran Lignans. Journal of Natural Products 65 (5), pp. 718-720. Fulltext not available.

Alban, S., Classen, B., Brunner, G., Franz, Gerhard and Blaschek, W. (2002) Differentiation between the Complement Modulating Effects of an Arabinogalactan-Protein from Echinacea purpurea and Heparin. (Dedicated to the 65th birthday of Prof. Dr. Gerhard Franz). Planta Medica 68, pp. 1118-1124. Fulltext not available.

Machein, U., Buss, B., Spiller, I., Braun, J., Rudwaleit, M., Faerber, L. and Sieper, J. (2002) Effective treatment of early rheumatoid arthritis with a combination of methotrexate, prednisolone and cyclosporin. Rheumatology 41 (1), pp. 110-111. Fulltext not available.

Lottner, Christian, Bart, Karl-Christian, Bernhardt, Günther and Brunner, Henri (2002) Hematoporphyrin-Derived Soluble Porphyrin−Platinum Conjugates with Combined Cytotoxic and Phototoxic Antitumor Activity. Journal of Medicinal Chemistry 45 (10), pp. 2064-2078. Fulltext not available.

Lottner, Christian, Bart, Karl-Christian, Bernhardt, Günther and Brunner, Henri (2002) Soluble Tetraarylporphyrin−Platinum Conjugates as Cytotoxic and Phototoxic Antitumor Agents. Journal of Medicinal Chemistry 45 (10), pp. 2079-2089. Fulltext not available.

Golob, Thomas, Liebl, Renate and von Angerer, Erwin (2002) Sulfamoyloxy-substituted 2-phenylindoles. Bioorganic & Medicinal Chemistry 10 (12), pp. 3941-3953. Fulltext not available.

2001

Otto, Angela, Schubert, Sybilla and Netzker, Roland (2001) Changes in the expression and binding properties of the estrogen receptor in MCF-7 breast cancer cells during growth inhibition by tamoxifen and cisplatin. Cancer Chemotherapy and Pharmacology 48 (4), pp. 305-311. Fulltext not available.

2000

Schönberger, Johann, Bauer, Johann, Spruß, Thilo, Weber, Gerhard, Chahoud, Ibrahim, Eilles, Christoph and Grimm, Daniela (2000) Establishment and characterization of the follicular thyroid carcinoma cell line ML-1. Journal of Molecular Medicine 78 (2), pp. 102-110. Fulltext not available.

This list was generated on Sun May 25 01:58:53 2025 CEST.

Export as	Atom RSS 1.0 RSS 2.0

2025

2024

2023

2022

2021

2020

2019

2018

2017

2016

2015

2014

2013

2012

2011

2010

2009

2008

2007

2006

2005

2004

2003

2002

2001

2000

University Library