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Publikationen von Grätz, Lukas
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Anzahl der Einträge: 13.
2023
Grätz, Lukas
(2023)
Luminescence-based methods for the investigation of ligand binding and GRK2 recruitment to GPCRs.
Dissertation, Universität Regensburg.
2022
Grätz, Lukas, Müller, Christoph, Pegoli, Andrea 
, Schindler, Lisa, Bernhardt, Günther und Littmann, Timo
(2022)
Insertion of Nanoluc into the Extracellular Loops as a Complementary Method To Establish BRET-Based Binding Assays for GPCRs.
ACS Pharmacology & Translational Science 5 (11), S. 1142-1155.
Schindler, Lisa, Moosbauer, Jutta, Schmidt, Daniel , Spruss, Thilo, Grätz, Lukas, Lüdeke, Steffen, Hofheinz, Frank, Meister, Sebastian, Echtenacher, Bernd, Bernhardt, Günther, Pietzsch, Jens , Hellwig, Dirk und Keller, Max
(2022)
Development of a Neurotensin-Derived 68Ga-Labeled PET Ligand with High In Vivo Stability for Imaging of NTS1 Receptor-Expressing Tumors.
Cancers 14 (19), S. 4922.
Tahk, Maris-Johanna , Torp, Jane , Ali, Mohammed A. S. , Fishman, Dmytro, Parts, Leopold , Grätz, Lukas , Müller, Christoph , Keller, Max , Veiksina, Santa , Laasfeld, Tõnis und Rinken, Ago
(2022)
Live-cell microscopy or fluorescence anisotropy with budded baculoviruses—which way to go with measuring ligand binding to M 4 muscarinic receptors?
Open Biology 12 (6).
Volltext nicht vorhanden.
, Torp, Jane , Ali, Mohammed A. S. , Fishman, Dmytro, Parts, Leopold , Grätz, Lukas , Müller, Christoph , Keller, Max , Veiksina, Santa , Laasfeld, Tõnis und Rinken, Ago
(2022)
Live-cell microscopy or fluorescence anisotropy with budded baculoviruses—which way to go with measuring ligand binding to M 4 muscarinic receptors?
Open Biology 12 (6).
Volltext nicht vorhanden.
Andreev, Stanislav, Pantsar, Tatu, Tesch, Roberta, Kahlke, Niclas, El-Gokha, Ahmed, Ansideri, Francesco, Grätz, Lukas, Romasco, Jenny, Sita, Giulia, Geibel, Christian , Lämmerhofer, Michael, Tarozzi, Andrea, Knapp, Stefan , Laufer, Stefan A. und Koch, Pierre
(2022)
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3β Inhibitors.
Journal of Medicinal Chemistry 65 (2), S. 1283-1301.
Volltext nicht vorhanden.
, Lämmerhofer, Michael, Tarozzi, Andrea, Knapp, Stefan , Laufer, Stefan A. und Koch, Pierre
(2022)
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3β Inhibitors.
Journal of Medicinal Chemistry 65 (2), S. 1283-1301.
Volltext nicht vorhanden.
2021
Rosier, Niklas, Grätz, Lukas, Schihada, Hannes , Möller, Jan, Işbilir, Ali , Humphrys, Laura J. , Nagl, Martin, Seibel, Ulla, Lohse, Martin J. und Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), S. 11695-11708.
Volltext nicht vorhanden.
, Möller, Jan, Işbilir, Ali , Humphrys, Laura J. , Nagl, Martin, Seibel, Ulla, Lohse, Martin J. und Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), S. 11695-11708.
Volltext nicht vorhanden.
Grätz, Lukas, Laasfeld, Tõnis, Allikalt, Anni , Gruber, Corinna G., Pegoli, Andrea, Tahk, Maris-Johanna, Tsernant, Mari-Liis, Keller, Max und Rinken, Ago
(2021)
BRET- and fluorescence anisotropy-based assays for real-time monitoring of ligand binding to M2 muscarinic acetylcholine receptors.
Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1868 (3), S. 118930.
Volltext nicht vorhanden.
, Gruber, Corinna G., Pegoli, Andrea, Tahk, Maris-Johanna, Tsernant, Mari-Liis, Keller, Max und Rinken, Ago
(2021)
BRET- and fluorescence anisotropy-based assays for real-time monitoring of ligand binding to M2 muscarinic acetylcholine receptors.
Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1868 (3), S. 118930.
Volltext nicht vorhanden.
Konieczny, Adam, Conrad, Marcus, Ertl, Fabian J., Gleixner, Jakob, Gattor, Albert O., Grätz, Lukas, Schmidt, Maximilian F., Neu, Eduard, Horn, Anselm H. C., Wifling, David, Gmeiner, Peter, Clark, Timothy, Sticht, Heinrich und Keller, Max
(2021)
N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y4 Receptor Ligands Results in Picomolar Binding Constants.
Journal of Medicinal Chemistry 64 (22), S. 16746-16769.
Volltext nicht vorhanden.
2020
Höring, Carina , Seibel, Ulla , Tropmann, Katharina, Grätz, Lukas , Mönnich, Denise , Pitzl, Sebastian, Bernhardt, Günther , Pockes, Steffen und Strasser, Andrea
(2020)
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.
International Journal of Molecular Sciences 21 (22), S. 8440.
Grätz, Lukas, Tropmann, Katharina, Bresinsky, Merlin, Müller, Christoph, Bernhardt, Günther und Pockes, Steffen
(2020)
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells.
Scientific Reports 10, S. 13288.
Forster, Lisa , Grätz, Lukas, Mönnich, Denise, Bernhardt, Günther und Pockes, Steffen
(2020)
A Split Luciferase Complementation Assay for the Quantification of β-Arrestin2 Recruitment to Dopamine D2-Like Receptors.
International Journal of Molecular Sciences 21 (17), S. 6103.
Bartole, Edith, Grätz, Lukas, Littmann, Timo, Wifling, David , Seibel, Ulla, Buschauer, Armin und Bernhardt, Günther
(2020)
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors.
Journal of Medicinal Chemistry 63 (10), S. 5297-5311.
Volltext nicht vorhanden.
, Seibel, Ulla, Buschauer, Armin und Bernhardt, Günther
(2020)
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors.
Journal of Medicinal Chemistry 63 (10), S. 5297-5311.
Volltext nicht vorhanden.
Gruber, Corinna G., Pegoli, Andrea, Müller, Christoph, Grätz, Lukas, She, Xueke und Keller, Max
(2020)
Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity.
RSC Medicinal Chemistry 11 (7), S. 823-832.
Volltext nicht vorhanden.
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