Anzahl der Einträge: 26.
2024
2023
Nagl, Martin,
Moennich, Denise,
Rosier, Niklas ,
Schihada, Hannes,
Sirbu, Alexei,
Konar, Nergis,
Reyes-Resina, Irene,
Navarro, Gemma,
Franco, Rafael,
Kolb, Peter,
Annibale, Paolo und
Pockes, Steffen
(2023)
Fluorescent Tools for the Imaging of Dopamine D2‐Like Receptors.
ChemBioChem.
Rosier, Niklas ,
Moennich, Denise,
Nagl, Martin,
Schihada, Hannes,
Sirbu, Alexei,
Konar, Nergis,
Reyes-Resina, Irene,
Navarro, Gemma,
Franco, Rafael,
Kolb, Peter,
Annibale, Paolo und
Pockes, Steffen
(2023)
Shedding Light on the D1‐Like Receptors: A Fluorescence‐Based Toolbox for Visualization of the D1 and D5 Receptors.
ChemBioChem.
2022
Bresinsky, Merlin,
Strasser, Jessica M.,
Hubmann, Alexander,
Vallaster, Bernadette,
McCue, William M.,
Fuller, Jessica,
Singh, Gurpreet,
Nelson, Kathryn M.,
Cuellar, Matthew E.,
Finzel, Barry C.,
Ashe, Karen H.,
Walters, Michael A. und
Pockes, Steffen
(2022)
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis.
Archiv der Pharmazie 355 (9), S. 2200095.
Singh, Gurpreet,
Liu, Peng,
Yao, Katherine R.,
Strasser, Jessica M.,
Hlynialuk, Chris,
Leinonen-Wright, Kailee,
Teravskis, Peter J.,
Choquette, Jessica M.,
Ikramuddin, Junaid,
Bresinsky, Merlin,
Nelson, Kathryn M.,
Liao, Dezhi,
Ashe, Karen H.,
Walters, Michael A. und
Pockes, Steffen
(2022)
Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy.
ACS Chemical Neuroscience 13 (10), S. 1549-1557.
Volltext nicht vorhanden.
Szczepańska, Katarzyna,
Podlewska, Sabina,
Dichiara, Maria,
Gentile, Davide,
Patamia, Vincenzo,
Rosier, Niklas,
Mönnich, Denise,
Ruiz Cantero, Ma Carmen,
Karcz, Tadeusz,
Łażewska, Dorota,
Siwek, Agata,
Pockes, Steffen,
Cobos, Enrique J.,
Marrazzo, Agostino,
Stark, Holger,
Rescifina, Antonio,
Bojarski, Andrzej J.,
Amata, Emanuele und
Kieć-Kononowicz, Katarzyna
(2022)
Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties.
ACS Chemical Neuroscience 13 (1), S. 1-15.
Volltext nicht vorhanden.
2021
Rosier, Niklas,
Grätz, Lukas,
Schihada, Hannes ,
Möller, Jan,
Işbilir, Ali ,
Humphrys, Laura J. ,
Nagl, Martin,
Seibel, Ulla,
Lohse, Martin J. und
Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), S. 11695-11708.
Volltext nicht vorhanden.
Tropmann, Katharina,
Bresinsky, Merlin,
Forster, Lisa,
Mönnich, Denise,
Buschauer, Armin ,
Wittmann, Hans-Joachim,
Hübner, Harald,
Gmeiner, Peter,
Pockes, Steffen und
Strasser, Andrea
(2021)
Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists.
Journal of Medicinal Chemistry 64 (12), S. 8684-8709.
Volltext nicht vorhanden.
Gergs, Ulrich,
Büxel, Maren L.,
Bresinsky, Merlin,
Kirchhefer, Uwe,
Fehse, Charlotte,
Höring, Carina,
Hofmann, Britt,
Marušáková, Margaréta,
Čináková, Aneta,
Schwarz, Rebecca,
Pockes, Steffen und
Neumann, Joachim
(2021)
Cardiac Effects of Novel Histamine H2 Receptor Agonists.
Journal of Pharmacology and Experimental Therapeutics 379 (3), S. 223-234.
Volltext nicht vorhanden.
Biselli, Sabrina,
Bresinsky, Merlin,
Tropmann, Katharina,
Forster, Lisa ,
Honisch, Claudia ,
Buschauer, Armin,
Bernhardt, Günther und
Pockes, Steffen
(2021)
Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H2R and D3R.
European Journal of Medicinal Chemistry 214, S. 113190.
Volltext nicht vorhanden.
Szczepańska, Katarzyna ,
Pockes, Steffen ,
Podlewska, Sabina,
Höring, Carina,
Mika, Kamil,
Latacz, Gniewomir,
Bednarski, Marek,
Siwek, Agata ,
Karcz, Tadeusz,
Nagl, Martin,
Bresinsky, Merlin,
Mönnich, Denise,
Seibel, Ulla,
Kuder, Kamil J. ,
Kotańska, Magdalena,
Stark, Holger,
Elz, Sigurd und
Kieć-Kononowicz, Katarzyna
(2021)
Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent.
European Journal of Medicinal Chemistry 213, S. 113041.
Volltext nicht vorhanden.
2020
Höring, Carina ,
Seibel, Ulla ,
Tropmann, Katharina,
Grätz, Lukas ,
Mönnich, Denise ,
Pitzl, Sebastian,
Bernhardt, Günther ,
Pockes, Steffen und
Strasser, Andrea
(2020)
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.
International Journal of Molecular Sciences 21 (22), S. 8440.
Grätz, Lukas,
Tropmann, Katharina,
Bresinsky, Merlin,
Müller, Christoph,
Bernhardt, Günther und
Pockes, Steffen
(2020)
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells.
Scientific Reports 10, S. 13288.
Schihada, Hannes ,
Ma, Xiaoyuan,
Zabel, Ulrike,
Vischer, Henry F.,
Schulte, Gunnar ,
Leurs, Rob,
Pockes, Steffen und
Lohse, Martin J.
(2020)
Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists.
ACS Sensors 5 (6), S. 1734-1742.
Volltext nicht vorhanden.
2019
2018
Pockes, Steffen ,
Wifling, David ,
Keller, Max,
Buschauer, Armin und
Elz, Sigurd
(2018)
Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists.
ACS Omega 2018 (3), S. 2865-2882.
2016
2014
Darras, Fouad,
Pockes, Steffen ,
Huang, Guozheng,
Wehle, Sarah,
Strasser, Andrea,
Wittmann, Hans-Joachim,
Nimczick, Martin,
Sotriffer, Christoph und
Decker, Michael
(2014)
Synthesis, biological evaluation, and computational studies of tri- and tetracyclic nitrogen-bridgehead compounds as potent dual-acting AChE inhibitors and hH3 receptor antagonists.
ACS Chemical Neuroscience 5 (3), S. 225-242.
Volltext nicht vorhanden.
Diese Liste wurde erzeugt am Fri Sep 27 08:14:47 2024 CEST.