Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties
Article
Szczepańska, Katarzyna, Podlewska, Sabina, Dichiara, Maria, Gentile, Davide, Patamia, Vincenzo, Rosier, Niklas, Mönnich, Denise, Ruiz Cantero, Ma Carmen, Karcz, Tadeusz, Łażewska, Dorota, Siwek, Agata, Pockes, Steffen, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Rescifina, Antonio, Bojarski, Andrzej J., Amata, Emanuele and Kieć-Kononowicz, Katarzyna (2022) Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties. ACS Chemical Neuroscience 13 (1), pp. 1-15.Alternative links to fulltext
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| Item type | Article | ||||
| Journal or Publication Title | ACS Chemical Neuroscience | ||||
| Publisher | AMER CHEMICAL SOC | ||||
| Place of Publication | WASHINGTON | ||||
| Volume | 13 | ||||
| Number of Issue or Book Chapter | 1 | ||||
| Page Range | pp. 1-15 | ||||
| Date | 2022 | ||||
| Date of publication | 29 Feb 2024 12:42 | ||||
| Institutions | Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry I (Prof. Elz) | ||||
| Identification Number |
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| Keywords | DIRECTED LIGANDS; INHIBITION; TARGET; POTENT; IDENTIFICATION; OPTIMIZATION; THERAPEUTICS; INVOLVEMENT; AGONISTS; BINDING; histamine H-3 receptor; sigma-1 receptor; sigma-2 receptor; piperazine derivatives; piperidine derivatives; dual targeting compounds; molecular docking; dynamics; functional characterization | ||||
| Dewey Decimal Classification | 600 Technology > 615 Pharmacy | ||||
| Status | Published | ||||
| Refereed | Yes, this version has been refereed | ||||
| Created at the University of Regensburg | Yes | ||||
| Item ID | 56903 |
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