Design and biological evaluation of tetrahydro-β-carboline derivatives as highly potent histone deacetylase 6 (HDAC6) inhibitors
Article
Leonhardt, Michel, Sellmer, Andreas
, Krämer, Oliver H., Dove, Stefan, Elz, Sigurd, Kraus, Birgit, Beyer, Mandy and Mahboobi, Siavosh
(2018)
Design and biological evaluation of tetrahydro-β-carboline derivatives as highly potent histone deacetylase 6 (HDAC6) inhibitors.
European Journal of Medicinal Chemistry 152, pp. 329-357.
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| Item type | Article | ||||
| Journal or Publication Title | European Journal of Medicinal Chemistry | ||||
| Publisher | ELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER | ||||
| Place of Publication | ISSY-LES-MOULINEAUX | ||||
| Volume | 152 | ||||
| Page Range | pp. 329-357 | ||||
| Date | 2018 | ||||
| Date of publication | 28 Jul 2021 17:15 | ||||
| Institutions | Chemistry and Pharmacy > Institute of Pharmacy Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry I (Prof. Elz) | ||||
| Identification Number |
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| Keywords | PICTET-SPENGLER REACTION; ACUTE MYELOID-LEUKEMIA; 1ST GLOBAL APPROVAL; T-REGULATORY CELLS; BENZODIAZEPINE RECEPTOR; PROTEASOMAL DEGRADATION; ORGANIC-MOLECULES; HYBRID MOLECULES; FORCE-FIELD; ACID; Histone deacetylase; HDAC; Histone deacetylase inhibitor; HDACi; Tetrahydro-beta-carboline; Histone deacetylase 6 inhibition assay | ||||
| Dewey Decimal Classification | 500 Science > 540 Chemistry & allied sciences | ||||
| Status | Published | ||||
| Refereed | Yes, this version has been refereed | ||||
| Created at the University of Regensburg | Yes | ||||
| Item ID | 47181 |
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