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Grätz, Lukas, Müller, Christoph, Pegoli, Andrea
, Schindler, Lisa, Bernhardt, Günther
und Littmann, Timo
(2022)
Insertion of Nanoluc into the Extracellular Loops as a Complementary Method To Establish BRET-Based Binding Assays for GPCRs.
ACS Pharmacology & Translational Science 5 (11), S. 1142-1155.
, Gruber, Corinna G., Pegoli, Andrea, Tahk, Maris-Johanna, Tsernant, Mari-Liis, Keller, Max und Rinken, Ago
(2021)
BRET- and fluorescence anisotropy-based assays for real-time monitoring of ligand binding to M2 muscarinic acetylcholine receptors.
Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1868 (3), S. 118930.
Volltext nicht vorhanden.
Pegoli, Andrea
(2020)
Dibenzodiazepinone-type mAChR ligands: radio- and fluorescence labeling enable unveiling of dualsteric M₂R binding and conjugation to short peptides as an avenue to highly selective M₂R ligands.
Dissertation, Universität Regensburg.
und Holliday, Nicholas D.
(2020)
Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
ACS Medicinal Chemistry Letters 11 (1), S. 16-22.
Volltext nicht vorhanden.
, Carpenter, Jessica, Hübner, Harald, Chen, Mengya, Wan, Jianfei, Bernhardt, Günther, Gmeiner, Peter
, Holliday, Nicholas D.
und Keller, Max
(2020)
Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M2 Receptor.
Journal of Medicinal Chemistry 63 (8), S. 4133-4154.
Volltext nicht vorhanden.
, Gruber, Corinna G., Xueke, She, Hübner, Harald, Bernhardt, Günther, Gmeiner, Peter
und Keller, Max
(2019)
Conjugation of Short Peptides to Dibenzodiazepinone-Type
She, Xueke, Pegoli, Andrea, Mayr, Judith, Hübner, Harald, Bernhardt, Günther
, Gmeiner, Peter und Keller, Max
(2017)
Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity.
ACS Omega 2 (10), S. 6741-6754.
, She, Xueke, Wifling, David
, Hübner, Harald, Bernhardt, Günther, Gmeiner, Peter
und Keller, Max
(2017)
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.
Journal of Medicinal Chemistry 60 (8), S. 3314-3334.
Volltext nicht vorhanden.
, Bernhardt, Günther, Buschauer, Armin und Read, Roger W.
(2015)
M2 subtype preferring dibenzodiazepinone-type muscarinic receptor ligands: effect of chemical homo-dimerization on orthosteric (and allosteric?) binding.
Bioorganic & Medicinal Chemistry 23 (14), S. 3970-3990.
Volltext nicht vorhanden.
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