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Dimeric argininamide-type neuropeptide Y receptor antagonists: chiral discrimination between Y1 and Y4 receptors

Keller, Max, Kaske, Melanie, Holzammer, Tobias, Bernhardt, Günther and Buschauer, Armin (2013) Dimeric argininamide-type neuropeptide Y receptor antagonists: chiral discrimination between Y1 and Y4 receptors. Bioorganic and Medicinal Chemistry 21 (21), pp. 6303-6322.

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Abstract

The structurally related peptides neuropeptide Y (NPY), peptide YY (PYY) and pancreatic polypeptide (PP) are endogenous agonists of the NPY receptor (YR) family, which in humans comprises four functionally expressed subtypes, designated Y1R, Y2R, Y4R and Y5R. Non-peptide antagonists with high affinity and selectivity have been described for the Y1R, Y2R and Y5R, but such compounds are still ...

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Item type:Article
Date:7 September 2013
Institutions:Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer)
Projects:GRK 1910, Graduiertenkolleg "Medicinal Chemistry of Selective GPCR Ligands", GRK 760, Graduiertenkolleg Medizinische Chemie
Identification Number:
ValueType
10.1016/j.bmc.2013.08.065DOI
24074877PubMed ID
Related URLs:
URLURL Type
http://www.sciencedirect.com/science/article/pii/S0968089613007682#MMCvFirstSupplementary Material
Keywords:neuropeptide Y, NPY Y1 receptor antagonist, Y4 receptor antagonist, bivalent ligand, dimeric argininamide derivatives
Dewey Decimal Classification:500 Science > 540 Chemistry & allied sciences
600 Technology > 615 Pharmacy
Status:Published
Refereed:Yes, this version has been refereed
Created at the University of Regensburg:Yes
Item ID:28432
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