Anzahl der Einträge: 10.
2022
Grätz, Lukas,
Müller, Christoph,
Pegoli, Andrea ,
Schindler, Lisa,
Bernhardt, Günther und
Littmann, Timo
(2022)
Insertion of Nanoluc into the Extracellular Loops as a Complementary Method To Establish BRET-Based Binding Assays for GPCRs.
ACS Pharmacology & Translational Science 5 (11), S. 1142-1155.
2021
Grätz, Lukas,
Laasfeld, Tõnis,
Allikalt, Anni ,
Gruber, Corinna G.,
Pegoli, Andrea,
Tahk, Maris-Johanna,
Tsernant, Mari-Liis,
Keller, Max und
Rinken, Ago
(2021)
BRET- and fluorescence anisotropy-based assays for real-time monitoring of ligand binding to M2 muscarinic acetylcholine receptors.
Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1868 (3), S. 118930.
Volltext nicht vorhanden.
2020
Gruber, Corinna G.,
Pegoli, Andrea,
Müller, Christoph,
Grätz, Lukas,
She, Xueke und
Keller, Max
(2020)
Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity.
RSC Medicinal Chemistry 11 (7), S. 823-832.
Volltext nicht vorhanden.
Keller, Max,
Mahuroof, Shahani A.,
Hong Yee, Vivyanne,
Carpenter, Jessica,
Schindler, Lisa,
Littmann, Timo,
Pegoli, Andrea,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter und
Holliday, Nicholas D.
(2020)
Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
ACS Medicinal Chemistry Letters 11 (1), S. 16-22.
Volltext nicht vorhanden.
She, Xueke,
Pegoli, Andrea,
Gruber, Corinna G.,
Wifling, David ,
Carpenter, Jessica,
Hübner, Harald,
Chen, Mengya,
Wan, Jianfei,
Bernhardt, Günther,
Gmeiner, Peter ,
Holliday, Nicholas D. und
Keller, Max
(2020)
Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M2 Receptor.
Journal of Medicinal Chemistry 63 (8), S. 4133-4154.
Volltext nicht vorhanden.
2019
Pegoli, Andrea,
Wifling, David ,
Gruber, Corinna G.,
Xueke, She,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter und
Keller, Max
(2019)
Conjugation of Short Peptides to Dibenzodiazepinone-Type
Muscarinic Acetylcholine Receptor Ligands Determines M2R
Selectivity.
Journal of Medicinal Chemistry 62, S. 5358-5369.
Volltext nicht vorhanden.
2017
She, Xueke,
Pegoli, Andrea,
Mayr, Judith,
Hübner, Harald,
Bernhardt, Günther ,
Gmeiner, Peter und
Keller, Max
(2017)
Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity.
ACS Omega 2 (10), S. 6741-6754.
Pegoli, Andrea ,
She, Xueke,
Wifling, David ,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter und
Keller, Max
(2017)
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.
Journal of Medicinal Chemistry 60 (8), S. 3314-3334.
Volltext nicht vorhanden.
2015
Keller, Max,
Tränkle, Christian,
She, Xueke,
Pegoli, Andrea ,
Bernhardt, Günther,
Buschauer, Armin und
Read, Roger W.
(2015)
M2 subtype preferring dibenzodiazepinone-type muscarinic receptor ligands: effect of chemical homo-dimerization on orthosteric (and allosteric?) binding.
Bioorganic & Medicinal Chemistry 23 (14), S. 3970-3990.
Volltext nicht vorhanden.
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