N(omega)-carbamoylation of the argininamide moiety: an avenue to insurmountable NPY Y1 receptor antagonists and a radiolabeled selective high affinity molecular tool ([3H]UR-MK299) with extended residence time
Keller, Max, Weiss, Stefan, Hutzler, Christoph
, Kuhn, Kilian K., Mollereau, Catherine , Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Günther, König, Burkhard and Buschauer, Armin
(2015)
N(omega)-carbamoylation of the argininamide moiety: an avenue to insurmountable NPY Y1 receptor antagonists and a radiolabeled selective high affinity molecular tool ([3H]UR-MK299) with extended residence time.
Journal of Medicinal Chemistry 58 (22), pp. 8834-8849.
Date of publication of this fulltext: 19 Oct 2015 10:30
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| Item type | Article | ||||||
| Journal or Publication Title | Journal of Medicinal Chemistry | ||||||
| Publisher: | AMER CHEMICAL SOC | ||||||
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| Place of Publication: | WASHINGTON | ||||||
| Volume: | 58 | ||||||
| Number of Issue or Book Chapter: | 22 | ||||||
| Page Range: | pp. 8834-8849 | ||||||
| Date | 2015 | ||||||
| Institutions | Chemistry and Pharmacy > Institute of Pharmacy Chemistry and Pharmacy > Institut für Organische Chemie > Lehrstuhl Prof. Dr. Burkhard König | ||||||
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| Keywords | ACYLGUANIDINE BIOISOSTERIC APPROACH; NEUROPEPTIDE-Y; CANCER; POTENT; RADIOLIGAND; INHIBITION; LIGANDS; DESIGN; CELLS; | ||||||
| Dewey Decimal Classification | 600 Technology > 615 Pharmacy 600 Technology > 615 Pharmacy | ||||||
| Status | Published | ||||||
| Refereed | Yes, this version has been refereed | ||||||
| Created at the University of Regensburg | Yes | ||||||
| Item ID | 31955 |
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