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Sellmer, Andreas ; Pilsl, Bernadette ; Beyer, Mandy ; Pongratz, Herwig ; Wirth, Lukas ; Elz, Sigurd ; Dove, Stefan ; Henninger, Sven Julian ; Spiekermann, Karsten ; Polzer, Harald ; Klaeger, Susan ; Kuster, Bernhard ; Böhmer, Frank D. ; Fiebig, Heinz-Herbert ; Krämer, Oliver H. ; Mahboobi, Siavosh

A series of novel aryl-methanone derivatives as inhibitors of FMS-like tyrosine kinase 3 (FLT3) in FLT3-ITD-positive acute myeloid leukemia

Article

Sellmer, Andreas, Pilsl, Bernadette, Beyer, Mandy, Pongratz, Herwig, Wirth, Lukas, Elz, Sigurd, Dove, Stefan, Henninger, Sven Julian, Spiekermann, Karsten, Polzer, Harald, Klaeger, Susan, Kuster, Bernhard, Böhmer, Frank D., Fiebig, Heinz-Herbert, Krämer, Oliver H. and Mahboobi, Siavosh (2020) A series of novel aryl-methanone derivatives as inhibitors of FMS-like tyrosine kinase 3 (FLT3) in FLT3-ITD-positive acute myeloid leukemia. European Journal of Medicinal Chemistry 193, p. 112232.



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Details

Item typeArticle
Journal or Publication TitleEuropean Journal of Medicinal Chemistry
PublisherELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER
Place of PublicationISSY-LES-MOULINEAUX
Volume193
Page Rangep. 112232
Date2020
Date of publication11 Oct 2021 12:51
InstitutionsChemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry I (Prof. Elz)
Identification Number
ValueType
10.1016/j.ejmech.2020.112232DOI
KeywordsINTERNAL TANDEM DUPLICATION; THERAPEUTIC TARGET; F691L MUTATION; IN-VITRO; AML; RESISTANCE; CRENOLANIB; POTENT; CELLS; VALIDATION; FLT3; FLT3-ITD; FLT3 D835Y; Tyrosine kinase inhibitor; Acute myeloid leukemia
Dewey Decimal Classification600 Technology > 615 Pharmacy
StatusPublished
RefereedYes, this version has been refereed
Created at the University of RegensburgYes
Item ID50072

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