Number of items at this level: 151.
2023
Kuck, Katrin,
Unterholzner, Anna,
Lipowicz, Bartosz,
Schwindl, Sebastian,
Jürgenliemk, Guido,
Schmidt, Thomas J. and
Heilmann, Jörg
(2023)
Terpenoids from Myrrh and Their Cytotoxic Activity against HeLa Cells.
Molecules 28 (4), p. 1637.
2022
Bresinsky, Merlin,
Strasser, Jessica M.,
Hubmann, Alexander,
Vallaster, Bernadette,
McCue, William M.,
Fuller, Jessica,
Singh, Gurpreet,
Nelson, Kathryn M.,
Cuellar, Matthew E.,
Finzel, Barry C.,
Ashe, Karen H.,
Walters, Michael A. and
Pockes, Steffen
(2022)
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis.
Archiv der Pharmazie 355 (9), p. 2200095.
Tahk, Maris-Johanna ,
Torp, Jane ,
Ali, Mohammed A. S. ,
Fishman, Dmytro,
Parts, Leopold ,
Grätz, Lukas ,
Müller, Christoph ,
Keller, Max ,
Veiksina, Santa ,
Laasfeld, Tõnis and
Rinken, Ago
(2022)
Live-cell microscopy or fluorescence anisotropy with budded baculoviruses—which way to go with measuring ligand binding to M 4 muscarinic receptors?
Open Biology 12 (6).
Fulltext not available.
Lier, Svenja,
Sellmer, Andreas,
Orben, Felix ,
Heinzlmeir, Stephanie,
Krauß, Lukas ,
Schneeweis, Christian,
Hassan, Zonera ,
Schneider, Carolin ,
Patricia Gloria Schäfer, Arlett,
Pongratz, Herwig,
Engleitner, Thomas,
Öllinger, Rupert,
Kuisl, Anna,
Bassermann, Florian,
Schlag, Christoph,
Kong, Bo,
Dove, Stefan,
Kuster, Bernhard,
Rad, Roland,
Reichert, Maximilian,
Wirth, Matthias ,
Saur, Dieter ,
Mahboobi, Siavosh and
Schneider, Günter
(2022)
A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer.
Bioorganic Chemistry 119, p. 105505.
Fulltext not available.
Schihada, Hannes,
Klompstra, Thomas M. ,
Humphrys, Laura J. ,
Cervenka, Igor,
Dadvar, Shamim ,
Kolb, Peter ,
Ruas, Jorge L. and
Schulte, Gunnar
(2022)
Isoforms of GPR35 have distinct extracellular N-termini that allosterically modify receptor-transducer coupling and mediate intracellular pathway bias.
Journal of Biological Chemistry 298 (9), p. 102328.
Fulltext not available.
Shcherbina, Nadezhda A.,
Kazakov, Igor V.,
Lisovenko, Anna S.,
Kryukova, Mariya A.,
Krasnova, Irina S. ,
Bodensteiner, Michael and
Timoshkin, Alexey Y.
(2022)
Molecular complexes of non-chelating polydentate Lewis bases with group 13 Lewis acids: crystal structure and computed energy of stepwise donor–acceptor bond formation.
Mendeleev Communications 32 (1), pp. 74-77.
Fulltext not available.
Schindler, Lisa,
Wohlfahrt, Katrin,
Gluhacevic von Krüchten, Lara,
Prante, Olaf,
Keller, Max and
Maschauer, Simone
(2022)
Neurotensin analogs by fluoroglycosylation at Nω-carbamoylated arginines for PET imaging of NTS1-positive tumors.
Scientific Reports 12 (1).
Fulltext not available.
Tang, Tingting,
Tan, Qiuxiang,
Han, Shuo,
Diemar, Anne,
Löbner, Kristin,
Wang, Hongyu,
Schüß, Corinna,
Behr, Victoria,
Mörl, Karin,
Wang, Mu,
Chu, Xiaojing,
Yi, Cuiying,
Keller, Max,
Kofoed, Jacob,
Reedtz-Runge, Steffen,
Kaiser, Anette,
Beck-Sickinger, Annette G.,
Zhao, Qiang and
Wu, Beili
(2022)
Receptor-specific recognition of NPY peptides revealed by structures of NPY receptors.
Science Advances 8 (18).
Fulltext not available.
Müller, Christoph,
Gleixner, Jakob ,
Tahk, Maris-Johanna ,
Kopanchuk, Sergei ,
Laasfeld, Tõnis,
Weinhart, Michael,
Schollmeyer, Dieter,
Betschart, Martin U.,
Lüdeke, Steffen,
Koch, Pierre,
Rinken, Ago and
Keller, Max
(2022)
Structure-Based Design of High-Affinity Fluorescent Probes for the Neuropeptide Y Y1 Receptor.
Journal of Medicinal Chemistry 65 (6), pp. 4832-4853.
Fulltext not available.
Rösch, G.,
El Bagdadi, K.,
Muschter, D.,
Taheri, S. ,
Dorn, C.,
Meurer, A.,
Straub, R.H.,
Zaucke, F. ,
Schilling, A.F.,
Grässel, S. and
Jenei-Lanzl, Z.
(2022)
Sympathectomy aggravates subchondral bone changes during osteoarthritis progression in mice without affecting cartilage degeneration or synovial inflammation.
Osteoarthritis and Cartilage 30 (3), pp. 461-474.
Fulltext not available.
2021
Rosier, Niklas,
Grätz, Lukas,
Schihada, Hannes ,
Möller, Jan,
Işbilir, Ali ,
Humphrys, Laura J. ,
Nagl, Martin,
Seibel, Ulla,
Lohse, Martin J. and
Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), pp. 11695-11708.
Fulltext not available.
Eap, C. B. ,
Gründer, G. ,
Baumann, P. ,
Ansermot, N.,
Conca, A.,
Corruble, E.,
Crettol, S.,
Dahl, M. L.,
de Leon, J. ,
Greiner, C.,
Howes, O.,
Kim, E.,
Lanzenberger, R.,
Meyer, J. H.,
Moessner, R.,
Mulder, H.,
Müller, D. J.,
Reis, M.,
Riederer, P.,
Ruhe, H. G.,
Spigset, O.,
Spina, E.,
Stegman, B.,
Steimer, W.,
Stingl, J. ,
Suzen, S.,
Uchida, H.,
Unterecker, S.,
Vandenberghe, F. and
Hiemke, C.
(2021)
Tools for optimising pharmacotherapy in psychiatry (therapeutic drug monitoring, molecular brain imaging and pharmacogenetic tests): focus on antidepressants.
The World Journal of Biological Psychiatry 22 (8), pp. 561-628.
Fulltext not available.
2020
Höring, Carina ,
Seibel, Ulla ,
Tropmann, Katharina,
Grätz, Lukas ,
Mönnich, Denise ,
Pitzl, Sebastian,
Bernhardt, Günther ,
Pockes, Steffen and
Strasser, Andrea
(2020)
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.
International Journal of Molecular Sciences 21 (22), p. 8440.
Grätz, Lukas,
Tropmann, Katharina,
Bresinsky, Merlin,
Müller, Christoph,
Bernhardt, Günther and
Pockes, Steffen
(2020)
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells.
Scientific Reports 10, p. 13288.
Bartole, Edith,
Grätz, Lukas,
Littmann, Timo,
Wifling, David ,
Seibel, Ulla,
Buschauer, Armin and
Bernhardt, Günther
(2020)
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors.
Journal of Medicinal Chemistry 63 (10), pp. 5297-5311.
Fulltext not available.
Maslanka Figueroa, Sara ,
Fleischmann, Daniel,
Beck, Sebastian,
Tauber, Philipp,
Witzgall, Ralph,
Schweda, Frank and
Goepferich, Achim
(2020)
Nanoparticles Mimicking Viral Cell Recognition Strategies Are Superior Transporters into Mesangial Cells.
Advanced Science 7 (11), p. 1903204.
Dorn, Christoph ,
Schießer, Selina,
Wulkersdorfer, Beatrix,
Hitzenbichler, Florian,
Kees, Martin G. and
Zeitlinger, Markus
(2020)
Determination of free clindamycin, flucloxacillin or tedizolid in plasma: Keep attention to physiological conditions when using ultrafiltration.
Biomedical Chromatography 34, e4820.
Fleischmann, Daniel,
Maslanka-Figueroa, Sara,
Beck, Sebastian,
Abstiens, Kathrin,
Witzgall, Ralph,
Schweda, Frank,
Tauber, Philipp and
Goepferich, Achim
(2020)
Adenovirus-Mimetic Nanoparticles: Sequential Ligand-Receptor Interplay as a Universal Tool for Enhanced In Vitro/In Vivo Cell Identification.
ACS Applied Materials & Interfaces 12 (31), pp. 34689-34702.
Fulltext not available.
Spinnler, Katrin,
von Krüchten, Lara,
Konieczny, Adam,
Schindler, Lisa,
Bernhardt, Günther and
Keller, Max
(2020)
An Alkyne-functionalized Arginine for Solid-Phase Synthesis Enabling “Bioorthogonal” Peptide Conjugation.
ACS Medicinal Chemistry Letters 11 (3), pp. 334-339.
Fulltext not available.
Weber, Laura,
Kuck, Katrin,
Jürgenliemk, Guido,
Heilmann, Jörg,
Lipowicz, Bartosz and
Vissiennon, Cica
(2020)
Anti-Inflammatory and Barrier-Stabilising Effects of Myrrh, Coffee Charcoal and Chamomile Flower Extract in a Co-Culture Cell Model of the Intestinal Mucosa.
Biomolecules 10 (7), p. 1033.
Fulltext not available.
Ullah, Sami,
Beer, Ronny,
Fuhr, Uwe,
Taubert, Max ,
Zeitlinger, Markus,
Kratzer, Alexander,
Dorn, Christoph,
Arshad, Usman,
Kofler, Mario and
Helbok, Raimund
(2020)
Brain Exposure to Piperacillin in Acute Hemorrhagic Stroke Patients Assessed by Cerebral Microdialysis and Population Pharmacokinetics.
Neurocritical Care.
Bohley, Marilena S.,
Birch, Emily,
Baumann, Felix J.,
Dillinger, Andrea E.,
Tamm, Ernst R. and
Goepferich, Achim M.
(2020)
Design of dye and superparamagnetic iron oxide nanoparticle loaded lipid nanocapsules with dual detectability in vitro and in vivo.
International Journal of Pharmaceutics 585, p. 119433.
Fulltext not available.
Gruber, Corinna G.,
Pegoli, Andrea,
Müller, Christoph,
Grätz, Lukas,
She, Xueke and
Keller, Max
(2020)
Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity.
RSC Medicinal Chemistry 11 (7), pp. 823-832.
Fulltext not available.
Keller, Max,
Mahuroof, Shahani A.,
Hong Yee, Vivyanne,
Carpenter, Jessica,
Schindler, Lisa,
Littmann, Timo,
Pegoli, Andrea,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter and
Holliday, Nicholas D.
(2020)
Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
ACS Medicinal Chemistry Letters 11 (1), pp. 16-22.
Fulltext not available.
Biselli, Sabrina,
Alencastre, Inês,
Tropmann, Katharina,
Erdmann, Daniela,
Chen, Mengya,
Littmann, Timo,
Maia, André F. ,
Gomez-Lazaro, Maria,
Tanaka, Miho,
Ozawa, Takeaki,
Keller, Max,
Lamghari, Meriem,
Buschauer, Armin and
Bernhardt, Günther
(2020)
Fluorescent H2 Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications.
ACS Medicinal Chemistry Letters 11 (8), pp. 1521-1528.
Fulltext not available.
Abdellatif, Ahmed ,
Hennig, Robert,
Pollinger, Klaus,
Tawfeek, Hesham,
Goepferich, Achim and
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(2020)
Fluorescent Nanoparticles Coated with a Somatostatin Analogue Target Blood Monocyte for Efficient Leukaemia Treatment.
Pharmaceutical Research 37 (11), p. 2017.
Sommer, Judith,
Dorn, Christoph ,
Gäbele, Erwin,
Bataille, Frauke,
Freese, Kim,
Seitz, Tatjana,
Thasler, Wolfgang E.,
Büttner, Reinhard,
Weiskirchen, Ralf ,
Bosserhoff, Anja and
Hellerbrand, Claus
(2020)
Four-And-A-Half LIM-Domain Protein 2 (FHL2) Deficiency Aggravates Cholestatic Liver Injury.
Cells 9 (1), p. 248.
Apaolaza, P.S. ,
Busch, M.,
Asin-Prieto, E. ,
Peynshaert, K. ,
Rathod, R.,
Remaut, K.,
Dünker, N. and
Göpferich, A.
(2020)
Hyaluronic acid coating of gold nanoparticles for intraocular drug delivery: Evaluation of the surface properties and effect on their distribution.
Experimental Eye Research 198, p. 108151.
Fulltext not available.
Biswas, Siladitta,
Kojonazarov, Baktybek,
Hadzic, Stefan,
Majer, Michael,
Bajraktari, Ganimete,
Novoyatleva, Tatyana,
Ghofrani, Hossein Ardeschir,
Grimminger, Friedrich,
Seeger, Werner,
Weissmann, Norbert,
Schlossmann, Jens and
Schermuly, Ralph Theo
(2020)
IRAG1 Deficient Mice Develop PKG1β Dependent Pulmonary Hypertension.
Cells 9 (10), p. 2280.
Fulltext not available.
Yagati, Ajay Kumar ,
Behrent, Arne,
Beck, Sebastian,
Rink, Simone,
Goepferich, Achim M.,
Min, Junhong ,
Lee, Min-Ho and
Baeumner, Antje J.
(2020)
Laser-induced graphene interdigitated electrodes for label-free or nanolabel-enhanced highly sensitive capacitive aptamer-based biosensors.
Biosensors and Bioelectronics 164, p. 112272.
Fulltext not available.
Pontes de Sousa, Ingrid,
Ferreira, Antônio Gilberto ,
Miller Crotti, Antônio Eduardo,
Alves dos Santos, Raquel,
Kiermaier, Josef,
Kraus, Birgit,
Heilmann, Jörg and
Jacometti Cardoso Furtado, Niege Araçari
(2020)
New antifungal ent-labdane diterpenes against Candida glabrata produced by microbial transformation of ent-polyalthic acid.
Bioorganic Chemistry 95, p. 103560.
Fulltext not available.
Ehmann, L.,
Simon, P.,
Busse, D.,
Petroff, D.,
Dorn, Christoph ,
Huisinga, W.,
Dietrich, A.,
Zeitlinger, M.,
Wrigge, H. and
Kloft, C.
(2020)
Risk of target non-attainment In obese compared to non-obese patients In Calculated linezolid therapy.
Clinical Microbiology and Infection.
Fulltext not available.
Stolwijk, Judith A.,
Mildner, Anne-Kathrin,
Kade, Christian,
Skiba, Michael,
Bernhardt, Guenther,
Buschauer, Armin,
Huebner, Harald,
Gmeiner, Peter and
Wegener, Joachim
(2020)
Stepwise Dosing Protocol for Increased Throughput in Label-Free Impedance-Based GPCR Assays.
Journal of Visualized Experiments (156).
Fulltext not available.
2019
Maschauer, Simone,
Ott, Julian J. ,
Bernhardt, Günther,
Kuwert, Torsten,
Keller, Max and
Prante, Olaf
(2019)
18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET Imaging of mammary carcinoma.
Scientific Reports 9, p. 12990.
Schramm, Andrea,
Schweda, Frank,
Sequeira-Lopez, Maria Luisa S.,
Hofmann, Franz,
Sandner, Peter and
Schlossmann, Jens
(2019)
Protein Kinase G Is Involved in Acute but Not in Long-Term Regulation of Renin Secretion.
Frontiers in Pharmacology 2019 (10), p. 800.
Dorn, Christoph,
Petroff, David,
Neumann, Nancy,
Kratzer, Alexander,
El-Najjar, Nahed ,
Dietrich, Arne,
Kloft, Charlotte,
Zeitlinger, Markus ,
Kees, Martin,
Kees, Frieder,
Wrigge, Hermann and
Simon, Philipp
(2019)
Plasma and tissue pharmacokinetics of fosfomycin in morbidly obese and non-obese surgical patients: a controlled clinical trial.
Journal of Antimicrobial Chemotherapy.
Fulltext not available.
Pegoli, Andrea,
Wifling, David ,
Gruber, Corinna G.,
Xueke, She,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter and
Keller, Max
(2019)
Conjugation of Short Peptides to Dibenzodiazepinone-Type
Muscarinic Acetylcholine Receptor Ligands Determines M2R
Selectivity.
Journal of Medicinal Chemistry 62, pp. 5358-5369.
Fulltext not available.
Schramm, Simon,
Agnetta, Luca,
Bermudez, Marcel,
Gerwe, Hubert,
Irmen, Matthias,
Holze, Janine,
Littmann, Timo,
Wolber, Gerhard ,
Tränkle, Christian and
Decker, Michael
(2019)
Novel BQCA‐ and TBPB‐Derived M 1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.
ChemMedChem 14 (14), pp. 1349-1358.
Fulltext not available.
Łażewska, Dorota ,
Mogilski, Szczepan,
Hagenow, Stefanie ,
Kuder, Kamil,
Głuch-Lutwin, Monika ,
Siwek, Agata ,
Więcek, Małgorzata,
Kaleta, Maria,
Seibel, Ulla,
Buschauer, Armin,
Filipek, Barbara,
Stark, Holger and
Kieć-Kononowicz, Katarzyna
(2019)
Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands.
Bioorganic & Medicinal Chemistry 27 (7), pp. 1254-1262.
Fulltext not available.
Polykandriotis, Elias,
Horch, Raymund E.,
Jost, Matthias,
Arkudas, Andreas,
Kees, Frieder and
Schmitz, Marweh
(2019)
Can systemically administered antibiotics be detected in wound tissues and surfaces under negative pressure wound therapy?
International Wound Journal 16 (2), pp. 503-510.
Fulltext not available.
Kowalewski, Christoph,
Haen, Ekkehard,
Hiemke, Christoph,
Ridders, Florian,
Endres, Katharina,
Gründer, Gerhard,
Paulzen, Michael and
Schoretsanitis, Georgios
(2019)
Cytochrome P450-mediated inhibition of venlafaxine metabolism by trimipramine.
International Clinical Psychopharmacology 34 (5), pp. 241-246.
Fulltext not available.
Dorn, Christoph ,
Kratzer, Alexander Ludwig,
Schießer, Selina,
Kees, Frieder ,
Wrigge, Hermann and
Simon, Philipp
(2019)
Determination of total or free cefazolin and metronidazole in human plasma or interstitial fluid by HPLC-UV for pharmacokinetic studies in man.
Journal of Chromatography B.
Fulltext not available.
Agnetta, Luca,
Bermudez, Marcel ,
Riefolo, Fabio ,
Matera, Carlo ,
Claro, Enrique ,
Messerer, Regina,
Littmann, Timo,
Wolber, Gerhard ,
Holzgrabe, Ulrike and
Decker, Michael
(2019)
Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties.
Journal of Medicinal Chemistry 62 (6), pp. 3009-3020.
Fulltext not available.
Walz, Johanna M.,
Wecker, Thomas ,
Zhang, Pei Pei,
Cakir, Bertan,
Gruening, Bjoern,
Agostini, Hansjuergen,
Reuer, Tristan,
Ludwig, Franziska,
Boneva, Stefaniya ,
Faerber, Lothar,
Lange, Clemens,
Schlunck, Guenther R. and
Stahl, Andreas
(2019)
Impact of angiogenic activation and inhibition on miRNA profiles of human retinal endothelial cells.
Experimental Eye Research 181, pp. 98-104.
Fulltext not available.
Stolwijk, J. A.,
Skiba, M.,
Kade, C.,
Bernhardt, G.,
Buschauer, Armin ,
Hübner, H.,
Gmeiner, P. and
Wegener, Joachim
(2019)
Increasing the throughput of label-free cell assays to study the activation of G-protein-coupled receptors by using a serial agonist exposure protocol.
Integrative Biology 11 (3), pp. 99-108.
Fulltext not available.
Gergs, U. ,
Bernhardt, Günther,
Buchwalow, I. B.,
Edler, H.,
Fröba, J.,
Keller, Max,
Kirchhefer, U.,
Köhler, F.,
Mißlinger, N.,
Wache, H. and
Neumann, J.
(2019)
Initial Characterization of Transgenic Mice Overexpressing Human Histamine H2 Receptors.
Journal of Pharmacology and Experimental Therapeutics 369 (1), pp. 129-141.
Fulltext not available.
Schoretsanitis, Georgios ,
Haen, Ekkehard,
Hiemke, Christoph,
Endres, Katharina,
Ridders, Florian,
Veselinovic, Tanja,
Gründer, Gerhard and
Paulzen, Michael
(2019)
Pharmacokinetic correlates of venlafaxine: associated adverse reactions.
European Archives of Psychiatry and Clinical Neuroscience 269 (7), pp. 851-857.
Fulltext not available.
Heider, Fabian ,
Ansideri, Francesco,
Tesch, Roberta,
Pantsar, Tatu,
Haun, Urs,
Döring, Eva,
Kudolo, Mark,
Poso, Antti ,
Albrecht, Wolfgang,
Laufer, Stefan A. and
Koch, Pierre
(2019)
Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors.
European Journal of Medicinal Chemistry 175, pp. 309-329.
Fulltext not available.
Nowak, Hartmuth,
Weidemann, Caroline,
Martini, Stefan,
Oesterreicher, Zoe Anne,
Dorn, Christoph,
Adamzik, Michael,
Kees, Frieder,
Zeitlinger, Markus and
Rahmel, Tim
(2019)
Repeated determination of moxifloxacin concentrations in interstitial space fluid of muscle and subcutis in septic patients.
Journal of Antimicrobial Chemotherapy.
Fulltext not available.
2018
Kratzer, Alexander,
Schießer, Selina,
Matzneller, Peter,
Wulkersdorfer, Beatrix,
Zeitlinger, Markus ,
Schlossmann, Jens ,
Kees, Frieder and
Dorn, Christoph
(2018)
Determination of Total and Free Ceftolozane and Tazobactam in Human Plasma and Interstitial Fluid by HPLC-UV.
Journal of Pharmaceutical and Biomedical Analysis.
Fulltext not available.
Walz, J. M.,
Bemme, S.,
Reichl, S.,
Akman, S.,
Breuß, H.,
Süsskind, D.,
Glitz, B.,
Müller, V. C.,
Wagenfeld, L.,
Gabel-Pfisterer, A.,
Aisenbrey, S.,
Engelmann, K.,
Koutsonas, A.,
Krohne, T. U. and
Stahl, A.
(2018)
Behandelte Frühgeborenenretinopathie in Deutschland.
Der Ophthalmologe 115 (6), pp. 476-488.
Fulltext not available.
Leonhardt, Michel,
Sellmer, Andreas ,
Krämer, Oliver H.,
Dove, Stefan,
Elz, Sigurd,
Kraus, Birgit,
Beyer, Mandy and
Mahboobi, Siavosh
(2018)
Design and biological evaluation of tetrahydro-β-carboline derivatives as highly potent histone deacetylase 6 (HDAC6) inhibitors.
European Journal of Medicinal Chemistry 152, pp. 329-357.
Fulltext not available.
Ridinger, Johannes,
Koeneke, Emily,
Kolbinger, Fiona R.,
Koerholz, Katharina,
Mahboobi, Siavosh,
Hellweg, Lars,
Gunkel, Nikolas,
Miller, Aubry K.,
Peterziel, Heike,
Schmezer, Peter,
Hamacher-Brady, Anne ,
Witt, Olaf and
Oehme, Ina
(2018)
Dual role of HDAC10 in lysosomal exocytosis and DNA repair promotes neuroblastoma chemoresistance.
Scientific Reports 8 (1).
Fulltext not available.
Dorn, Christoph,
Kratzer, Alexander,
Liebchen, Uwe,
Schleibinger, Michael,
Murschhauser, Alexandra,
Schlossmann, Jens ,
Kees, Frieder,
Simon, Philipp and
Kees, Martin G.
(2018)
Impact of Experimental Variables on the Protein Binding of Tigecycline in Human Plasma as Determined by Ultrafiltration.
Journal of Pharmaceutical Sciences 107 (2), pp. 739-744.
Fulltext not available.
Sellmer, Andreas,
Stangl, Hubert,
Beyer, Mandy,
Grünstein, Elisabeth,
Leonhardt, Michel,
Pongratz, Herwig,
Eichhorn, Emerich,
Elz, Sigurd,
Striegl, Birgit,
Jenei-Lanzl, Zsuzsa,
Dove, Stefan,
Straub, Rainer H.,
Krämer, Oliver H. and
Mahboobi, Siavosh
(2018)
Marbostat-100 Defines a New Class of Potent and Selective Antiinflammatory and Antirheumatic Histone Deacetylase 6 Inhibitors.
Journal of Medicinal Chemistry 61 (8), pp. 3454-3477.
Fulltext not available.
Schoretsanitis, Georgios,
de Leon, Jose,
Haen, Ekkehard,
Stegmann, Benedikt,
Hiemke, Christoph,
Gründer, Gerhard and
Paulzen, Michael
(2018)
Pharmacokinetics of risperidone in different application forms – Comparing long-acting injectable and oral formulations.
European Neuropsychopharmacology 28 (1), pp. 130-137.
Fulltext not available.
Mathioudaki, Angeliki,
Berzesta, Ariola,
Kypriotakis, Zacharias,
Skaltsa, Helen and
Heilmann, Jörg
(2018)
Phenolic metabolites from Hypericum kelleri Bald., an endemic species of Crete (Greece).
Phytochemistry 146, pp. 1-7.
Fulltext not available.
Peña-Solórzano, Diana,
Scholler, Matthias,
Bernhardt, Günther,
Buschauer, Armin ,
König, Burkhard and
Ochoa-Puentes, Cristian
(2018)
Tariquidar-Related Chalcones and Ketones as ABCG2 Modulators.
ACS Medicinal Chemistry Letters 9, pp. 854-859.
Fulltext not available.
2017
She, Xueke,
Pegoli, Andrea,
Mayr, Judith,
Hübner, Harald,
Bernhardt, Günther ,
Gmeiner, Peter and
Keller, Max
(2017)
Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity.
ACS Omega 2 (10), pp. 6741-6754.
Dukorn, Stefanie,
Littmann, Timo,
Keller, Max,
Kuhn, Kilian K.,
Cabrele, Chiara ,
Baumeister, Paul,
Bernhardt, Günther and
Buschauer, Armin
(2017)
Fluorescence- and radio-labeling of Lys4,Nle17,30hPP yields molecular tools for the NPY Y4 receptor.
Bioconjugate Chemistry.
Fulltext not available.
Noack, Katrin,
Mahendrarajah, Nisintha,
Hennig, Dorle,
Schmidt, Luisa,
Grebien, Florian ,
Hildebrand, Dagmar,
Christmann, Markus,
Kaina, Bernd,
Sellmer, Andreas,
Mahboobi, Siavosh,
Kubatzky, Katharina,
Heinzel, Thorsten and
Krämer, Oliver H.
(2017)
Analysis of the interplay between all-trans retinoic acid and histone deacetylase inhibitors in leukemic cells.
Archives of Toxicology 91 (5), pp. 2191-2208.
Fulltext not available.
Schäfer, Claudia,
Göder, Anja,
Beyer, Mandy,
Kiweler, Nicole,
Mahendrarajah, Nisintha,
Rauch, Anke,
Nikolova, Teodora,
Stojanovic, Natasa,
Wieczorek, Martin,
Reich, Thomas R.,
Tomicic, Maja T.,
Linnebacher, Michael,
Sonnemann, Jürgen,
Dietrich, Sascha,
Sellmer, Andreas,
Mahboobi, Siavosh,
Heinzel, Thorsten,
Schneider, Günter and
Krämer, Oliver H.
(2017)
Class I histone deacetylases regulate p53/NF-κB crosstalk in cancer cells.
Cellular Signalling 29, pp. 218-225.
Fulltext not available.
Schoretsanitis, Georgios ,
Haen, Ekkehard,
Stegmann, Benedikt,
Hiemke, Christoph,
Gründer, Gerhard and
Paulzen, Michael
(2017)
Effect of smoking on risperidone pharmacokinetics – A multifactorial approach to better predict the influence on drug metabolism.
Schizophrenia Research 185, pp. 51-57.
Fulltext not available.
Mahendrarajah, Nisintha,
Borisova, Marina E.,
Reichardt, Sigrid,
Godmann, Maren,
Sellmer, Andreas,
Mahboobi, Siavosh,
Haitel, Andrea,
Schmid, Katharina,
Kenner, Lukas ,
Heinzel, Thorsten,
Beli, Petra and
Krämer, Oliver H.
(2017)
HSP90 is necessary for the ACK1-dependent phosphorylation of STAT1 and STAT3.
Cellular Signalling 39, pp. 9-17.
Fulltext not available.
Kuhn, Kilian K.,
Littmann, Timo,
Dukorn, Stefanie,
Tanaka, Miho,
Keller, Max,
Ozawa, Takeaki,
Bernhardt, Günther and
Buschauer, Armin
(2017)
In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists.
ACS Omega 2 (7), pp. 3616-3631.
Pegoli, Andrea ,
She, Xueke,
Wifling, David ,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter and
Keller, Max
(2017)
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.
Journal of Medicinal Chemistry 60 (8), pp. 3314-3334.
Fulltext not available.
2016
Lieb, Sebastian,
Littmann, Timo,
Plank, Nicole,
Felixberger, Johannes,
Tanaka, Miho,
Schäfer, Thorsten,
Krief, Stéphane,
Elz, Sigurd,
Friedland, Kristina,
Bernhardt, Günther,
Wegener, Joachim,
Ozawa, Takeaki and
Buschauer, Armin
(2016)
Label-free versus conventional cellular assays: functional investigations on the human histamine H1 receptor.
Pharmacological Research 114, pp. 13-26.
Fulltext not available.
Töpper, Christoph,
Steinbach, Cathérine Louise,
Dorn, Christoph ,
Kratzer, Alexander,
Wicha, Sebastian G.,
Schleibinger, Michael,
Liebchen, Uwe,
Kees, Frieder,
Salzberger, Bernd and
Kees, Martin G.
(2016)
Variable linezolid exposure in ICU patients—possible role of drug-drug interactions.
Therapeutic Drug Monitoring 38 (5), pp. 573-578.
Fulltext not available.
Schlossmann, Jens,
Wetzl, Veronika,
Schinner, Elisabeth,
Kees, Frieder K.,
Hofmann, Franz and
Faerber, Lothar
(2016)
Involvement of cyclic guanosine monophosphate-dependent protein kinase I in renal antifibrotic effects of serelaxin.
Frontiers in Pharmacology 7 (195), pp. 1-27.
Kuhn, Kilian K.,
Ertl, Thomas,
Dukorn, Stefanie,
Keller, Max,
Bernhardt, Günther,
Reiser, Oliver and
Buschauer, Armin
(2016)
High affinity agonists of the neuropeptide Y (NPY) Y4 receptor derived from the C-terminal pentapeptide of human pancreatic polypeptide (hPP): synthesis, stereochemical discrimination and radiolabeling.
Journal of Medicinal Chemistry 59 (13), pp. 6045-6058.
Fulltext not available.
Lorenz, Peter,
Knittel, Diana N.,
Conrad, Jürgen,
Lotter, Eva M.,
Heilmann, Jörg,
Stintzing, Florian C. and
Kammerer, Dietmar R.
(2016)
1-Acetyl-3-[(3R)-hydroxyfatty acyl]glycerols: Lipid Compounds fromEuphrasia rostkovianaHayneandE. tetraquetra(Bréb.)Arrond.
Chemistry & Biodiversity 13 (5), pp. 602-612.
Fulltext not available.
Hammer, Sebastian,
Gobleder, Susanne,
Naporra, Franziska,
Wittmann, Hans-Joachim,
Elz, Sigurd,
Heinrich, Markus and
Strasser, Andrea
(2016)
2,4-Diaminopyrimidines as dual ligands at the histamine H1 and H4 receptor - H1/H4-receptor selectivity.
Bioorganic & Medicinal Chemistry Letters 26, pp. 292-300.
Fulltext not available.
Sawatzky, Edgar,
Wehle, Sarah,
Kling, Beata,
Wendrich, Jan,
Bringmann, Gerhard,
Sotriffer, Christoph A.,
Heilmann, Jörg and
Decker, Michael
(2016)
Discovery of Highly Selective and Nanomolar Carbamate-Based Butyrylcholinesterase Inhibitors by Rational Investigation into Their Inhibition Mode.
Journal of Medicinal Chemistry 59 (5), pp. 2067-2082.
Fulltext not available.
Keller, Max,
Kuhn, Kilian K.,
Einsiedel, Jürgen,
Hübner, Harald,
Biselli, Sabrina,
Mollereau, Catherine ,
Wifling, David,
Svobodova, Jaroslava,
Bernhardt, Günther,
Cabrele, Chiara ,
Vanderheyden, Patrick,
Gmeiner, Peter and
Buschauer, Armin
(2016)
Mimicking of arginine by functionalized Nω-carbamoylated arginine as a new broadly applicable approach to labeled bioactive peptides: high affinity angiotensin, neuropeptide Y, neuropeptide FF and neurotensin receptor ligands as examples.
Journal of Medicinal Chemistry 59 (5), pp. 1925-1945.
Fulltext not available.
Khan, Nadia,
Saad, Ali,
Nurulain, Syed M.,
Darras, Fouad H.,
Decker, Michael and
Sadek, Bassem
(2016)
The dual-acting H3 receptor antagonist and AChE inhibitor UW-MD-71 dose-dependently enhances memory retrieval and reverses dizocilpine-induced memory impairment in rats.
Behavioural Brain Research 297, pp. 155-164.
Fulltext not available.
Huang, Guozheng ,
Schramm, Simon,
Heilmann, Jörg,
Biedermann, David,
Křen, Vladimír and
Decker, Michael
(2016)
Unconventional application of the Mitsunobu reaction: Selective flavonolignan dehydration yielding hydnocarpins.
Beilstein Journal of Organic Chemistry 12, pp. 662-669.
Fulltext not available.
2015
Dolles, Dominik,
Nimczick, Martin,
Scheiner, Matthias,
Ramler, Jacqueline,
Stadtmüller, Patricia,
Sawatzky, Edgar,
Drakopoulos, Antonios ,
Sotriffer, Christoph,
Wittmann, Hans-Joachim,
Strasser, Andrea and
Decker, Michael
(2015)
Aminobenzimidazoles and Structural Isomers as Templates for Dual-Acting Butyrylcholinesterase Inhibitors andhCB2R Ligands To Combat Neurodegenerative Disorders.
ChemMedChem 11 (12), pp. 1270-1283.
Fulltext not available.
2014
2013
2012
2011
2009
2008
Egger, M.,
Pellett, P.,
Nickl, K.,
Geiger, S.,
Graetz, S.,
Seifert, R.,
Heilmann, J. and
König, B.
(2008)
Synthesis and Cannabinoid Receptor Activity of Ketoalkenes from Echinacea pallida and Non-natural Analogues.
Chem. Eur. J. 14, 10978 - 10984.
Fulltext not available.
2007
Schlegel, Birgit,
Laggner, Christian,
Meier, Rene,
Langer, Thierry,
Schnell, David,
Seifert, Roland,
Stark, Holger,
Höltje, Hans-Dieter and
Sippl, Wolfgang
(2007)
Generation of a homology model of the human histamine H₃ receptor for ligand docking and pharmacophore-based screening.
Journal of Computer-Aided Molecular Design.
2006
2005
2004
2003
2002
This list was generated on Wed Sep 11 16:14:11 2024 CEST.