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Publikationen von Pockes, Steffen
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Anzahl der Einträge: 25.
2023
Nagl, Martin, Moennich, Denise, Rosier, Niklas 
, Schihada, Hannes, Sirbu, Alexei, Konar, Nergis, Reyes-Resina, Irene, Navarro, Gemma, Franco, Rafael, Kolb, Peter, Annibale, Paolo und Pockes, Steffen
(2023)
Fluorescent Tools for the Imaging of Dopamine D2‐Like Receptors.
ChemBioChem.
Rosier, Niklas , Moennich, Denise, Nagl, Martin, Schihada, Hannes, Sirbu, Alexei, Konar, Nergis, Reyes-Resina, Irene, Navarro, Gemma, Franco, Rafael, Kolb, Peter, Annibale, Paolo und Pockes, Steffen
(2023)
Shedding Light on the D1‐Like Receptors: A Fluorescence‐Based Toolbox for Visualization of the D1 and D5 Receptors.
ChemBioChem.
2022
Forster, Lisa und Pockes, Steffen
(2022)
Investigating the ligand agonism and antagonism at the D2long receptor by dynamic mass redistribution.
Scientific Reports 12 (1).
Bresinsky, Merlin, Strasser, Jessica M., Hubmann, Alexander, Vallaster, Bernadette, McCue, William M., Fuller, Jessica, Singh, Gurpreet, Nelson, Kathryn M., Cuellar, Matthew E., Finzel, Barry C., Ashe, Karen H., Walters, Michael A. und Pockes, Steffen
(2022)
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis.
Archiv der Pharmazie 355 (9), S. 2200095.
Singh, Gurpreet, Liu, Peng, Yao, Katherine R., Strasser, Jessica M., Hlynialuk, Chris, Leinonen-Wright, Kailee, Teravskis, Peter J., Choquette, Jessica M., Ikramuddin, Junaid, Bresinsky, Merlin, Nelson, Kathryn M., Liao, Dezhi, Ashe, Karen H., Walters, Michael A. und Pockes, Steffen
(2022)
Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy.
ACS Chemical Neuroscience 13 (10), S. 1549-1557.
Volltext nicht vorhanden.
Szczepańska, Katarzyna, Podlewska, Sabina, Dichiara, Maria, Gentile, Davide, Patamia, Vincenzo, Rosier, Niklas, Mönnich, Denise, Ruiz Cantero, Ma Carmen, Karcz, Tadeusz, Łażewska, Dorota, Siwek, Agata, Pockes, Steffen, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Rescifina, Antonio, Bojarski, Andrzej J., Amata, Emanuele und Kieć-Kononowicz, Katarzyna
(2022)
Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties.
ACS Chemical Neuroscience 13 (1), S. 1-15.
Volltext nicht vorhanden.
2021
Pockes, Steffen und Tropmann, Katharina
(2021)
Histamine H2 receptor radioligands: triumphs and challenges.
Future Medicinal Chemistry 13 (12), S. 1073-1081.
Rosier, Niklas, Grätz, Lukas, Schihada, Hannes , Möller, Jan, Işbilir, Ali , Humphrys, Laura J. , Nagl, Martin, Seibel, Ulla, Lohse, Martin J. und Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), S. 11695-11708.
Volltext nicht vorhanden.
, Möller, Jan, Işbilir, Ali , Humphrys, Laura J. , Nagl, Martin, Seibel, Ulla, Lohse, Martin J. und Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), S. 11695-11708.
Volltext nicht vorhanden.
Tropmann, Katharina, Bresinsky, Merlin, Forster, Lisa, Mönnich, Denise, Buschauer, Armin , Wittmann, Hans-Joachim, Hübner, Harald, Gmeiner, Peter, Pockes, Steffen und Strasser, Andrea
(2021)
Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists.
Journal of Medicinal Chemistry 64 (12), S. 8684-8709.
Volltext nicht vorhanden.
, Wittmann, Hans-Joachim, Hübner, Harald, Gmeiner, Peter, Pockes, Steffen und Strasser, Andrea
(2021)
Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists.
Journal of Medicinal Chemistry 64 (12), S. 8684-8709.
Volltext nicht vorhanden.
Gergs, Ulrich, Büxel, Maren L., Bresinsky, Merlin, Kirchhefer, Uwe, Fehse, Charlotte, Höring, Carina, Hofmann, Britt, Marušáková, Margaréta, Čináková, Aneta, Schwarz, Rebecca, Pockes, Steffen und Neumann, Joachim
(2021)
Cardiac Effects of Novel Histamine H2 Receptor Agonists.
Journal of Pharmacology and Experimental Therapeutics 379 (3), S. 223-234.
Volltext nicht vorhanden.
und Neumann, Joachim
(2021)
Cardiac Effects of Novel Histamine H2 Receptor Agonists.
Journal of Pharmacology and Experimental Therapeutics 379 (3), S. 223-234.
Volltext nicht vorhanden.
Biselli, Sabrina, Bresinsky, Merlin, Tropmann, Katharina, Forster, Lisa , Honisch, Claudia , Buschauer, Armin, Bernhardt, Günther und Pockes, Steffen
(2021)
Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H2R and D3R.
European Journal of Medicinal Chemistry 214, S. 113190.
Volltext nicht vorhanden.
, Honisch, Claudia , Buschauer, Armin, Bernhardt, Günther und Pockes, Steffen
(2021)
Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H2R and D3R.
European Journal of Medicinal Chemistry 214, S. 113190.
Volltext nicht vorhanden.
Szczepańska, Katarzyna , Pockes, Steffen , Podlewska, Sabina, Höring, Carina, Mika, Kamil, Latacz, Gniewomir, Bednarski, Marek, Siwek, Agata , Karcz, Tadeusz, Nagl, Martin, Bresinsky, Merlin, Mönnich, Denise, Seibel, Ulla, Kuder, Kamil J. , Kotańska, Magdalena, Stark, Holger, Elz, Sigurd und Kieć-Kononowicz, Katarzyna
(2021)
Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent.
European Journal of Medicinal Chemistry 213, S. 113041.
Volltext nicht vorhanden.
, Pockes, Steffen , Podlewska, Sabina, Höring, Carina, Mika, Kamil, Latacz, Gniewomir, Bednarski, Marek, Siwek, Agata , Karcz, Tadeusz, Nagl, Martin, Bresinsky, Merlin, Mönnich, Denise, Seibel, Ulla, Kuder, Kamil J. , Kotańska, Magdalena, Stark, Holger, Elz, Sigurd und Kieć-Kononowicz, Katarzyna
(2021)
Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent.
European Journal of Medicinal Chemistry 213, S. 113041.
Volltext nicht vorhanden.
2020
Höring, Carina , Seibel, Ulla , Tropmann, Katharina, Grätz, Lukas , Mönnich, Denise , Pitzl, Sebastian, Bernhardt, Günther , Pockes, Steffen und Strasser, Andrea
(2020)
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.
International Journal of Molecular Sciences 21 (22), S. 8440.
Grätz, Lukas, Tropmann, Katharina, Bresinsky, Merlin, Müller, Christoph, Bernhardt, Günther und Pockes, Steffen
(2020)
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells.
Scientific Reports 10, S. 13288.
Forster, Lisa , Grätz, Lukas, Mönnich, Denise, Bernhardt, Günther und Pockes, Steffen
(2020)
A Split Luciferase Complementation Assay for the Quantification of β-Arrestin2 Recruitment to Dopamine D2-Like Receptors.
International Journal of Molecular Sciences 21 (17), S. 6103.
Schihada, Hannes , Ma, Xiaoyuan, Zabel, Ulrike, Vischer, Henry F., Schulte, Gunnar , Leurs, Rob, Pockes, Steffen und Lohse, Martin J.
(2020)
Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists.
ACS Sensors 5 (6), S. 1734-1742.
Volltext nicht vorhanden.
, Ma, Xiaoyuan, Zabel, Ulrike, Vischer, Henry F., Schulte, Gunnar , Leurs, Rob, Pockes, Steffen und Lohse, Martin J.
(2020)
Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists.
ACS Sensors 5 (6), S. 1734-1742.
Volltext nicht vorhanden.
Tropmann, Katharina, Höring, Carina , Plank, Nicole und Pockes, Steffen
(2020)
Discovery of a G Protein-Biased Radioligand for the Histamine H2 Receptor with Reversible Binding Properties.
Journal of Medicinal Chemistry 63 (21), S. 13090-13102.
Volltext nicht vorhanden.
, Plank, Nicole und Pockes, Steffen
(2020)
Discovery of a G Protein-Biased Radioligand for the Histamine H2 Receptor with Reversible Binding Properties.
Journal of Medicinal Chemistry 63 (21), S. 13090-13102.
Volltext nicht vorhanden.
2019
Pockes, Steffen, Wifling, David , Buschauer, Armin und Elz, Sigurd
(2019)
Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands †.
ChemistryOpen 8 (3), S. 285-297.
Rustler, Karin , Pockes, Steffen und König, Burkhard
(2019)
Light-Switchable Antagonists for the Histamine H1 Receptor at the Isolated Guinea Pig Ileum.
ChemMedChem 14 (6), S. 636-644.
Volltext nicht vorhanden.
, Pockes, Steffen und König, Burkhard
(2019)
Light-Switchable Antagonists for the Histamine H1 Receptor at the Isolated Guinea Pig Ileum.
ChemMedChem 14 (6), S. 636-644.
Volltext nicht vorhanden.
Rustler, Karin , Pockes, Steffen und König, Burkhard
(2019)
Cover Feature: Light‐Switchable Antagonists for the Histamine H 1 Receptor at the Isolated Guinea Pig Ileum (ChemMedChem 6/2019).
ChemMedChem 14 (6), S. 614.
Volltext nicht vorhanden.
, Pockes, Steffen und König, Burkhard
(2019)
Cover Feature: Light‐Switchable Antagonists for the Histamine H 1 Receptor at the Isolated Guinea Pig Ileum (ChemMedChem 6/2019).
ChemMedChem 14 (6), S. 614.
Volltext nicht vorhanden.
Soliman, Beatrice, Wang, Ning, Zagotto, Giuseppe und Pockes, Steffen
(2019)
Synthesis and biological evaluation of heteroalicyclic cyanoguanidines at histamine receptors.
Archiv der Pharmazie 352 (9), S. 1900107.
Volltext nicht vorhanden.
(2019)
Synthesis and biological evaluation of heteroalicyclic cyanoguanidines at histamine receptors.
Archiv der Pharmazie 352 (9), S. 1900107.
Volltext nicht vorhanden.
2018
Pockes, Steffen , Wifling, David , Keller, Max, Buschauer, Armin und Elz, Sigurd
(2018)
Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists.
ACS Omega 2018 (3), S. 2865-2882.
Pockes, Steffen
(2018)
Synthese und pharmakologische Charakterisierung von Heteroarylpropylguanidin-Derivaten an Histamin-Rezeptorsubtypen: Struktur-Wirkungsbeziehungen mono- und bivalenter Liganden.
Dissertation, Universität Regensburg.
2016
Sadek, Bassem, Khan, Nadia, Darras, Fouad H., Pockes, Steffen und Decker, Michael
(2016)
The dual-acting AChE inhibitor and H3 receptor antagonist UW-MD-72 reverses amnesia induced by scopolamine or dizocilpine in passive avoidance paradigm in rats.
Physiology & Behavior 165, S. 383-391.
Volltext nicht vorhanden.
und Decker, Michael
(2016)
The dual-acting AChE inhibitor and H3 receptor antagonist UW-MD-72 reverses amnesia induced by scopolamine or dizocilpine in passive avoidance paradigm in rats.
Physiology & Behavior 165, S. 383-391.
Volltext nicht vorhanden.
2014
Darras, Fouad, Pockes, Steffen , Huang, Guozheng, Wehle, Sarah, Strasser, Andrea, Wittmann, Hans-Joachim, Nimczick, Martin, Sotriffer, Christoph und Decker, Michael
(2014)
Synthesis, biological evaluation, and computational studies of tri- and tetracyclic nitrogen-bridgehead compounds as potent dual-acting AChE inhibitors and hH3 receptor antagonists.
ACS Chemical Neuroscience 5 (3), S. 225-242.
Volltext nicht vorhanden.
, Huang, Guozheng, Wehle, Sarah, Strasser, Andrea, Wittmann, Hans-Joachim, Nimczick, Martin, Sotriffer, Christoph und Decker, Michael
(2014)
Synthesis, biological evaluation, and computational studies of tri- and tetracyclic nitrogen-bridgehead compounds as potent dual-acting AChE inhibitors and hH3 receptor antagonists.
ACS Chemical Neuroscience 5 (3), S. 225-242.
Volltext nicht vorhanden.
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