Number of items: 9.
2022
Grätz, Lukas,
Müller, Christoph,
Pegoli, Andrea 
,
Schindler, Lisa,
Bernhardt, Günther 
and
Littmann, Timo
(2022)
Insertion of Nanoluc into the Extracellular Loops as a Complementary Method To Establish BRET-Based Binding Assays for GPCRs.
ACS Pharmacology & Translational Science 5 (11), pp. 1142-1155.
2020
Gruber, Corinna G.,
Pegoli, Andrea,
Müller, Christoph,
Grätz, Lukas,
She, Xueke and
Keller, Max
(2020)
Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity.
RSC Medicinal Chemistry 11 (7), pp. 823-832.
Fulltext not available.
Keller, Max,
Mahuroof, Shahani A.,
Hong Yee, Vivyanne,
Carpenter, Jessica,
Schindler, Lisa,
Littmann, Timo,
Pegoli, Andrea,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter 
and
Holliday, Nicholas D. 
(2020)
Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
ACS Medicinal Chemistry Letters 11 (1), pp. 16-22.
Fulltext not available.
She, Xueke,
Pegoli, Andrea,
Gruber, Corinna G.,
Wifling, David 
,
Carpenter, Jessica,
Hübner, Harald,
Chen, Mengya,
Wan, Jianfei,
Bernhardt, Günther,
Gmeiner, Peter 
,
Holliday, Nicholas D. 
and
Keller, Max
(2020)
Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M2 Receptor.
Journal of Medicinal Chemistry 63 (8), pp. 4133-4154.
Fulltext not available.
2019
Pegoli, Andrea,
Wifling, David 
,
Gruber, Corinna G.,
Xueke, She,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter 
and
Keller, Max
(2019)
Conjugation of Short Peptides to Dibenzodiazepinone-Type
Muscarinic Acetylcholine Receptor Ligands Determines M2R
Selectivity.
Journal of Medicinal Chemistry 62, pp. 5358-5369.
Fulltext not available.
2017
She, Xueke,
Pegoli, Andrea,
Mayr, Judith,
Hübner, Harald,
Bernhardt, Günther 
,
Gmeiner, Peter and
Keller, Max 
(2017)
Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity.
ACS Omega 2 (10), pp. 6741-6754.
Pegoli, Andrea 
,
She, Xueke,
Wifling, David 
,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter 
and
Keller, Max
(2017)
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.
Journal of Medicinal Chemistry 60 (8), pp. 3314-3334.
Fulltext not available.
2015
Keller, Max,
Tränkle, Christian,
She, Xueke,
Pegoli, Andrea,
Bernhardt, Günther,
Buschauer, Armin and
Read, Roger W.
(2015)
M2 subtype preferring dibenzodiazepinone-type muscarinic receptor ligands: effect of chemical homo-dimerization on orthosteric (and allosteric?) binding.
Bioorganic & Medicinal Chemistry 23 (14), pp. 3970-3990.
Fulltext not available.
This list was generated on Thu Nov 30 07:51:54 2023 CET.