Number of items at this level: 270.
2025
2024
Gonzalez-Valerio, Carlos,
Peregrina-Lucano, Alejandro A. 
,
Manríquez-González, Ricardo,
Pérez-Fonseca, Aida A.,
Robledo-Ortíz, Jorge R.,
Shenderovich, Ilya G. 
and
Gómez-Salazar, Sergio
(2024)
Color Compounds Removal from Tequila Vinasses Using Silica Gel Adsorbents Functionalized with Thiol Moieties: Equilibrium and Kinetics Studies.
Molecules 29 (24), p. 5910.
Becker, Jasmin,
Ellerkmann, Clara S.,
Schmelzer, Hannah,
Hermann, Christian,
Lützel, Kyra,
Gudermann, Thomas,
Konrad, David B.,
Trauner, Dirk,
Storch, Ursula 
and
Mederos y Schnitzler, Michael
(2024)
Optical Control of TRPM8 Channels with Photoswitchable Menthol.
Angewandte Chemie International Edition.
Ertl, Fabian J.,
Kopanchuk, Sergei 
,
Dijon, Nicola C.,
Veikšina, Santa,
Tahk, Maris-Johanna 
,
Laasfeld, Tõnis,
Schettler, Franziska,
Gattor, Albert O.,
Hübner, Harald,
Archipowa, Nataliya 
,
Köckenberger, Johannes,
Heinrich, Markus R.,
Gmeiner, Peter 
,
Kutta, Roger Jan 
,
Holliday, Nicholas D. 
,
Rinken, Ago 
and
Keller, Max 
(2024)
Dually Labeled Neurotensin NTS1R Ligands for Probing Radiochemical and Fluorescence-Based Binding Assays.
Journal of Medicinal Chemistry 67 (18), pp. 16664-16691.
2023
Mönnich, Denise,
Nagl, Martin,
Forster, Lisa,
Rosier, Niklas,
Igel, Patrick and
Pockes, Steffen
(2023)
Discovery of a Tritiated Radioligand with High Affinity and Selectivity for the Histamine H3 Receptor.
ACS Medicinal Chemistry Letters 14 (11), pp. 1589-1595.
Fulltext not available.
Szczepańska, Katarzyna,
Karcz, Tadeusz,
Dichiara, Maria,
Mogilski, Szczepan,
Kalinowska-Tłuścik, Justyna,
Pilarski, Bogusław,
Leniak, Arkadiusz,
Pietruś, Wojciech 
,
Podlewska, Sabina 
,
Popiołek-Barczyk, Katarzyna,
Humphrys, Laura J. 
,
Ruiz-Cantero, M. Carmen,
Reiner-Link, David 
,
Leitzbach, Luisa,
Łażewska, Dorota,
Pockes, Steffen 
,
Górka, Michał,
Zmysłowski, Adam,
Calmels, Thierry,
Cobos, Enrique J.,
Marrazzo, Agostino,
Stark, Holger,
Bojarski, Andrzej J.,
Amata, Emanuele and
Kieć-Kononowicz, Katarzyna
(2023)
Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain.
Journal of Medicinal Chemistry 66 (14), pp. 9658-9683.
Fulltext not available.
Plut, Eva 
,
Calderón, Jacqueline C.,
Stanojlović, Vesna,
Gattor, Albert O.,
Höring, Carina,
Humphrys, Laura J.,
Konieczny, Adam,
Kerres, Sabine,
Schubert, Mario 
,
Keller, Max,
Cabrele, Chiara,
Clark, Timothy and
Reiser, Oliver
(2023)
Stereochemistry-Driven Interactions of α,γ-Peptide Ligands with the Neuropeptide Y Y4-Receptor.
Journal of Medicinal Chemistry 66 (14), pp. 9642-9657.
Fulltext not available.
2022
Bresinsky, Merlin,
Strasser, Jessica M.,
Hubmann, Alexander,
Vallaster, Bernadette,
McCue, William M.,
Fuller, Jessica,
Singh, Gurpreet,
Nelson, Kathryn M.,
Cuellar, Matthew E.,
Finzel, Barry C.,
Ashe, Karen H.,
Walters, Michael A. and
Pockes, Steffen 
(2022)
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis.
Archiv der Pharmazie 355 (9), p. 2200095.
Tahk, Maris-Johanna 
,
Torp, Jane 
,
Ali, Mohammed A. S. 
,
Fishman, Dmytro,
Parts, Leopold 
,
Grätz, Lukas 
,
Müller, Christoph 
,
Keller, Max 
,
Veiksina, Santa 
,
Laasfeld, Tõnis 
and
Rinken, Ago 
(2022)
Live-cell microscopy or fluorescence anisotropy with budded baculoviruses—which way to go with measuring ligand binding to M 4 muscarinic receptors?
Open Biology 12 (6).
Fulltext not available.
Lier, Svenja,
Sellmer, Andreas,
Orben, Felix 
,
Heinzlmeir, Stephanie,
Krauß, Lukas 
,
Schneeweis, Christian,
Hassan, Zonera 
,
Schneider, Carolin 
,
Patricia Gloria Schäfer, Arlett,
Pongratz, Herwig,
Engleitner, Thomas,
Öllinger, Rupert,
Kuisl, Anna,
Bassermann, Florian,
Schlag, Christoph,
Kong, Bo,
Dove, Stefan,
Kuster, Bernhard,
Rad, Roland,
Reichert, Maximilian,
Wirth, Matthias 
,
Saur, Dieter 
,
Mahboobi, Siavosh and
Schneider, Günter 
(2022)
A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer.
Bioorganic Chemistry 119, p. 105505.
Fulltext not available.
Schihada, Hannes,
Klompstra, Thomas M. 
,
Humphrys, Laura J. 
,
Cervenka, Igor,
Dadvar, Shamim 
,
Kolb, Peter 
,
Ruas, Jorge L. 
and
Schulte, Gunnar 
(2022)
Isoforms of GPR35 have distinct extracellular N-termini that allosterically modify receptor-transducer coupling and mediate intracellular pathway bias.
Journal of Biological Chemistry 298 (9), p. 102328.
Fulltext not available.
Shcherbina, Nadezhda A.,
Kazakov, Igor V.,
Lisovenko, Anna S.,
Kryukova, Mariya A.,
Krasnova, Irina S. 
,
Bodensteiner, Michael and
Timoshkin, Alexey Y.
(2022)
Molecular complexes of non-chelating polydentate Lewis bases with group 13 Lewis acids: crystal structure and computed energy of stepwise donor–acceptor bond formation.
Mendeleev Communications 32 (1), pp. 74-77.
Fulltext not available.
Schindler, Lisa,
Wohlfahrt, Katrin,
Gluhacevic von Krüchten, Lara,
Prante, Olaf,
Keller, Max and
Maschauer, Simone
(2022)
Neurotensin analogs by fluoroglycosylation at Nω-carbamoylated arginines for PET imaging of NTS1-positive tumors.
Scientific Reports 12 (1).
Fulltext not available.
Tang, Tingting,
Tan, Qiuxiang,
Han, Shuo,
Diemar, Anne,
Löbner, Kristin,
Wang, Hongyu,
Schüß, Corinna,
Behr, Victoria,
Mörl, Karin,
Wang, Mu,
Chu, Xiaojing,
Yi, Cuiying,
Keller, Max,
Kofoed, Jacob,
Reedtz-Runge, Steffen,
Kaiser, Anette,
Beck-Sickinger, Annette G.,
Zhao, Qiang and
Wu, Beili
(2022)
Receptor-specific recognition of NPY peptides revealed by structures of NPY receptors.
Science Advances 8 (18).
Fulltext not available.
Müller, Christoph,
Gleixner, Jakob 
,
Tahk, Maris-Johanna 
,
Kopanchuk, Sergei 
,
Laasfeld, Tõnis,
Weinhart, Michael,
Schollmeyer, Dieter,
Betschart, Martin U.,
Lüdeke, Steffen,
Koch, Pierre,
Rinken, Ago 
and
Keller, Max
(2022)
Structure-Based Design of High-Affinity Fluorescent Probes for the Neuropeptide Y Y1 Receptor.
Journal of Medicinal Chemistry 65 (6), pp. 4832-4853.
Fulltext not available.
Rösch, G.,
El Bagdadi, K.,
Muschter, D.,
Taheri, S. 
,
Dorn, C.,
Meurer, A.,
Straub, R.H.,
Zaucke, F. 
,
Schilling, A.F.,
Grässel, S. and
Jenei-Lanzl, Z. 
(2022)
Sympathectomy aggravates subchondral bone changes during osteoarthritis progression in mice without affecting cartilage degeneration or synovial inflammation.
Osteoarthritis and Cartilage 30 (3), pp. 461-474.
Fulltext not available.
2021
Rosier, Niklas,
Grätz, Lukas,
Schihada, Hannes 
,
Möller, Jan,
Işbilir, Ali 
,
Humphrys, Laura J. 
,
Nagl, Martin,
Seibel, Ulla,
Lohse, Martin J. 
and
Pockes, Steffen 
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), pp. 11695-11708.
Fulltext not available.
Eap, C. B. 
,
Gründer, G. 
,
Baumann, P. 
,
Ansermot, N.,
Conca, A.,
Corruble, E.,
Crettol, S.,
Dahl, M. L.,
de Leon, J. 
,
Greiner, C.,
Howes, O.,
Kim, E.,
Lanzenberger, R.,
Meyer, J. H.,
Moessner, R.,
Mulder, H.,
Müller, D. J.,
Reis, M.,
Riederer, P.,
Ruhe, H. G.,
Spigset, O.,
Spina, E.,
Stegman, B.,
Steimer, W.,
Stingl, J. 
,
Suzen, S.,
Uchida, H.,
Unterecker, S.,
Vandenberghe, F. 
and
Hiemke, C. 
(2021)
Tools for optimising pharmacotherapy in psychiatry (therapeutic drug monitoring, molecular brain imaging and pharmacogenetic tests): focus on antidepressants.
The World Journal of Biological Psychiatry 22 (8), pp. 561-628.
Fulltext not available.
2020
Höring, Carina 
,
Seibel, Ulla 
,
Tropmann, Katharina,
Grätz, Lukas 
,
Mönnich, Denise 
,
Pitzl, Sebastian,
Bernhardt, Günther 
,
Pockes, Steffen 
and
Strasser, Andrea
(2020)
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.
International Journal of Molecular Sciences 21 (22), p. 8440.
Grätz, Lukas,
Tropmann, Katharina,
Bresinsky, Merlin,
Müller, Christoph,
Bernhardt, Günther 
and
Pockes, Steffen
(2020)
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells.
Scientific Reports 10, p. 13288.
Bartole, Edith,
Grätz, Lukas,
Littmann, Timo,
Wifling, David 
,
Seibel, Ulla,
Buschauer, Armin 
and
Bernhardt, Günther
(2020)
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors.
Journal of Medicinal Chemistry 63 (10), pp. 5297-5311.
Fulltext not available.
Maslanka Figueroa, Sara 
,
Fleischmann, Daniel,
Beck, Sebastian,
Tauber, Philipp,
Witzgall, Ralph,
Schweda, Frank and
Goepferich, Achim
(2020)
Nanoparticles Mimicking Viral Cell Recognition Strategies Are Superior Transporters into Mesangial Cells.
Advanced Science 7 (11), p. 1903204.
Dorn, Christoph 
,
Schießer, Selina,
Wulkersdorfer, Beatrix,
Hitzenbichler, Florian,
Kees, Martin G. 
and
Zeitlinger, Markus
(2020)
Determination of free clindamycin, flucloxacillin or tedizolid in plasma: Keep attention to physiological conditions when using ultrafiltration.
Biomedical Chromatography 34, e4820.
Fleischmann, Daniel,
Maslanka-Figueroa, Sara,
Beck, Sebastian,
Abstiens, Kathrin,
Witzgall, Ralph,
Schweda, Frank,
Tauber, Philipp and
Goepferich, Achim 
(2020)
Adenovirus-Mimetic Nanoparticles: Sequential Ligand-Receptor Interplay as a Universal Tool for Enhanced In Vitro/In Vivo Cell Identification.
ACS Applied Materials & Interfaces 12 (31), pp. 34689-34702.
Fulltext not available.
Spinnler, Katrin,
von Krüchten, Lara,
Konieczny, Adam,
Schindler, Lisa,
Bernhardt, Günther and
Keller, Max
(2020)
An Alkyne-functionalized Arginine for Solid-Phase Synthesis Enabling “Bioorthogonal” Peptide Conjugation.
ACS Medicinal Chemistry Letters 11 (3), pp. 334-339.
Fulltext not available.
Weber, Laura,
Kuck, Katrin,
Jürgenliemk, Guido,
Heilmann, Jörg,
Lipowicz, Bartosz and
Vissiennon, Cica 
(2020)
Anti-Inflammatory and Barrier-Stabilising Effects of Myrrh, Coffee Charcoal and Chamomile Flower Extract in a Co-Culture Cell Model of the Intestinal Mucosa.
Biomolecules 10 (7), p. 1033.
Fulltext not available.
Ullah, Sami,
Beer, Ronny,
Fuhr, Uwe,
Taubert, Max 
,
Zeitlinger, Markus,
Kratzer, Alexander,
Dorn, Christoph,
Arshad, Usman,
Kofler, Mario and
Helbok, Raimund
(2020)
Brain Exposure to Piperacillin in Acute Hemorrhagic Stroke Patients Assessed by Cerebral Microdialysis and Population Pharmacokinetics.
Neurocritical Care.
Bohley, Marilena S.,
Birch, Emily,
Baumann, Felix J.,
Dillinger, Andrea E.,
Tamm, Ernst R. and
Goepferich, Achim M.
(2020)
Design of dye and superparamagnetic iron oxide nanoparticle loaded lipid nanocapsules with dual detectability in vitro and in vivo.
International Journal of Pharmaceutics 585, p. 119433.
Fulltext not available.
Gruber, Corinna G.,
Pegoli, Andrea,
Müller, Christoph,
Grätz, Lukas,
She, Xueke and
Keller, Max
(2020)
Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity.
RSC Medicinal Chemistry 11 (7), pp. 823-832.
Fulltext not available.
Keller, Max,
Mahuroof, Shahani A.,
Hong Yee, Vivyanne,
Carpenter, Jessica,
Schindler, Lisa,
Littmann, Timo,
Pegoli, Andrea,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter 
and
Holliday, Nicholas D. 
(2020)
Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
ACS Medicinal Chemistry Letters 11 (1), pp. 16-22.
Fulltext not available.
Biselli, Sabrina,
Alencastre, Inês,
Tropmann, Katharina,
Erdmann, Daniela,
Chen, Mengya,
Littmann, Timo,
Maia, André F. 
,
Gomez-Lazaro, Maria,
Tanaka, Miho,
Ozawa, Takeaki,
Keller, Max,
Lamghari, Meriem,
Buschauer, Armin and
Bernhardt, Günther
(2020)
Fluorescent H2 Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications.
ACS Medicinal Chemistry Letters 11 (8), pp. 1521-1528.
Fulltext not available.
Sommer, Judith,
Dorn, Christoph 
,
Gäbele, Erwin,
Bataille, Frauke,
Freese, Kim,
Seitz, Tatjana,
Thasler, Wolfgang E.,
Büttner, Reinhard,
Weiskirchen, Ralf 
,
Bosserhoff, Anja 
and
Hellerbrand, Claus
(2020)
Four-And-A-Half LIM-Domain Protein 2 (FHL2) Deficiency Aggravates Cholestatic Liver Injury.
Cells 9 (1), p. 248.
Apaolaza, P.S. 
,
Busch, M.,
Asin-Prieto, E. 
,
Peynshaert, K. 
,
Rathod, R.,
Remaut, K.,
Dünker, N. and
Göpferich, A.
(2020)
Hyaluronic acid coating of gold nanoparticles for intraocular drug delivery: Evaluation of the surface properties and effect on their distribution.
Experimental Eye Research 198, p. 108151.
Fulltext not available.
Biswas, Siladitta,
Kojonazarov, Baktybek,
Hadzic, Stefan,
Majer, Michael,
Bajraktari, Ganimete,
Novoyatleva, Tatyana,
Ghofrani, Hossein Ardeschir,
Grimminger, Friedrich,
Seeger, Werner,
Weissmann, Norbert,
Schlossmann, Jens and
Schermuly, Ralph Theo
(2020)
IRAG1 Deficient Mice Develop PKG1β Dependent Pulmonary Hypertension.
Cells 9 (10), p. 2280.
Fulltext not available.
Yagati, Ajay Kumar 
,
Behrent, Arne,
Beck, Sebastian,
Rink, Simone,
Goepferich, Achim M.,
Min, Junhong 
,
Lee, Min-Ho 
and
Baeumner, Antje J. 
(2020)
Laser-induced graphene interdigitated electrodes for label-free or nanolabel-enhanced highly sensitive capacitive aptamer-based biosensors.
Biosensors and Bioelectronics 164, p. 112272.
Fulltext not available.
Pontes de Sousa, Ingrid,
Ferreira, Antônio Gilberto 
,
Miller Crotti, Antônio Eduardo,
Alves dos Santos, Raquel,
Kiermaier, Josef,
Kraus, Birgit,
Heilmann, Jörg and
Jacometti Cardoso Furtado, Niege Araçari
(2020)
New antifungal ent-labdane diterpenes against Candida glabrata produced by microbial transformation of ent-polyalthic acid.
Bioorganic Chemistry 95, p. 103560.
Fulltext not available.
Ehmann, L.,
Simon, P.,
Busse, D.,
Petroff, D.,
Dorn, Christoph 
,
Huisinga, W.,
Dietrich, A.,
Zeitlinger, M.,
Wrigge, H. and
Kloft, C.
(2020)
Risk of target non-attainment In obese compared to non-obese patients In Calculated linezolid therapy.
Clinical Microbiology and Infection.
Fulltext not available.
Stolwijk, Judith A.,
Mildner, Anne-Kathrin,
Kade, Christian,
Skiba, Michael,
Bernhardt, Guenther,
Buschauer, Armin,
Huebner, Harald,
Gmeiner, Peter and
Wegener, Joachim
(2020)
Stepwise Dosing Protocol for Increased Throughput in Label-Free Impedance-Based GPCR Assays.
Journal of Visualized Experiments (156).
Fulltext not available.
2019
Maschauer, Simone,
Ott, Julian J. 
,
Bernhardt, Günther,
Kuwert, Torsten,
Keller, Max and
Prante, Olaf
(2019)
18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET Imaging of mammary carcinoma.
Scientific Reports 9, p. 12990.
Schramm, Andrea,
Schweda, Frank,
Sequeira-Lopez, Maria Luisa S.,
Hofmann, Franz,
Sandner, Peter and
Schlossmann, Jens
(2019)
Protein Kinase G Is Involved in Acute but Not in Long-Term Regulation of Renin Secretion.
Frontiers in Pharmacology 2019 (10), p. 800.
Dorn, Christoph,
Petroff, David,
Neumann, Nancy,
Kratzer, Alexander,
El-Najjar, Nahed 
,
Dietrich, Arne,
Kloft, Charlotte,
Zeitlinger, Markus 
,
Kees, Martin,
Kees, Frieder,
Wrigge, Hermann and
Simon, Philipp
(2019)
Plasma and tissue pharmacokinetics of fosfomycin in morbidly obese and non-obese surgical patients: a controlled clinical trial.
Journal of Antimicrobial Chemotherapy.
Fulltext not available.
Pegoli, Andrea,
Wifling, David 
,
Gruber, Corinna G.,
Xueke, She,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter 
and
Keller, Max
(2019)
Conjugation of Short Peptides to Dibenzodiazepinone-Type
Muscarinic Acetylcholine Receptor Ligands Determines M2R
Selectivity.
Journal of Medicinal Chemistry 62, pp. 5358-5369.
Fulltext not available.
Schramm, Simon,
Agnetta, Luca,
Bermudez, Marcel,
Gerwe, Hubert,
Irmen, Matthias,
Holze, Janine,
Littmann, Timo,
Wolber, Gerhard 
,
Tränkle, Christian and
Decker, Michael
(2019)
Novel BQCA‐ and TBPB‐Derived M 1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.
ChemMedChem 14 (14), pp. 1349-1358.
Fulltext not available.
Łażewska, Dorota 
,
Mogilski, Szczepan,
Hagenow, Stefanie 
,
Kuder, Kamil,
Głuch-Lutwin, Monika 
,
Siwek, Agata 
,
Więcek, Małgorzata,
Kaleta, Maria,
Seibel, Ulla,
Buschauer, Armin,
Filipek, Barbara,
Stark, Holger 
and
Kieć-Kononowicz, Katarzyna
(2019)
Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands.
Bioorganic & Medicinal Chemistry 27 (7), pp. 1254-1262.
Fulltext not available.
Polykandriotis, Elias,
Horch, Raymund E.,
Jost, Matthias,
Arkudas, Andreas,
Kees, Frieder and
Schmitz, Marweh
(2019)
Can systemically administered antibiotics be detected in wound tissues and surfaces under negative pressure wound therapy?
International Wound Journal 16 (2), pp. 503-510.
Fulltext not available.
Kowalewski, Christoph,
Haen, Ekkehard,
Hiemke, Christoph,
Ridders, Florian,
Endres, Katharina,
Gründer, Gerhard,
Paulzen, Michael and
Schoretsanitis, Georgios
(2019)
Cytochrome P450-mediated inhibition of venlafaxine metabolism by trimipramine.
International Clinical Psychopharmacology 34 (5), pp. 241-246.
Fulltext not available.
Dorn, Christoph 
,
Kratzer, Alexander Ludwig,
Schießer, Selina,
Kees, Frieder 
,
Wrigge, Hermann and
Simon, Philipp
(2019)
Determination of total or free cefazolin and metronidazole in human plasma or interstitial fluid by HPLC-UV for pharmacokinetic studies in man.
Journal of Chromatography B.
Fulltext not available.
Agnetta, Luca,
Bermudez, Marcel 
,
Riefolo, Fabio 
,
Matera, Carlo 
,
Claro, Enrique 
,
Messerer, Regina,
Littmann, Timo,
Wolber, Gerhard 
,
Holzgrabe, Ulrike and
Decker, Michael
(2019)
Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties.
Journal of Medicinal Chemistry 62 (6), pp. 3009-3020.
Fulltext not available.
Walz, Johanna M.,
Wecker, Thomas 
,
Zhang, Pei Pei,
Cakir, Bertan,
Gruening, Bjoern,
Agostini, Hansjuergen,
Reuer, Tristan,
Ludwig, Franziska,
Boneva, Stefaniya 
,
Faerber, Lothar,
Lange, Clemens,
Schlunck, Guenther R. and
Stahl, Andreas
(2019)
Impact of angiogenic activation and inhibition on miRNA profiles of human retinal endothelial cells.
Experimental Eye Research 181, pp. 98-104.
Fulltext not available.
Stolwijk, J. A.,
Skiba, M.,
Kade, C.,
Bernhardt, G.,
Buschauer, Armin 
,
Hübner, H.,
Gmeiner, P. and
Wegener, Joachim 
(2019)
Increasing the throughput of label-free cell assays to study the activation of G-protein-coupled receptors by using a serial agonist exposure protocol.
Integrative Biology 11 (3), pp. 99-108.
Fulltext not available.
Gergs, U. 
,
Bernhardt, Günther,
Buchwalow, I. B.,
Edler, H.,
Fröba, J.,
Keller, Max,
Kirchhefer, U.,
Köhler, F.,
Mißlinger, N.,
Wache, H. and
Neumann, J.
(2019)
Initial Characterization of Transgenic Mice Overexpressing Human Histamine H2 Receptors.
Journal of Pharmacology and Experimental Therapeutics 369 (1), pp. 129-141.
Fulltext not available.
Schoretsanitis, Georgios 
,
Haen, Ekkehard,
Hiemke, Christoph,
Endres, Katharina,
Ridders, Florian,
Veselinovic, Tanja,
Gründer, Gerhard and
Paulzen, Michael
(2019)
Pharmacokinetic correlates of venlafaxine: associated adverse reactions.
European Archives of Psychiatry and Clinical Neuroscience 269 (7), pp. 851-857.
Fulltext not available.
Heider, Fabian 
,
Ansideri, Francesco,
Tesch, Roberta,
Pantsar, Tatu,
Haun, Urs,
Döring, Eva,
Kudolo, Mark,
Poso, Antti 
,
Albrecht, Wolfgang,
Laufer, Stefan A. 
and
Koch, Pierre
(2019)
Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors.
European Journal of Medicinal Chemistry 175, pp. 309-329.
Fulltext not available.
Nowak, Hartmuth,
Weidemann, Caroline,
Martini, Stefan,
Oesterreicher, Zoe Anne,
Dorn, Christoph,
Adamzik, Michael,
Kees, Frieder,
Zeitlinger, Markus 
and
Rahmel, Tim 
(2019)
Repeated determination of moxifloxacin concentrations in interstitial space fluid of muscle and subcutis in septic patients.
Journal of Antimicrobial Chemotherapy.
Fulltext not available.
2018
Kratzer, Alexander,
Schießer, Selina,
Matzneller, Peter,
Wulkersdorfer, Beatrix,
Zeitlinger, Markus 
,
Schlossmann, Jens 
,
Kees, Frieder 
and
Dorn, Christoph
(2018)
Determination of Total and Free Ceftolozane and Tazobactam in Human Plasma and Interstitial Fluid by HPLC-UV.
Journal of Pharmaceutical and Biomedical Analysis.
Fulltext not available.
Walz, J. M.,
Bemme, S.,
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Journal of Medicinal Chemistry 59 (13), pp. 6045-6058.
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Discovery of Highly Selective and Nanomolar Carbamate-Based Butyrylcholinesterase Inhibitors by Rational Investigation into Their Inhibition Mode.
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Mimicking of arginine by functionalized Nω-carbamoylated arginine as a new broadly applicable approach to labeled bioactive peptides: high affinity angiotensin, neuropeptide Y, neuropeptide FF and neurotensin receptor ligands as examples.
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Unconventional application of the Mitsunobu reaction: Selective flavonolignan dehydration yielding hydnocarpins.
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N(omega)-carbamoylation of the argininamide moiety: an avenue to insurmountable NPY Y1 receptor antagonists and a radiolabeled selective high affinity molecular tool ([3H]UR-MK299) with extended residence time.
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New insights into the cross-linking and degradation mechanism of Diels–Alder hydrogels.
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Loratadine and analogs: Discovery and preliminary SAR of inhibitors of the amino acid transporter B0AT2.
Journal of Medicinal Chemistry 57 (22), pp. 9473-9479.
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Aqueous Extracts of the Marine Brown Alga Lobophora variegata Inhibit HIV-1 Infection at the Level of Virus Entry into Cells.
PloS ONE 9, e103895.
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Biodistribution of quantum dots in the kidney after intravenous injection.
Journal of Nanoscience and Nanotechnology 14 (5), pp. 3313-3319.
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Determination of free vancomycin, ceftriaxone, cefazolin and ertapenem in plasma by ultrafiltration: Impact of experimental conditions.
Journal of Chromatography B 961, pp. 97-102.
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Kees, Martin Georg,
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Population pharmacokinetics and pharmacodynamic evaluation of intravenous and enteral moxifloxacin in surgical intensive care unit patients.
The Journal of antimicrobial chemotherapy.
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Knuth, Susanne,
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Catechol Conjugates Are In Vivo Metabolites of Salicis cortex.
Planta Medica 79 (16), pp. 1489-1494.
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Miller, Tobias,
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Pharmacokinetics, biocompatibility and bioavailability of a controlled release monoclonal antibody formulation.
Journal of Controlled Release 172 (3), pp. 975-982.
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Miller, Tobias,
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Premature drug release of polymeric micelles and its effects on tumor targeting.
International Journal of Pharmaceutics 445 (1-2), pp. 117-124.
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Memminger, Martin,
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The Neuropeptide Y Y1 receptor: a diagnostic marker? Expression in MCF-7 breast cancer cells is down-regulated by antiestrogens in vitro and in xenografts.
PLoS ONE 7 (12), e51032.
Bubik, Martin F.,
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A novel approach to prevent endothelial hyperpermeability: The Crataegus extract WS® 1442 targets the cAMP/Rap1 pathway.
Journal of Molecular and Cellular Cardiology 52 (1), pp. 196-205.
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Freischmidt, A.,
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Contribution of flavonoids and catechol to the reduction of ICAM-1 expression in endothelial cells by a standardised Willow bark extract.
Phytomedicine 19 (3-4), pp. 245-252.
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Cytotoxic tetraoxygenated xanthones from the bark of Garcinia schomburgkiana.
Phytochemistry Letters 5 (3), pp. 553-557.
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Posavec, Damir,
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Functionalized derivatives of 1,4-dimethylnaphthalene as precursors for biomedical applications: synthesis, structures, spectroscopy and photochemical activation in the presence of dioxygen.
Organic & biomolecular chemistry 10 (35), pp. 7062-7069.
Saugspier, Michael,
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Hop bitter acids inhibit tumorigenicity of hepatocellular carcinoma cells in vitro.
Oncology Reports 28 (4), pp. 1423-1428.
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Appl, Heidrun,
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Interactions of recombinant human histamine H₁R, H₂R, H₃R, and H₄R receptors with 34 antidepressants and antipsychotics.
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Pollinger, Klaus,
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Kidney Podocytes as Specific Targets for cyclo(RGDfC)-Modified Nanoparticles.
Small 8, pp. 3368-3375.
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Elbakry, Asmaa Mohamed,
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Layer-by-Layer Coated Gold Nanoparticles: Size-Dependent Delivery of DNA into Cells.
Small 8 (24), pp. 3847-3856.
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Nguyen, Le-Thu T.,
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Polyisoprenylated acylphloroglucinols and a polyisoprenylated tetracyclic xanthone from the bark of Calophyllum thorelii.
Tetrahedron Letters 53 (34), pp. 4487-4493.
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Ulrich-Merzenich, G.,
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Prediction of adverse events by in vivo gene expression profiling exemplified for phytopharmaceuticals containing salicylates and the antidepressant imipramine.
Phytomedicine 19 (3-4), pp. 322-329.
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Schmidt, Jennifer,
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Targeting melanoma metastasis and immunosuppression with a new mode of melanoma inhibitory activity (MIA) protein inhibition.
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cGMP-Prkg1 signaling and Pde5 inhibition shelter cochlear hair cells and hearing function.
Nature Medicine 18 (2), pp. 252-259.
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Pop, Nathalie,
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Functional reconstitution of human neuropeptide Y (NPY) Y2 and Y4 receptors in Sf9 insect cells.
Journal of Receptors and Signal Transduction 31 (4), pp. 271-285.
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How Stealthy are PEG-PLA Nanoparticles? An NIR In Vivo Study Combined with Detailed Size Measurements.
Pharmaceutical Research 28 (8), pp. 1995-2007.
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Dayoub, Rania 
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Oldenburg, J.,
Jilg, W. and
Eis-Hübinger, A. M.
(2010)
Prevalence of nucleic acid sequences specific for human parvoviruses, hepatitis A and hepatitis E viruses in coagulation factor concentrates.
Vox sanguinis.
Fulltext restricted.
Amann, Thomas,
Bataille, Frauke,
Spruss, Thilo,
Dettmer, Katja 
,
Wild, Peter J.,
Liedtke, Christian 
,
Mühlbauer, Marcus,
Kiefer, Paul,
Oefner, Peter J. 
,
Trautwein, Christian,
Bosserhoff, Anja-Katrin 
and
Hellerbrand, Claus
(2010)
Reduced expression of fibroblast growth factor receptor 2IIIb in hepatocellular carcinoma induces a more aggressive growth.
The American journal of pathology 176 (3), pp. 1433-42.
Fulltext not available.
Fürst, R,
Bubik, M,
Bihari, P,
Jürgenliemk, G,
Ammer, H,
Krombach, F,
Zahler, S and
Vollmar, A
(2010)
The hawthorn special extract WS® 1442 protects against endothelial barrier dysfunction – elucidation of the underlying molecular mechanisms.
Planta Medica 76 (12).
Fulltext not available.
2009
Sander, Kerstin,
Kottke, Tim,
Tanrikulu, Yusuf,
Proschak, Ewgenij,
Weizel, Lilia,
Schneider, Erich H. 
,
Seifert, Roland,
Schneider, Gisbert 
and
Stark, Holger 
(2009)
2,4-Diaminopyrimidines as histamine H4 receptor ligands—Scaffold optimization and pharmacological characterization.
Bioorganic & Medicinal Chemistry 17 (20), pp. 7186-7196.
Fulltext not available.
Amann, Thomas,
Bataille, Frauke,
Spruss, Thilo,
Mühlbauer, Marcus,
Gäbele, Erwin,
Schölmerich, Jürgen,
Kiefer, Paul,
Bosserhoff, Anja‐Katrin 
and
Hellerbrand, Claus
(2009)
Activated hepatic stellate cells promote tumorigenicity of hepatocellular carcinoma.
Cancer Science 100 (4), pp. 646-653.
Fulltext not available.
Weiser, Barbara,
Sommer, Florian,
Neubauer, M.,
Seitz, Anna Katharina,
Teßmar, Jörg 
,
Göpferich, Achim 
and
Blunk, Torsten
(2009)
Ascorbic Acid Enhances Adipogenesis of Bone Marrow-Derived Mesenchymal Stromal Cells.
Cells Tissues Organs 189 (6), pp. 373-381.
Fulltext not available.
Göttle, Martin,
Geduhn, Jens,
König, Burkhard 
,
Gille, Andreas 
,
Höcherl, Klaus and
Seifert, Roland
(2009)
Characterization of Mouse Heart Adenylyl Cyclase.
Journal of Pharmacology and Experimental Therapeutics 329 (3), pp. 1156-1165.
Fulltext not available.
Mahboobi, Siavosh,
Dove, Stefan,
Sellmer, Andreas,
Winkler, Matthias,
Eichhorn, Emerich,
Pongratz, Herwig,
Ciossek, Thomas,
Baer, Thomas,
Maier, Thomas and
Beckers, Thomas
(2009)
Design of chimeric histone deacetylase- and tyrosine kinase-inhibitors: a series of imatinib hybrides as potent inhibitors of wild-type and mutant BCR-ABL, PDGF-Rbeta, and histone deacetylases.
Journal of medicinal chemistry 52 (8), pp. 2265-79.
Fulltext not available.
Massoumi, Ramin,
Kuphal, Silke,
Hellerbrand, Claus,
Haas, Bodo 
,
Wild, Peter,
Spruss, Thilo,
Pfeifer, Alexander,
Fässler, Reinhard and
Bosserhoff, Anja K. 
(2009)
Down-regulation of CYLD expression by Snail promotes tumor progression in malignant melanoma.
Journal of Experimental Medicine 206 (1), pp. 221-232.
Fulltext not available.
2008
Vogel, Susanne,
Kaufmann, Doris,
Pojarová, Michaela,
Müller, Christine,
Pfaller, Tobias,
Kühne, Sybille,
Bednarski, Patrick J. and
Angerer, Erwin von
(2008)
Aroyl hydrazones of 2-phenylindole-3-carbaldehydes as novel antimitotic agents.
Bioorganic & Medicinal Chemistry 16 (12), pp. 6436-6447.
Fulltext not available.
Sommer, Florian,
Pollinger, Klaus,
Brandl, Ferdinand,
Weiser, Barbara,
Teßmar, Jörg 
,
Blunk, Torsten and
Göpferich, Achim 
(2008)
Hyalocyte proliferation and ECM accumulation modulated by bFGF and TGF-β1.
Graefe's Archive for Clinical and Experimental Ophthalmology 246 (9), pp. 1275-1284.
Fulltext not available.
Weiser, Barbara,
Prantl, Lukas,
Schubert, Thomas E. O.,
Zellner, J. 
,
Fischbach-Teschl, Claudia,
Spruss, Thilo,
Seitz, Anna Katharina,
Teßmar, Jörg 
,
Göpferich, Achim 
and
Blunk, Torsten
(2008)
In Vivo Development and Long-Term Survival of Engineered Adipose Tissue Depend on In Vitro Precultivation Strategy.
Tissue Engineering Part A 14 (2), pp. 275-284.
Fulltext not available.
Egger, M.,
Pellett, P.,
Nickl, K.,
Geiger, S.,
Graetz, S.,
Seifert, R.,
Heilmann, J. and
König, B. 
(2008)
Synthesis and Cannabinoid Receptor Activity of Ketoalkenes from Echinacea pallida and Non-natural Analogues.
Chem. Eur. J. 14, 10978 - 10984.
Fulltext not available.
Hellerbrand, C,
Amann, T,
Schlegel, J,
Wild, P,
Bataille, F,
Spruss, T,
Hartmann, A and
Bosserhoff, A-K 
(2008)
The novel gene MIA2 acts as a tumour suppressor in hepatocellular carcinoma.
Gut 57 (2), pp. 243-251.
Fulltext not available.
2007
Göttle, Martin,
Dove, Stefan,
Steindel, Phillip,
Shen, Yuequan,
Tang, Wei-Jen 
,
Geduhn, Jens,
König, Burkhard 
and
Seifert, Roland
(2007)
Molecular Analysis of the Interaction of Bordetella pertussis Adenylyl Cyclase with Fluorescent Nucleotides.
Molecular Pharmacology 72 (3), pp. 526-535.
Kaufmann, Doris,
Pojarová, Michaela,
Vogel, Susanne,
Liebl, Renate,
Gastpar, Robert,
Gross, Dietmar,
Nishino, Tsuyuki,
Pfaller, Tobias and
Angerer, Erwin von
(2007)
Antimitotic activities of 2-phenylindole-3-carbaldehydes in human breast cancer cells.
Bioorganic & medicinal chemistry 15 (15), pp. 5122-36.
Fulltext not available.
Amann, T.,
Spruss, T.,
Bataille, F.,
Liedtke, C.,
Muhlbauer, M.,
Trautwein, C.,
Bosserhoff, A.K. and
Hellerbrand, C.
(2007)
[69] IDENTIFICATION OF FIBROBLAST GROWTH FACTOR RECEPTOR 2IIIB (FGFR2IIIB) AS TUMOR SUPPRESSOR IN HEPATOCANCEROGENESIS.
Journal of Hepatology 46, S31.
Fulltext not available.
2006
Hellerbrand, C.,
Amann, T.,
Schlegel, J.,
Spruss, T.,
Bataille, F.,
Hartmann, A.,
Mühlbauer, M.,
Schölmerich, J. and
Bosserhoff, A.K.
(2006)
98 The novel gene MIA2 promotes progression of hepatocellular carcinoma.
Journal of Hepatology 44, S43.
Fulltext not available.
Fischer, Thomas,
Bohmer, Frank D.,
Huber, Christoph,
Dove, Stefan,
Breitenbucher, Frank,
Mirea, Fian K. and
Heidel, Florian
(2006)
Bis(1H-indol-2yl)methanones Are Effective Inhibitors of Mutated FLT3 Tyrosine Kinase, Overcome Resistance to PKC412A In Vitro and Show Synergy with Chemotherapy.
Blood 108 (11), p. 1369.
Fulltext not available.
2005
2004
Bernhardt, Günther,
Brunner, Henri,
Gruber, Nick,
Lottner, Christian,
Pushpan, Simi K.,
Tsuno, Takashi 
and
Zabel, Manfred
(2004)
Carboplatin derivatives with superior antitumor activity compared to the parent compound.
Inorganica Chimica Acta 357 (15), pp. 4452-4466.
Fulltext not available.
Dittmar, Michael,
Kiourkenidis, Georgios,
Horn, Markus,
Bollwein, Susanne and
Bernhardt, Günther
(2004)
Cerebral Ischemia, Matrix Metalloproteinases, and TNF-α: MMP Inhibitors May Act Not Exclusively by Reducing MMP Activity.
Stroke 35 (7).
Fulltext not available.
Schertl, Sabine,
Hartmann, Rolf W.,
Batzl-Hartmann, Christine,
Bernhardt, Günther,
Spruß, Thilo,
Beckenlehner, Karin,
Koch, Marion,
Krauser, Rudolf,
Schlemmer, Richard,
Gust, Ronald and
Schönenberger, Helmut
(2004)
[1, 2-Bis(2, 6-difluoro-3-hydroxyphenyl)ethylene-diamine]platinum(II) complexes, compounds for the endocrine therapy of breast cancer - mode of action I: antitumor activity due to the reduction of the endogenous estrogen level.
Archiv der Pharmazie 337 (6), pp. 335-348.
Fulltext not available.
2003
Böhmer, Frank D.,
Karagyozov, Luchezar,
Uecker, Andrea,
Serve, Hubert,
Botzki, Alexander 
,
Mahboobi, Siavosh and
Dove, Stefan
(2003)
A Single Amino Acid Exchange Inverts Susceptibility of Related Receptor Tyrosine Kinases for the ATP Site Inhibitor STI-571.
Journal of Biological Chemistry 278 (7), pp. 5148-5155.
Fulltext not available.
2002
Apers, Sandra,
Paper, Dietrich,
Bürgermeister, Jutta,
Baronikova, Slavka,
Van Dyck, Stefaan,
Lemière, Guy,
Vlietinck, Arnold and
Pieters, Luc 
(2002)
Antiangiogenic Activity of Synthetic Dihydrobenzofuran Lignans.
Journal of Natural Products 65 (5), pp. 718-720.
Fulltext not available.
Machein, U.,
Buss, B.,
Spiller, I.,
Braun, J.,
Rudwaleit, M.,
Faerber, L. and
Sieper, J.
(2002)
Effective treatment of early rheumatoid arthritis with a combination of methotrexate, prednisolone and cyclosporin.
Rheumatology 41 (1), pp. 110-111.
Fulltext not available.
2001
2000
Schönberger, Johann,
Bauer, Johann,
Spruß, Thilo,
Weber, Gerhard,
Chahoud, Ibrahim,
Eilles, Christoph and
Grimm, Daniela
(2000)
Establishment and characterization of the follicular thyroid carcinoma cell line ML-1.
Journal of Molecular Medicine 78 (2), pp. 102-110.
Fulltext not available.
This list was generated on Sun May 25 01:58:53 2025 CEST.