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Number of items: 161.
A
Appl, Heidrun, Holzammer, Tobias, Dove, Stefan, Haen, Ekkehard, Strasser, Andrea and Seifert, Roland
(2012)
Interactions of recombinant human histamine H₁R, H₂R, H₃R, and H₄R receptors with 34 antidepressants and antipsychotics.
Naunyn-Schmiedeberg's archives of pharmacology 385 (2), pp. 145-170.
Fulltext not available.
B
Brunskole Hummel, Irena, Kälble, Solveig, Burhenne, Heike, Reinartz, Michael T., Schwede, Frank, Buschauer, Armin and Seifert, Roland
(2013)
Dissociations in the effects of beta2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: Support for the concept of functional selectivity.
PLoS One 8 (5), e64556.
Bodensteiner, Julian, Baumeister, Paul, Geyer, Roland, Buschauer, Armin and Reiser, Oliver 
(2013)
Synthesis and pharmacological characterization of new tetrahydrofuran based compounds as conformationally constrained histamine receptor ligands.
Organic & biomolecular chemistry 11 (24), pp. 4040-4055.
Birnkammer, Tobias, Spickenreither, Anja, Brunskole, Irena, Lopuch, Miroslaw, Kagermeier, Nicole, Bernhardt, Günther, Dove, Stefan, Seifert, Roland, Elz, Sigurd and Buschauer, Armin
(2012)
The bivalent ligand approach leads to highly potent and selective acylguanidine-type histamine H2 receptor agonists.
Journal of Medicinal Chemistry 55 (3), pp. 1147-1160.
Fulltext not available.
Brunskole, Irena, Strasser, Andrea, Seifert, Roland and Buschauer, Armin
(2011)
Role of the second and third extracellular loops of the histamine H4 receptor in receptor activation.
Naunyn-Schmiedeberg's Archives of Pharmacology 384 (3), pp. 301-317.
Fulltext not available.
Braun, Stephan, Botzki, Alexander , Salmen, Sunnhild, Textor, Christian, Bernhardt, Günther, Dove, Stefan and Buschauer, Armin
(2011)
Design of benzimidazole- and benzoxazole-2-thione derivatives as inhibitors of bacterial hyaluronan lyase.
European Journal of Medicinal Chemistry 46 (9), pp. 4419-4429.
Fulltext not available.
, Salmen, Sunnhild, Textor, Christian, Bernhardt, Günther, Dove, Stefan and Buschauer, Armin
(2011)
Design of benzimidazole- and benzoxazole-2-thione derivatives as inhibitors of bacterial hyaluronan lyase.
European Journal of Medicinal Chemistry 46 (9), pp. 4419-4429.
Fulltext not available.
Brennauer, Albert, Keller, Max, Freund, Matthias, Bernhardt, Günther and Buschauer, Armin
(2007)
Decomposition of 1-(w-aminoalkanoyl)guanidines under alkaline conditions.
Tetrahedron Letters 48 (39), pp. 6996-6999.
Fulltext not available.
Bonauer, Christoph, Walenzyk, Thomas and König, Burkhard
(2006)
α,β-Dehydroamino Acids.
Synthesis (1), pp. 1-20.
Fulltext restricted.
Botzki, Alexander, Salmen, Sunnhild, Bernhardt, Günther, Buschauer, Armin and Dove, Stefan
(2005)
Structure-Based Design Of Bacterial Hyaluronan Lyase Inhibitors,.
QSAR & Combinatorial Science 24 (4), pp. 458-469.
Fulltext not available.
Bonauer, C. and König, B.
(2005)
Synthesis and Structure of Chiral Methoxypyrrole Amino Acids (MOPAS).
Synthesis, 2367 - 2372.
Fulltext not available.
Botzki, Alexander, Rigden, Daniel J., Braun, Stephan, Nukui, Masatoshi, Salmen, Sunnhild, Hoechstetter, Julia, Bernhardt, Günther, Dove, Stefan, Buschauer, Armin and Jedrzejas, Mark J.
(2004)
L-ascorbic acid-6-hexadecanoate, a potent hyaluronidase inhibitor: X-ray structure and molecular modeling of enzyme-inhibitor complexes.
The Journal of Biological Chemistry 279 (44), pp. 45990-45997.
Fulltext not available.
Brennauer, Albert, Dove, Stefan and Buschauer, Armin
(2004)
18. Structure-Activity Relationships of Nonpeptide Neuropeptide Y Receptor Antagonists.
In: Michel, M. C., (ed.)
Neuropeptide Y and Related Peptides.
Handbook of Experimental Pharmacology, 162 (18).
Springer, Heidelberg, pp. 505-546.
ISBN 978-3-540-40581-8.
Fulltext not available.
Bonauer, C., Zabel, M. and König, B.
(2004)
Synthesis and peptide binding properties of methoxypyrrole amino acids (MOPAS).
Org. Lett. 6, 1349 - 1352.
Fulltext not available.
D
Dove, Stefan and Buschauer, Armin
(2013)
G-Protein-gekoppelte Rezeptoren: „Sinnesorgane“ der Zellen.
Blick in die Wissenschaft 22 (28), pp. 3-9.
Fulltext not available.
Desch, Matthias, Schinner, Elisabeth, Kees, Frieder K., Hofmann, F., Seifert, Roland and Schlossmann, Jens
(2010)
Cyclic cytidine 3´,5´-monophosphate (cCMP) signals via cGMP kinase I.
FEBS Letters 584 (18), pp. 3979-3984.
Fulltext not available.
Desch, Matthias, Sigl, K., Hieke, Bernhard, Salb, Katharina, Kees, F., Bernhard, D., make_name_string expected hash reference, make_name_string expected hash reference, make_name_string expected hash reference, make_name_string expected hash reference , make_name_string expected hash reference , make_name_string expected hash reference, make_name_string expected hash reference, make_name_string expected hash reference and make_name_string expected hash reference
(2010)
IRAG determines nitric oxide- and atrial natriuretic peptide-mediated smooth muscle relaxation.
Cardiovascular Research 86 (3), pp. 496-505.
Fulltext not available.
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(2010)
IRAG determines nitric oxide- and atrial natriuretic peptide-mediated smooth muscle relaxation.
Cardiovascular Research 86 (3), pp. 496-505.
Fulltext not available.
Dirscherl, G., Schwab, M., Seufert, W. and König, Burkhard
(2009)
Enhancing the Separation of Phosphorylated Proteins in Gel Electrophoresis with Dinuclear Bispyridylmethylamine-Tyrosine-Acrylamide Complexes.
Inorg. Chim Acta 362, 537 - 542.
Fulltext not available.
and König, Burkhard
(2009)
Enhancing the Separation of Phosphorylated Proteins in Gel Electrophoresis with Dinuclear Bispyridylmethylamine-Tyrosine-Acrylamide Complexes.
Inorg. Chim Acta 362, 537 - 542.
Fulltext not available.
Dirscherl, G. and König, B.
(2008)
The Use of Solid-Phase Synthesis Techniques for the Preparation of Peptide - Metal Complex Conjugates.
Eur. J. Org. Chem., 597 - 634.
Fulltext not available.
Dirscherl, G., Knape, R., Hanson, P. and König, B.
(2007)
Solid Phase Synthesis of Metal-Complex containing Peptides.
Tetrahedron 63, 4918 – 4928.
Fulltext not available.
(2007)
Solid Phase Synthesis of Metal-Complex containing Peptides.
Tetrahedron 63, 4918 – 4928.
Fulltext not available.
Dove, Stefan, Elz, Sigurd, Seifert, Roland and Buschauer, Armin
(2004)
Structure-Activity Relationships of Histamine H_2 Receptor Ligands,.
Mini-Rev. Med. Chem. 4 (9), pp. 941-954.
Fulltext not available.
E
Ehlers, I., Maity, P., Aube, J. and König, Burkhard
(2011)
Modular Synthesis of Triazole-Containing Triaryl α-Helix Mimetics.
European Journal of Organic Chemistry, pp. 2474-2490.
Fulltext not available.
and König, Burkhard
(2011)
Modular Synthesis of Triazole-Containing Triaryl α-Helix Mimetics.
European Journal of Organic Chemistry, pp. 2474-2490.
Fulltext not available.
Egger, Michael, Maity, Prantik, Hübner, Melanie, Seifert, Roland and König, Burkhard
(2009)
Synthesis and pharmacological properties of new tetracyclic forskolin analogues.
European Journal of Organic Chemistry 2009 (21), pp. 3613-3618.
Fulltext not available.
(2009)
Synthesis and pharmacological properties of new tetracyclic forskolin analogues.
European Journal of Organic Chemistry 2009 (21), pp. 3613-3618.
Fulltext not available.
Engel, E., Ulrich, H., Vasold, R., König, B. , Landthaler, M., Süttinger, R. and Bäumler, W.
(2008)
Azo Pigment and a Basal Cell Carcinoma at the Thumb.
Dermatology 216, pp. 76-80.
Fulltext not available.
, Landthaler, M., Süttinger, R. and Bäumler, W.
(2008)
Azo Pigment and a Basal Cell Carcinoma at the Thumb.
Dermatology 216, pp. 76-80.
Fulltext not available.
Egger, M., Pellett, P., Nickl, K., Geiger, S., Graetz, S., Seifert, R., Heilmann, J. and König, B.
(2008)
Synthesis and Cannabinoid Receptor Activity of Ketoalkenes from Echinacea pallida and Non-natural Analogues.
Chem. Eur. J. 14, 10978 - 10984.
Fulltext not available.
(2008)
Synthesis and Cannabinoid Receptor Activity of Ketoalkenes from Echinacea pallida and Non-natural Analogues.
Chem. Eur. J. 14, 10978 - 10984.
Fulltext not available.
Engel, E., Spannberger, A., Vasold, R., König, B., Landthaler, M. and Bäumler, W.
(2007)
Photochemical cleavage of a tattoo pigment by UVB radiation or natural sunlight.
JDDG 5 (7), 583–589.
Fulltext not available.
Egger, Michael, Li, Xuqin, Müller, Christine, Bernhardt, Günther, Buschauer, Armin and König, Burkhard
(2007)
Tariquidar analogues: synthesis by Cu(I)-catalysed N/O–aryl coupling and inhibitory activity against the ABCB1 transporter.
European Journal of Organic Chemistry 2007 (16), pp. 2643-2649.
Fulltext not available.
(2007)
Tariquidar analogues: synthesis by Cu(I)-catalysed N/O–aryl coupling and inhibitory activity against the ABCB1 transporter.
European Journal of Organic Chemistry 2007 (16), pp. 2643-2649.
Fulltext not available.
Engel, E., Santarelli, F., Vasold, R., Ulrich, H., Maisch, T., König, B. , Landthaler, M., Gopee, N. V., Howard, P. C. and Bäumler, W.
(2006)
Establishment of an Extraction Method for the Recovery of Tattoo Pigments from Human Skin Using HPLC Diode Array Detector Technology.
Anal. Chem. 78, 6440 - 6447.
Fulltext not available.
, Landthaler, M., Gopee, N. V., Howard, P. C. and Bäumler, W.
(2006)
Establishment of an Extraction Method for the Recovery of Tattoo Pigments from Human Skin Using HPLC Diode Array Detector Technology.
Anal. Chem. 78, 6440 - 6447.
Fulltext not available.
F
Fischer, Carolin and König, Burkhard
(2011)
Palladium and copper mediated N-aryl bond formation reactions for the synthesis of biological active compounds.
Beilstein Journal of Organic Chemistry (7), pp. 59-74.
Fulltext not available.
(2011)
Palladium and copper mediated N-aryl bond formation reactions for the synthesis of biological active compounds.
Beilstein Journal of Organic Chemistry (7), pp. 59-74.
Fulltext not available.
Federwisch, G., Kleinmaier, R., Drettwan, D. and Gschwind, R. M.
(2008)
The H-Bonding Network of Acylguanidine Complexes: Combined Intermolecular 2hJH,P and 3hJN,P Scalar Couplings Provide an Insight into the Geometric Arrangement.
Journal of the American Chemical Society 130 (50), pp. 16846-16847.
Fulltext not available.
(2008)
The H-Bonding Network of Acylguanidine Complexes: Combined Intermolecular 2hJH,P and 3hJN,P Scalar Couplings Provide an Insight into the Geometric Arrangement.
Journal of the American Chemical Society 130 (50), pp. 16846-16847.
Fulltext not available.
G
Geyer, Roland, Nordemann, Uwe, Strasser, Andrea, Wittmann, Hans-Joachim and Buschauer, Armin
(2016)
Conformational restriction and enantioseparation increase potency and selectivity of cyanoguanidine-type histamine H4 receptor agonists.
Journal of Medicinal Chemistry 59 (7), pp. 3452-3470.
Fulltext not available.
Geyer, Roland, Kaske, Melanie, Baumeister, Paul and Buschauer, Armin
(2014)
Synthesis and functional characterization of imbutamine analogs as histamine H3 and H4 receptor ligands.
Archiv der Pharmazie (Weinheim, Germany) 347 (2), pp. 77-88.
Fulltext not available.
Geyer, Roland, Igel, Patrick, Kaske, Melanie, Elz, Sigurd and Buschauer, Armin
(2014)
Synthesis, SAR and selectivity of 2-acyl- and 2-cyano-1-hetarylalkyl-guanidines at the four histamine receptor subtypes: a bioisosteric approach.
MedChemComm 5 (1), pp. 72-81.
Fulltext not available.
Geyer, Roland and Buschauer, Armin
(2011)
Synthesis and histamine H3 and H4 receptor activity of conformationally restricted cyanoguanidines related to UR-PI376.
Archiv der Pharmazie 344 (12), pp. 775-785.
Fulltext not available.
Geduhn, Jens, Dove, Stefan, Shen, Yuequan, Tang, Wei-Jen , König, Burkhard and Seifert, Roland
(2011)
Bis-Halogen-Anthraniloyl-Substituted Nucleoside 5'-triphosphates as Potent and Selective Inhibitors of Bordetella pertussis CyaA.
The Journal of pharmacology and experimental therapeutics 336 (1), pp. 104-115.
Fulltext not available.
, König, Burkhard and Seifert, Roland
(2011)
Bis-Halogen-Anthraniloyl-Substituted Nucleoside 5'-triphosphates as Potent and Selective Inhibitors of Bordetella pertussis CyaA.
The Journal of pharmacology and experimental therapeutics 336 (1), pp. 104-115.
Fulltext not available.
Ghorai, Prasanta, Kraus, Anja, Birnkammer, Tobias, Geyer, Roland, Bernhardt, Günther, Dove, Stefan, Seifert, Roland, Elz, Sigurd and Buschauer, Armin
(2010)
Chiral N(G)-acylated hetarylpropylguanidine-type histamine H2 receptor agonists do not show significant stereoselectivity.
Bioorganic & Medicinal Chemistry Letters 20 (10), pp. 3173-3176.
Fulltext not available.
Geiger, Sarah, Nickl, Kathrin, Schneider, Erich H., Seifert, Roland and Heilmann, Jörg
(2010)
Establishment of recombinant cannabinoid receptor assays and characterization of several natural and synthetic ligands.
Naunyn-Schmiedebergs Archiv für Pharmakologie 382 (2), pp. 177-191.
Fulltext not available.
Grauer, Andreas, Späth, Andreas, Ma, Dawei and König, Burkhard
(2009)
Metal-catalyzed derivatization of C alpha-tetrasubstituted amino acids and their use in the synthesis of cyclic peptides.
Chemistry - An Asian Journal 4 (7), pp. 1134-1140.
Fulltext not available.
(2009)
Metal-catalyzed derivatization of C alpha-tetrasubstituted amino acids and their use in the synthesis of cyclic peptides.
Chemistry - An Asian Journal 4 (7), pp. 1134-1140.
Fulltext not available.
Grauer, Andreas and König, Burkhard
(2009)
Peptidomimetics – A versatile route to biologically active compounds.
European Journal of Organic Chemistry, pp. 5099-5111.
Fulltext not available.
Grauer, Andreas, Cabrele, C. , Zabel, M. and König, Burkhard
(2009)
Stable right- and left-handed peptide helices containing Cα-tetrasubstituted α amino acids.
The Journal of Organic Chemistry 74 (10), pp. 3718-3726.
Fulltext not available.
, Zabel, M. and König, Burkhard
(2009)
Stable right- and left-handed peptide helices containing Cα-tetrasubstituted α amino acids.
The Journal of Organic Chemistry 74 (10), pp. 3718-3726.
Fulltext not available.
Grauer, Andreas and König, Burkhard
(2009)
Synthesis of new Ca-tetrasubstituted a-amino acids.
Beilstein Journal of Organic Chemistry 5 (5).
Fulltext not available.
Ghorai, Prasanta, Kraus, Anja, Keller, Max, Götte, Carsten, Igel, Patrick, Schneider, Erich , Schnell, David, Bernhardt, Günther, Dove, Stefan, Zabel, Manfred, Elz, Sigurd, Seifert, Roland and Buschauer, Armin
(2008)
Acylguanidines as bioisosteres of guanidines: N(G)-acylated imidazolylpropylguanidines, a new class of histamine H2 receptor agonists.
Journal of Medicinal Chemistry 51 (22), pp. 7193-7204.
Fulltext not available.
, Schnell, David, Bernhardt, Günther, Dove, Stefan, Zabel, Manfred, Elz, Sigurd, Seifert, Roland and Buschauer, Armin
(2008)
Acylguanidines as bioisosteres of guanidines: N(G)-acylated imidazolylpropylguanidines, a new class of histamine H2 receptor agonists.
Journal of Medicinal Chemistry 51 (22), pp. 7193-7204.
Fulltext not available.
Grauer, A., Riechers, A., Ritter, S. and König, B.
(2008)
Synthetic Receptors for the Differentiation of Phosphorylated Peptides with Nanomolar Affinities.
Chem. Eur. J. 14, 8922 - 8927.
Fulltext not available.
(2008)
Synthetic Receptors for the Differentiation of Phosphorylated Peptides with Nanomolar Affinities.
Chem. Eur. J. 14, 8922 - 8927.
Fulltext not available.
Göttle, Martin, Dove, Stefan, Steindel, Phillip, Shen, Yuequan, Tang, Wei-Jen , Geduhn, Jens, König, Burkhard and Seifert, Roland
(2007)
Molecular Analysis of the Interaction of Bordetella pertussis Adenylyl Cyclase with Fluorescent Nucleotides.
Molecular Pharmacology 72 (3), pp. 526-535.
Gschwind, R. M.
(2005)
Residual Dipolar Couplings - AValuable NMR Parameter for Small Organic Molecules.
Angewandte Chemie International Edition 44 (30), pp. 4666-4668.
Fulltext not available.
(2005)
Residual Dipolar Couplings - AValuable NMR Parameter for Small Organic Molecules.
Angewandte Chemie International Edition 44 (30), pp. 4666-4668.
Fulltext not available.
Gschwind, R. M., Armbrüster, M. and Zubrzycki, I. Z.
(2004)
NMR detection of intermolecular NH×××OP hydrogen bonds between guanidinium protons and bisposphonate moieties in an artificial arginine receptor.
Journal of the American Chemical Society 126 (33), pp. 10228-10229.
Fulltext not available.
Gallmeier, H.-C. and König, B.
(2003)
Heteroaromatic Oligoamides with dDNA Affinity (review).
Eur. J. Org. Chem., 3473 - 3483.
Fulltext not available.
H
Hübner, Melanie, Dixit, A., Mou, T.-C., Lushington, Gerald H., Pinto, Cibele S., Gille, A. , Geduhn, Jens, König, Burkhard , Sprang, S. R. and Seifert, Roland
(2011)
Structural Basis for the High-Affinity Inhibition of Mammalian Membranous Adenylyl Cyclase by 2`,3`-O-(N-Methylanthraniloyl)-Inosine 5`-Triphosphate.
Molecular Pharmacology 80 (1), pp. 87-96.
Fulltext not available.
, Geduhn, Jens, König, Burkhard , Sprang, S. R. and Seifert, Roland
(2011)
Structural Basis for the High-Affinity Inhibition of Mammalian Membranous Adenylyl Cyclase by 2`,3`-O-(N-Methylanthraniloyl)-Inosine 5`-Triphosphate.
Molecular Pharmacology 80 (1), pp. 87-96.
Fulltext not available.
Hild, Wolfgang, Pollinger, Klaus, Caporale, Andrea , Cabrele, Chiara , Keller, Max, Pluym, Nicola , Buschauer, Armin, Rachel, Reinhard, Tessmar, Joerg , Breunig, Miriam and Goepferich, Achim
(2010)
G protein-coupled receptors function as logic gates for nanoparticle binding and cell uptake.
Proceedings of the National Academy of Sciences USA: PNAS 107 (23), pp. 10667-10672.
Fulltext not available.
, Cabrele, Chiara , Keller, Max, Pluym, Nicola , Buschauer, Armin, Rachel, Reinhard, Tessmar, Joerg , Breunig, Miriam and Goepferich, Achim
(2010)
G protein-coupled receptors function as logic gates for nanoparticle binding and cell uptake.
Proceedings of the National Academy of Sciences USA: PNAS 107 (23), pp. 10667-10672.
Fulltext not available.
Hild, Wolfgang, Pollinger, Klaus, Caporale, Andrea, Cabrele, Chiara, Breunig, Miriam, Tessmar, Joerg and Göpferich, Achim
(2009)
"Nanoparticle Delivery into Target Cells by G-Protein Coupled Receptors".
In: 36th Annual Meeting of Controlled release Society, 18. - 22. Juli 2009, Kopenhagen, Dänemark.
Fulltext not available.
Hofinger, Edith S. A., Hoechstetter, Julia, Oettl, Martin, Bernhardt, Günther and Buschauer, Armin
(2008)
Isoenzyme-specific differences in the degradation of hyaluronic acid by mammalian-type hyaluronidases.
Glycoconjugate Journal 25 (2), pp. 101-109.
Fulltext not available.
Hild, Wolfgang, Pollinger, Klaus, Caporale, Andrea, Cabrele, Chiara, Breunig, Miriam, Tessmar, Joerg and Goepferich, Achim
(2008)
Peptide-mediated nanoparticle delivery by G-protein coupled receptors (GPCRs).
In: Summer school "Medicinal Chemistry: Molecular Recognition – Ligand Receptor Interactions”, 29. September - 1. Oktober 2008, Regensburg.
Fulltext not available.
Hild, W. A., Breunig, Miriam and Göpferich, Achim
(2008)
Quantum dots - Nano-sized probes for the exploration of cellular and intracellular targeting.
European Journal of Pharmaceutics and Biopharmaceutics 68 (2), pp. 153-168.
Fulltext not available.
Hild, W., Zenger, Katharina, Caporale, A., Cabrele, C., Breunig, Miriam, Teßmar, Jörg and Göpferich, Achim
(2008)
Towards peptide-modified nanocrystals for drug targeting applications.
In: Controlled Release Society, Local Chapter, Braunschweig.
Fulltext not available.
Hild, W., Breunig, Miriam, Teßmar, Jörg and Göpferich, Achim
(2007)
Custom designed Quantum Dots for cellular uptake.
In: Partec 2007, Nuernberg.
Fulltext not available.
Hofinger, Edith S. A., Bernhardt, Günther and Buschauer, Armin
(2007)
Kinetics of Hyal1 and PH-20 hyaluronidases: comparison of minimal substrates and analysis of the transglycosylation reaction.
Glycobiology 17 (9), pp. 963-971.
Fulltext not available.
Hofinger, Edith S. A., Spickenreither, Martin, Oschmann, Jan, Bernhardt, Günther, Rudolph, Rainer and Buschauer, Armin
(2007)
Recombinant human hyaluronidase Hyal-1: insect cells versus E. coli as expression system and identification of low molecular weight inhibitors.
Glycobiology 17 (4), pp. 444-453.
Fulltext not available.
Hild, W., Lang, R., Winter, G. and Göpferich, Achim
(2007)
Towards the characterization of quantum dots by asymmetrical flow field-flow fractionation.
In: Jahrestagung der DPhG, Erlangen.
Fulltext not available.
Hild, W., Teßmar, Jörg and Göpferich, Achim
(2006)
Quantum dot colloids for cell-uptake studies.
In: 3rd Summer School "Medicinal Chemistry", Regensburg.
Fulltext not available.
I
Igel, Patrick, Dove, Stefan and Buschauer, Armin
(2010)
Histamine H4 receptor agonists.
Bioorganic & Medicinal Chemistry Letters 20 (24), pp. 7191-7199.
Fulltext not available.
Igel, Patrick, Geyer, Roland, Straßer, Andrea, Dove, Stefan, Seifert, Roland and Buschauer, Armin
(2009)
Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H(4) receptor agonists.
Journal of Medicinal Chemistry 52 (20), pp. 6297-6313.
Fulltext not available.
Igel, Patrick, Schneider, Erich , Schnell, David, Elz, Sigurd, Seifert, Roland and Buschauer, Armin
(2009)
N(G)-Acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.
Journal of Medicinal Chemistry 52 (8), pp. 2623-2627.
Fulltext not available.
, Schnell, David, Elz, Sigurd, Seifert, Roland and Buschauer, Armin
(2009)
N(G)-Acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.
Journal of Medicinal Chemistry 52 (8), pp. 2623-2627.
Fulltext not available.
Igel, Patrick, Schnell, David, Bernhardt, Günther, Seifert, Roland and Buschauer, Armin
(2009)
Tritium-labeled N1-[3-(1H-imidazol-4-yl)propyl]-N2-propionylguanidine ([3H]UR-PI294), a high affinity histamine H3 and H4 receptor radioligand.
ChemMedChem 4 (2), pp. 225-231.
Fulltext not available.
K
Keller, Max, Kaske, Melanie, Holzammer, Tobias, Bernhardt, Günther and Buschauer, Armin
(2013)
Dimeric argininamide-type neuropeptide Y receptor antagonists: chiral discrimination between Y1 and Y4 receptors.
Bioorganic and Medicinal Chemistry 21 (21), pp. 6303-6322.
Fulltext not available.
Keller, Max, Bernhardt, Günther and Buschauer, Armin
(2011)
[3H]UR-MK136 - a highly potent and selective radioligand for neuropeptide Y Y1 receptors.
ChemMedChem 6 (9), pp. 1566-1571.
Fulltext not available.
Keller, Max, Erdmann, Daniela, Teng, Shangjun, Pop, Nathalie , Pluym, Nikola, Bernhardt, Günther and Buschauer, Armin
(2011)
Red-fluorescent argininamide-type NPY Y(1) receptor antagonists as pharmacological tools.
Bioorganic & Medicinal Chemistry 19 (9), pp. 2859-2878.
Fulltext not available.
, Pluym, Nikola, Bernhardt, Günther and Buschauer, Armin
(2011)
Red-fluorescent argininamide-type NPY Y(1) receptor antagonists as pharmacological tools.
Bioorganic & Medicinal Chemistry 19 (9), pp. 2859-2878.
Fulltext not available.
Kleinmaier, R. and Gschwind, R. M.
(2010)
Chemical Shift Assignment and Conformational Analysis of Monoalkylated Acylguanidines.
Magn. Reson. Chem. 48 (9), pp. 687-684.
Fulltext not available.
(2010)
Chemical Shift Assignment and Conformational Analysis of Monoalkylated Acylguanidines.
Magn. Reson. Chem. 48 (9), pp. 687-684.
Fulltext not available.
Kleinmaier, Roland, Igel, Patrick, Keller, Max, Buschauer, Armin and Gschwind, Ruth M.
(2010)
Conformations, Conformational Preferences, and Conformational Exchange of N'-Substituted N-Acylguanidines: Intermolecular Interactions Hold the Key.
J. Am. Chem. Soc. 132 (32), pp. 11223-11233.
Fulltext not available.
(2010)
Conformations, Conformational Preferences, and Conformational Exchange of N'-Substituted N-Acylguanidines: Intermolecular Interactions Hold the Key.
J. Am. Chem. Soc. 132 (32), pp. 11223-11233.
Fulltext not available.
König, Burkhard, Späth, A. and Koch, C.
(2010)
Luminescent Hybrids Combining a Metal Complex and a Crown Ether – Receptors for Peptidic Ammonium Phosphates.
European Journal of Inorganic Chemistry (19), pp. 2926-2935.
Fulltext not available.
(2010)
Luminescent Hybrids Combining a Metal Complex and a Crown Ether – Receptors for Peptidic Ammonium Phosphates.
European Journal of Inorganic Chemistry (19), pp. 2926-2935.
Fulltext not available.
Keller, Max, Teng, Shangjun, Bernhardt, Günther and Buschauer, Armin
(2009)
Bivalent argininamide-type neuropeptide Y Y1 antagonists do not support the hypothesis of receptor dimerisation.
ChemMedChem 4 (10), pp. 1733-1745.
Fulltext not available.
Kraus, Anja, Ghorai, Prasanta, Birnkammer, Tobias, Schnell, David, Elz, Sigurd, Seifert, Roland, Dove, Stefan, Bernhardt, Günther and Buschauer, Armin
(2009)
N(G)-Acylated aminothiazolylpropylguanidines as potent and selective histamine H2 receptor agonists.
ChemMedChem 4 (2), pp. 232-240.
Fulltext not available.
Kühnle, Matthias, Egger, Michael, Müller, Christine, Mahringer, Anne, Bernhardt, Günther, Fricker, Gert , König, Burkhard and Buschauer, Armin
(2009)
Potent and selective inhibitors of breast cancer resistance protein (ABCG2) derived from the p-glycoprotein (ABCB1) modulator tariquidar.
Journal of Medicinal Chemistry 52 (4), pp. 1190-1197.
Fulltext not available.
, König, Burkhard and Buschauer, Armin
(2009)
Potent and selective inhibitors of breast cancer resistance protein (ABCG2) derived from the p-glycoprotein (ABCB1) modulator tariquidar.
Journal of Medicinal Chemistry 52 (4), pp. 1190-1197.
Fulltext not available.
Kleinmaier, R. and Gschwind, R. M.
(2009)
Selective [15N.eta.2] labelling of an NG-propionylated arginine derivative.
Journal of Labelled Compounds and Radiopharmaceuticals 52 (2), pp. 29-32.
Fulltext not available.
(2009)
Selective [15N.eta.2] labelling of an NG-propionylated arginine derivative.
Journal of Labelled Compounds and Radiopharmaceuticals 52 (2), pp. 29-32.
Fulltext not available.
Keller, Max, Pop, Nathalie, Hutzler, Christoph , Beck-Sickinger, Annette G., Bernhardt, Günther and Buschauer, Armin
(2008)
Guanidine - acylguanidine bioisosteric approach in the design of radioligands: Synthesis of a tritium-labeled N(G)-propionylargininamide ([3H]UR-MK114) as a highly potent and selective neuropeptide Y Y1 receptor antagonist.
Journal of Medicinal Chemistry 51 (24), pp. 8168-8172.
Fulltext not available.
, Beck-Sickinger, Annette G., Bernhardt, Günther and Buschauer, Armin
(2008)
Guanidine - acylguanidine bioisosteric approach in the design of radioligands: Synthesis of a tritium-labeled N(G)-propionylargininamide ([3H]UR-MK114) as a highly potent and selective neuropeptide Y Y1 receptor antagonist.
Journal of Medicinal Chemistry 51 (24), pp. 8168-8172.
Fulltext not available.
Kiewitz, S. D., Kruppa, M., Riechers, A., König, B. and Cabrele, C.
(2008)
Recognition of the Helix-Loop-Helix Domain of the Id Proteins by an Artificial Luminescent Metal Complex Receptor.
J. Mol. Recognit 21, 79 - 88.
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and Cabrele, C.
(2008)
Recognition of the Helix-Loop-Helix Domain of the Id Proteins by an Artificial Luminescent Metal Complex Receptor.
J. Mol. Recognit 21, 79 - 88.
Fulltext not available.
Kruppa, Michael, Frank, Daniel, Leffler-Schuster, Helga and König, Burkhard
(2006)
Screening of Metal Complex – Amino Acid Side Chain Interactions by Potentiometric Titration.
Inorganica Chimica Acta 359 (4), pp. 1159-1168.
Fulltext restricted.
Knerr, Robert, Weiser, Barbara, Drotleff, S., Steinem, C. and Göpferich, Achim
(2006)
Measuring cell adhesion on RGD-modified, self-assembled PEG monolayers using the quartz crystal microbalance technique.
Macromolecular Bioscience 6 (10), pp. 827-838.
Fulltext not available.
Knerr, Robert, Drotleff, S., Steinem, C. and Göpferich, Achim
(2006)
Self-assembling PEG Derivatives for Protein-repellant Biomimetic Model Surfaces on Gold.
Biomaterialien 7 (1), pp. 12-20.
Fulltext not available.
Knerr, Robert, Weiser, Barbara, Drotleff, Sigrid and Steinem, Claudia
(2005)
"Protein adsorption and cell adhesion on RGD modified PEG monolayers".
In: "European Symposium on polymeric Biomaterials", 2005, Madrid, Spanien.
Fulltext not available.
Kruppa, M., Mandl, C., Miltschitzky, S. and König, B.
(2005)
A Luminescent Receptor with Affinity for N-terminal Histidine in Peptides in Aqueous Solution.
J. Am. Chem. Soc. 127, 3362 - 3365.
Fulltext not available.
Kalbitzer, H. R., Spoerner, M., Graf, T. and König, B.
(2005)
A Novel Mechanism for the Modulation of the Ras-Effector Interaction by small molecules.
Biochem. Biophys. Res. Commun. 334, 709 – 713.
Fulltext not available.
Kruppa, M., Bonauer, C., Michlová, V. and König, B.
(2005)
Enhanced Peptide β-Sheet Affinity by Metal to Ligand Coordination.
J. Org. Chem. 70, 5305 - 5308.
Fulltext not available.
Knerr, Robert, Weiser, Barbara, Drotleff, S., Steinem, C. and Göpferich, Achim
(2005)
Protein adsorption and cell adhesion on RGD modified PEG monolayers.
In: Life Science Interface Summer School, University of Nottingham, Nottingham, UK.
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König, B. and Miltschitzky, S.
(2005)
Small Peptides with a β-Hairpin Structure.
Org. Prep. Proced. Int. 37, pp. 307-336.
Fulltext not available.
(2005)
Small Peptides with a β-Hairpin Structure.
Org. Prep. Proced. Int. 37, pp. 307-336.
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Knerr, Robert, Steinem, C., Roberts, C. J. and Göpferich, Achim
(2004)
A model to investigate cell surface interactions: PEGylated alkanethiolates on gold - protein resistance and visualization.
In: Transactions, 31st annual meeting and exposition of the Controlled Release Society, Honolulu, HI.
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Klein, M., Walenzyk, T. and König, B.
(2004)
Electronic Effects on the Bergman Cyclisation of Enediynes. A Review.
Collect. Czech. Chem. Commun. 69, 945 – 965.
Fulltext not available.
Knerr, Robert, Steinem, C., Roberts, C. J. and Göpferich, Achim
(2004)
Self - assembled monolayers of PEGylated alkanethiolates on gold - A model to investigate cell - surface interactions.
In: DPHG, ÖPHG, CPS Joint Meeting 2004, Regensburg, Germany.
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Knerr, Robert, Steinem, C., Roberts, C. J. and Göpferich, Achim
(2004)
Self - assembled monolayers of PEGylated alkanethiolates on gold - A model to investigate cell - surface interactions.
In: 2nd Summer School Medicinal Chemistry, University of Regensburg, Regensburg, Germany.
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Klein, M. and König, B.
(2004)
Synthesis and Thermal Cyclization of an Enediyne-Sulfonamide.
Tetrahedron 60, 1087 - 1092.
Fulltext not available.
Klein, Michael, Zabel, Manfred, Bernhardt, Günther and König, Burkhard
(2003)
Tetrahydroxy 10-membered cyclic enediynes.
The Journal of organic chemistry 68 (24), pp. 9379-9383.
Fulltext not available.
Knerr, Robert, Steinem, Claudia and Göpferich, Achim
(2002)
Intergin-mediated interactions between cells amd biomimetic materials.
In: "Summer School Medicinal Chemistry", 15. - 18. September 2002, Regensburg.
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König, B., Pitsch, W., Klein, M., Vasold, R., Prall, M. and Schreiner, P. R.
(2001)
Carbonyl- and Carboxyl-substituted Enediynes: Synthesis, Computations, and Thermal Reactivity.
J. Org. Chem. 66, pp. 1742-1746.
Fulltext not available.
(2001)
Carbonyl- and Carboxyl-substituted Enediynes: Synthesis, Computations, and Thermal Reactivity.
J. Org. Chem. 66, pp. 1742-1746.
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König, B.
(2000)
Changing the Reactivity of Enediynes by Metal Ion Coordination (review).
Eur. J. Org. Chem., pp. 381-385.
L
Li, X., Miltschitzky, Stefan and König, B.
(2006)
Luminescent Pyrimidine Hydrazide Oligomers with Peptide Affinity.
Bioorganic & Medicinal Chemistry 14, 6075 -6084.
Fulltext not available.
(2006)
Luminescent Pyrimidine Hydrazide Oligomers with Peptide Affinity.
Bioorganic & Medicinal Chemistry 14, 6075 -6084.
Fulltext not available.
Li, X., Miltschitzky, S., Grauer, A., Michlová, V. and König, B.
(2006)
Synthesis and Peptide-binding Properties of a Luminescent Pyrimidine Zinc(II) Complex.
Tetrahedron 62, 12191 - 12196.
Fulltext not available.
(2006)
Synthesis and Peptide-binding Properties of a Luminescent Pyrimidine Zinc(II) Complex.
Tetrahedron 62, 12191 - 12196.
Fulltext not available.
Li, Liantao, Mayer, Matthias, Schneider, Erich , Schreiber, Elvira, Bernhardt, Günther, Peng, Shiqi and Buschauer, Armin
(2003)
Preparation of fluorescent nonpeptidic neuropeptide Y receptor ligands: analogues of the quinazoline-type anti-obesity Y5 antagonist CGP 71683A.
Arch Pharm (Weinheim) 336 (12), pp. 585-590.
Fulltext not available.
, Schreiber, Elvira, Bernhardt, Günther, Peng, Shiqi and Buschauer, Armin
(2003)
Preparation of fluorescent nonpeptidic neuropeptide Y receptor ligands: analogues of the quinazoline-type anti-obesity Y5 antagonist CGP 71683A.
Arch Pharm (Weinheim) 336 (12), pp. 585-590.
Fulltext not available.
M
Memminger, Martin, Keller, Max, Lopuch, Miroslaw, Pop, Nathalie, Bernhardt, Günther, von Angerer, Erwin and Buschauer, Armin
(2012)
The Neuropeptide Y Y1 receptor: a diagnostic marker? Expression in MCF-7 breast cancer cells is down-regulated by antiestrogens in vitro and in xenografts.
PLoS ONE 7 (12), e51032.
Maity, P. and König, B.
(2008)
Synthesis and Structure of 1,4-Dipiperazino Benzenes - Chiral Terphenyl-type Peptide.
Org. Lett. 10, 1473 - 1476.
Fulltext not available.
Maity, P. and König, Burkhard
(2007)
Enantio- and Diastereoselective Syntheses of Cyclic Cα-Tetrasubstituted α-Amino Acids and Their Use to Induce Stable Conformations in Short Peptides (Review).
Pept. Sci. 90, 8 - 27.
Fulltext not available.
(2007)
Enantio- and Diastereoselective Syntheses of Cyclic Cα-Tetrasubstituted α-Amino Acids and Their Use to Induce Stable Conformations in Short Peptides (Review).
Pept. Sci. 90, 8 - 27.
Fulltext not available.
Maity, P., Zabel, M. and König, B.
(2007)
Tetrahydrofuran Cα-Tetrasubstituted Amino Acids: Two Consecutive β Turns in a Crystalline Linear Tripeptide.
J. Org. Chem. 72, 8046 – 8053.
Fulltext not available.
(2007)
Tetrahydrofuran Cα-Tetrasubstituted Amino Acids: Two Consecutive β Turns in a Crystalline Linear Tripeptide.
J. Org. Chem. 72, 8046 – 8053.
Fulltext not available.
Miltschitzky, Stefan, Michlova, Veronika, Stadlbauer, Stefan and König, Burkhard
(2006)
Synthesis of substituted pyrimidine hydrazine acids (PHA) and their use in peptide recognition.
Heterocycles 67 (1), pp. 135-160.
Fulltext not available.
Maity, P. and König, B.
(2006)
Synthesis of 3-Oxo-2,3-dihydro-pyrrole Amino Acids as Chiral Dipeptidomimics.
Synthesis (16), pp. 2719-2724.
Fulltext not available.
(2006)
Synthesis of 3-Oxo-2,3-dihydro-pyrrole Amino Acids as Chiral Dipeptidomimics.
Synthesis (16), pp. 2719-2724.
Fulltext not available.
Mandl, C. P. and König, B.
(2005)
Luminescent Crown Ether Amino Acids - Selective Binding to N-terminal Lysine in Peptides.
J. Org. Chem. 70, 670 – 674.
Fulltext not available.
N
Nordemann, Uwe, Wifling, David , Schnell, David, Bernhardt, Günther, Stark, Holger , Seifert, Roland and Buschauer, Armin
(2013)
Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts.
PLoS One 8 (9), e73961.
Nickl, Kathrin, Gardner, Eric E., Geiger, Sarah, Heilmann, Jörg and Seifert, Roland
(2008)
Differential coupling of the human cannabinoid receptors hCB1R and hCB2R to the G-protein Galpha i2beta 1gamma 2.
Neuroscience letters 447 (1), pp. 68-72.
Fulltext not available.
O
Ochoa Puentes, Cristian, Höcherl, Peter, Kühnle, Matthias, Bauer, Stefanie, Kürger, Kira, Bernhardt, Günther, Buschauer, Armin and König, Burkhard
(2011)
Solid phase synthesis of tariquidar-related modulators of ABC transporters preferring breast cancer resistance protein (ABCG2).
Bioorganic & Medicinal Chemistry Letters 21 (12), pp. 3654-3657.
Fulltext not available.
(2011)
Solid phase synthesis of tariquidar-related modulators of ABC transporters preferring breast cancer resistance protein (ABCG2).
Bioorganic & Medicinal Chemistry Letters 21 (12), pp. 3654-3657.
Fulltext not available.
P
Pluym, Nikola , Baumeister, Paul, Keller, Max, Bernhardt, Günther and Buschauer, Armin
(2013)
[3H]UR-PLN196: A Selective Nonpeptide Radioligand and Insurmountable Antagonist for the Neuropeptide Y Y2 Receptor.
ChemMedChem 8 (4), pp. 587-593.
Fulltext not available.
, Baumeister, Paul, Keller, Max, Bernhardt, Günther and Buschauer, Armin
(2013)
[3H]UR-PLN196: A Selective Nonpeptide Radioligand and Insurmountable Antagonist for the Neuropeptide Y Y2 Receptor.
ChemMedChem 8 (4), pp. 587-593.
Fulltext not available.
Pluym, Nikola, Brennauer, Albert, Keller, Max, Ziemek, Ralf, Pop, Nathalie, Bernhardt, Günther and Buschauer, Armin
(2011)
Application of the guanidine – acylguanidine bioisosteric approach to argininamide-type NPY Y2 receptor antagonists.
ChemMedChem 6 (9), pp. 1727-1738.
Fulltext not available.
Pop, Nathalie, Igel, Patrick, Brennauer, Albert, Cabrele, Chiara , Bernhardt, Günther, Seifert, Roland and Buschauer, Armin
(2011)
Functional reconstitution of human neuropeptide Y (NPY) Y2 and Y4 receptors in Sf9 insect cells.
Journal of Receptors and Signal Transduction 31 (4), pp. 271-285.
Fulltext not available.
, Bernhardt, Günther, Seifert, Roland and Buschauer, Armin
(2011)
Functional reconstitution of human neuropeptide Y (NPY) Y2 and Y4 receptors in Sf9 insect cells.
Journal of Receptors and Signal Transduction 31 (4), pp. 271-285.
Fulltext not available.
Pollinger, Klaus, Breunig, Miriam, Tessmar, Joerg and Göpferich, Achim
(2010)
"Receptor mediated targeting of micelles - the folate receptor as proof of principle".
In: "5th Summer School Medicinal Chemistry", 13. - 15. September 2010, Regensburg.
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Preuss, Hendrik, Ghorai, Prasanta, Kraus, Anja, Dove, Stefan, Buschauer, Armin and Seifert, Roland
(2007)
Constitutive Activity and Ligand Selectivity of Human,Guinea Pig, Rat, and Canine Histamine H₂ Receptors. Journal of Pharmacology and Experimental Therapeutics 321 (3), pp. 983-995.
Preuss, Hendrik, Ghorai, Prasanta, Kraus, Anja, Dove, Stefan, Buschauer, Armin and Seifert, Roland
(2007)
Mutations of Cys-17 and Ala-271 in the Human Histamine H₂Receptor Determine the Species Selectivity of Guanidine-Type Agonists and Increase Constitutive Activity. Journal of Pharmacology and Experimental Therapeutics 321 (3), pp. 975-982.
Preuss, Hendrik, Ghorai, Prasanta, Kraus, Anja, Dove, Stefan, Buschauer, Armin and Seifert, Roland
(2007)
Point Mutations in the Second Extracellular Loop of the Histamine H2 Receptor do not affect the Species-Selective Activity of Guanidine-Type Agonists.
Naunyn Schmiedebergs Arch. Pharmacol. 376 (4), pp. 253-264.
Fulltext restricted.
Pitsch, W., Klein, M., Zabel, M. and König, B.
(2002)
Synthesis and Structure of a Stabilized 10-Membered Cyclic Enediyne.
J. Org. Chem. 67, 6805 - 6807.
Fulltext not available.
R
Reher, Till M., Neumann, Detlef, Buschauer, Armin and Seifert, Roland
(2012)
Incomplete activation of human eosinophils via the histamine H(4)-receptor: Evidence for ligand-specific receptor conformations.
Biochemical Pharmacology 84 (2), pp. 192-203.
Fulltext not available.
Rosnizeck, I. C., Graf, T., Spoerner, M., Tränkle, J., Filchtinski, D., Herrmann, C., Gremer, L. , Vetter, I., Wittinghofer, A., König, Burkhard and Kalbitzer, H. R.
(2010)
Stabilizing a Weak Binding State for Effectors in the Human Ras Protein by Cyclen Complexes.
Angewandte Chemie International Edition (49), pp. 3830-3833.
Fulltext not available.
, Vetter, I., Wittinghofer, A., König, Burkhard and Kalbitzer, H. R.
(2010)
Stabilizing a Weak Binding State for Effectors in the Human Ras Protein by Cyclen Complexes.
Angewandte Chemie International Edition (49), pp. 3830-3833.
Fulltext not available.
Riechers, Alexander, Schmidt, Florian, Stadlbauer, Stefan and König, Burkhard
(2009)
Detection of protein phosphorylation on SDS-PAGE using probes with a phosphate-sensitive emmision response.
Bioconjugate Chemistry 20, pp. 804-807.
Fulltext not available.
(2009)
Detection of protein phosphorylation on SDS-PAGE using probes with a phosphate-sensitive emmision response.
Bioconjugate Chemistry 20, pp. 804-807.
Fulltext not available.
Rigden, Daniel J. , Botzki, Alexander , Nukui, Masatoshi, Mewbourne, R. Brandon, Lamani, Ejvis, Braun, Stephan, von Angerer, Erwin, Bernhardt, Günther, Dove, Stefan, Buschauer, Armin and Jedrzejas, Mark J.
(2006)
Design of new benzoxazole-2-thione derived inhibitors of Streptococcus pneumoniae hyaluronan lyase: structure of a complex with a 2-phenylindole.
Glycobiology 16 (8), pp. 757-765.
Fulltext not available.
, Botzki, Alexander , Nukui, Masatoshi, Mewbourne, R. Brandon, Lamani, Ejvis, Braun, Stephan, von Angerer, Erwin, Bernhardt, Günther, Dove, Stefan, Buschauer, Armin and Jedrzejas, Mark J.
(2006)
Design of new benzoxazole-2-thione derived inhibitors of Streptococcus pneumoniae hyaluronan lyase: structure of a complex with a 2-phenylindole.
Glycobiology 16 (8), pp. 757-765.
Fulltext not available.
Ritter, S., Eiblmeier, M., Michlova, V. and König, B.
(2005)
Chiral NADH Model Systems functionalized with Zn(II)-cyclen as Flavin Binding Site.
Tetrahedron 61, 5241 - 5251.
Fulltext not available.
Rzepecki, P., Gallmeier, H., Geib, N., König, B. and Schrader, T.
(2004)
New heterocyclic β-sheet ligands with peptidic recognition elements.
J. Org. Chem. 69, 5168 – 5178.
Fulltext not available.
S
Schreeb, Annemarie, Łażewska, Dorota, Dove, Stefan, Buschauer, Armin, Kieć-Kononiwcz, Katarzyna and Stark, Holger
(2013)
2. Histamine H4 receptor ligands.
In: Stark, Holger, (ed.)
Histamine H4 receptor: a novel drug target for immunoregulation and inflammation.
Versita, London, pp. 21-62.
ISBN 9788376560564.
Fulltext not available.
Seifert, Roland, Strasser, Andrea, Schneider, Erich H., Neumann, Detlef, Dove, Stefan and Buschauer, Armin
(2013)
Molecular and cellular analysis of human histamine receptor subtypes.
Trends in Pharmacological Sciences 34 (1), pp. 33-58.
Fulltext not available.
Strasser, Andrea, Wittmann, Hans-Joachim, Buschauer, Armin, Schneider, Erich H. and Seifert, Roland
(2013)
Species-dependent activities of GPCR ligands: Lessons from histamine receptor orthologs.
Trends in Pharmacological Sciences 34 (1), pp. 13-32.
Fulltext not available.
Schnell, David, Brunskole, Irena, Ladova, Katerina, Schneider, Erich H. , Igel, Patrick, Dove, Stefan, Buschauer, Armin and Seifert, Roland
(2011)
Expression and functional properties of canine, rat and murine histamine H4-receptors in Sf9 insect cells.
Naunyn-Schmiedeberg's Archives of Pharmacology 383 (5), pp. 457-470.
Fulltext not available.
, Igel, Patrick, Dove, Stefan, Buschauer, Armin and Seifert, Roland
(2011)
Expression and functional properties of canine, rat and murine histamine H4-receptors in Sf9 insect cells.
Naunyn-Schmiedeberg's Archives of Pharmacology 383 (5), pp. 457-470.
Fulltext not available.
Seifert, Roland, Schneider, Erich H. , Dove, Stefan, Brunskole, Irena, Neumann, Detlef , Strasser, Andrea and Buschauer, Armin
(2011)
Paradoxical stimulatory effects of the “standard” histamine H4-receptor antagonist JNJ7777120: The H4-receptor joins the club of 7TM receptors exhibiting functional selectivity.
Molecular Pharmacology 79 (4), pp. 631-638.
Fulltext not available.
, Dove, Stefan, Brunskole, Irena, Neumann, Detlef , Strasser, Andrea and Buschauer, Armin
(2011)
Paradoxical stimulatory effects of the “standard” histamine H4-receptor antagonist JNJ7777120: The H4-receptor joins the club of 7TM receptors exhibiting functional selectivity.
Molecular Pharmacology 79 (4), pp. 631-638.
Fulltext not available.
Schinner, Elisabeth, Salb, Katharina and Schlossmann, Jens
(2011)
Signaling via IRAG is essential for NO/cGMP-dependent inhibition of platelet activitation.
Platelets.
Fulltext not available.
Silva, Maria Elena, Heim, Ralf, Strasser, Andrea, Elz, Sigurd and Dove, Stefan
(2011)
Theoretical studies on the interaction of partial agonists with the 5-HT(2A) receptor.
Journal of computer-aided molecular design 25 (1), pp. 51-66.
Fulltext not available.
Späth, A. and König, Burkhard
(2010)
Ditopic crown ether – guanidinium ion receptors for the molecular recognition of amino acids and small peptides.
Tetrahedron (66), pp. 1859-1873.
Fulltext not available.
(2010)
Ditopic crown ether – guanidinium ion receptors for the molecular recognition of amino acids and small peptides.
Tetrahedron (66), pp. 1859-1873.
Fulltext not available.
Schneider, Erich H., Schnell, David, Strasser, Andrea, Dove, Stefan and Seifert, Roland
(2010)
Impact of the DRY Motif and the Missing "Ionic Lock" on Constitutive Activity and G-Protein Coupling of the Human Histamine H-4 Receptor.
Journal of Pharmacology and Experimental Therapeutics 333 (2), pp. 382-392.
Fulltext not available.
Seifert, Roland and Dove, Stefan
(2009)
Functional Selectivity of GPCR Ligand Stereoisomers: New Pharmacological Opportunities.
Mol. Pharmacol. 75 (1), pp. 13-18.
Fulltext not available.
Späth, A. and König, Burkhard
(2009)
Modular Synthesis of Di- and Tripeptides of Luminescent Crown Ether Aminocarboxylic Acids.
Tetrahedron 65, 690 - 695.
Fulltext not available.
(2009)
Modular Synthesis of Di- and Tripeptides of Luminescent Crown Ether Aminocarboxylic Acids.
Tetrahedron 65, 690 - 695.
Fulltext not available.
Schmid, M., Fleischmann, M., D'Elia, V., Reiser, O. , Gronwald, W. and Gschwind, R. M.
(2009)
RDCs in Short Peptidic Foldamers: Combined Analyses of Backbone and Side Chain Conformations and Evaluation of Structure Coordinates of Rigid Unnatural Amino Acids.
ChemBioChem 10 (3), pp. 440-444.
Fulltext not available.
, Gronwald, W. and Gschwind, R. M.
(2009)
RDCs in Short Peptidic Foldamers: Combined Analyses of Backbone and Side Chain Conformations and Evaluation of Structure Coordinates of Rigid Unnatural Amino Acids.
ChemBioChem 10 (3), pp. 440-444.
Fulltext not available.
Subat, M., Woinaroschy, K., Gerstl, C., Sarkar, B., Kaim, W. and König, B.
(2008)
1,4,7,10 - Tetraazacyclododecane Metal Complexes as Potent Promoters of Phosphodiester Hydrolysis under Physiologica.
Inorg. Chem. 47, 4661 - 4668.
Fulltext not available.
Stadlbauer, S., Riechers, A., Späth, A. and König, B.
(2008)
Utilizing Reversible Copper(II) Peptide Coordination in a Sequence Selective Luminescent Receptor.
Chem. Eur. J. 14, 2536 - 2541.
Fulltext not available.
(2008)
Utilizing Reversible Copper(II) Peptide Coordination in a Sequence Selective Luminescent Receptor.
Chem. Eur. J. 14, 2536 - 2541.
Fulltext not available.
Schneider, Erich , Keller, Max, Brennauer, Albert, Hoefelschweiger, Bianca K., Gross, Dietmar, Wolfbeis, Otto S. , Bernhardt, Günther and Buschauer, Armin
(2007)
Synthesis and Characterization of the First Fluorescent Nonpeptide NPY Y1 Receptor Antagonist.
ChemBioChem 8 (16), pp. 1981-1988.
Fulltext restricted.
, Keller, Max, Brennauer, Albert, Hoefelschweiger, Bianca K., Gross, Dietmar, Wolfbeis, Otto S. , Bernhardt, Günther and Buschauer, Armin
(2007)
Synthesis and Characterization of the First Fluorescent Nonpeptide NPY Y1 Receptor Antagonist.
ChemBioChem 8 (16), pp. 1981-1988.
Fulltext restricted.
Schneider, Erich , Mayer, Matthias, Ziemek, Ralf, Li, Liantao, Hutzler, Christoph , Bernhardt, Günther and Buschauer, Armin
(2006)
A Simple and Powerful Flow Cytometric Method for the Simultaneous Determination of Multiple Parameters at G-Protein-coupled Receptor Subtypes.
ChemBioChem 7 (9), pp. 1400-1409.
Fulltext not available.
, Mayer, Matthias, Ziemek, Ralf, Li, Liantao, Hutzler, Christoph , Bernhardt, Günther and Buschauer, Armin
(2006)
A Simple and Powerful Flow Cytometric Method for the Simultaneous Determination of Multiple Parameters at G-Protein-coupled Receptor Subtypes.
ChemBioChem 7 (9), pp. 1400-1409.
Fulltext not available.
Spickenreither, Martin, Braun, Stephan, Bernhardt, Günther, Dove, Stefan and Buschauer, Armin
(2006)
Novel 6-O-acylated vitamin C derivatives as hyaluronidase inhibitors with selectivity for bacterial lyases.
Bioorganic & Medicinal Chemistry Letters 16 (20), pp. 5313-5316.
Fulltext not available.
Suhs, T. and König, B.
(2006)
Synthesis of Functionalized Guanidino Amino Acids.
Chem. Eur. J. 12, 8150 – 8157.
Fulltext not available.
(2006)
Synthesis of Functionalized Guanidino Amino Acids.
Chem. Eur. J. 12, 8150 – 8157.
Fulltext not available.
Suhs, Thomas and König, Burkhard
(2006)
Synthesis of Guanidines in Solution.
Mini-Reviews in Organic Chemistry 3, pp. 315-331.
Fulltext not available.
Salmen, Sunnhild, Hoechstetter, Julia, Käsbauer, Christian, Paper, Dieter H., Bernhardt, Günther and Buschauer, Armin
(2005)
Sulphated Oligosaccharides as Inhibitors of Hyaluronidases from Bovine Testis, Bee Venom and Streptococcus agalactiae.
Planta Med. 71, pp. 727-732.
Fulltext not available.
Subat, M., Borovik, A. S. and König, B.
(2004)
A Synthetic Creatinine Receptor: Imprinting of a Lewis-Acidic Zinc(II)cyclen Binding Site to Shape its Molecular Recognition Selectivity.
J. Am. Chem. Soc. 126, 3185 - 3190.
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Taha, H. M., Schmidt, J., Göttle, M., Suryanarayana, S., Shen, Y., Tang, W.-J. , Gille, A. , Geduhn, Jens, König, Burkhard , Dove, Stefan and Seifert, Roland
(2009)
Molecular Analysis of the Interaction of Anthrax Adenylyl Cyclase Toxin, Edema Factor, with 2'(3')-O-(N-(methyl)anthraniloyl)-Substituted Purine and Pyrimidine Nucleotides.
Mol. Pharmacol. 75 (3), pp. 693-703.
Fulltext not available.
, Gille, A. , Geduhn, Jens, König, Burkhard , Dove, Stefan and Seifert, Roland
(2009)
Molecular Analysis of the Interaction of Anthrax Adenylyl Cyclase Toxin, Edema Factor, with 2'(3')-O-(N-(methyl)anthraniloyl)-Substituted Purine and Pyrimidine Nucleotides.
Mol. Pharmacol. 75 (3), pp. 693-703.
Fulltext not available.
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Vomasta, Daniel, Innocenti, A., König, Burkhard and Supuran, T.
(2009)
Carbonic anhydrase inhibitors: Two-prong versus mono-prong inhibitors of isoformsI, II, IX and XII exemplified by photochromics cis-1,2-a-dithienylethene derivates.
Bioorganic & Medicinal Chemistry Letters 19, pp. 1283-1286.
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and Supuran, T.
(2009)
Carbonic anhydrase inhibitors: Two-prong versus mono-prong inhibitors of isoformsI, II, IX and XII exemplified by photochromics cis-1,2-a-dithienylethene derivates.
Bioorganic & Medicinal Chemistry Letters 19, pp. 1283-1286.
Fulltext not available.
Vasold, R., Engel, E., König, B. , Landthaler, M. and Baeumler, W.
(2008)
Health risks of tattoo colors.
Anal. Bioanal. Chem. 391, 9 - 13.
Fulltext not available.
, Landthaler, M. and Baeumler, W.
(2008)
Health risks of tattoo colors.
Anal. Bioanal. Chem. 391, 9 - 13.
Fulltext not available.
Vomasta, D., Högner, C., Branda, N. R. and König, B.
(2008)
Regulation of Human Carbonic Anhydrase I (hCAI) Activity by Using a Photochromic Inhibitor.
Angew. Chem. 120, pp. 7756-7759.
Fulltext not available.
(2008)
Regulation of Human Carbonic Anhydrase I (hCAI) Activity by Using a Photochromic Inhibitor.
Angew. Chem. 120, pp. 7756-7759.
Fulltext not available.
Vasold, R., Naarmann, N., Ulrich, H., Fischer, D., König, B., Landthaler, M. and Bäumler, W.
(2004)
Tattoo Pigments are Cleaved by Laser Light – The Chemical Analysis In Vitro Provide Evidence for Hazardous Compounds.
Photochem. Photobiol. 80, 185 – 190.
Fulltext not available.
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Wifling, David , Bernhardt, Günther, Dove, Stefan and Buschauer, Armin
(2015)
The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity.
PLoS One 10 (1), pp. 1-14.
Wifling, David , Löffel, Karolin, Nordemann, Uwe, Strasser, Andrea, Bernhardt, Günther, Dove, Stefan, Seifert, Roland and Buschauer, Armin
(2015)
Molecular determinants for the high constitutive activity of the human histamine H4 receptor: Functional studies on orthologs and mutants.
British Journal of Pharmacology 172, pp. 785-798.
Fulltext not available.
, Löffel, Karolin, Nordemann, Uwe, Strasser, Andrea, Bernhardt, Günther, Dove, Stefan, Seifert, Roland and Buschauer, Armin
(2015)
Molecular determinants for the high constitutive activity of the human histamine H4 receptor: Functional studies on orthologs and mutants.
British Journal of Pharmacology 172, pp. 785-798.
Fulltext not available.
Weiss, Stefan, Bernhardt, Günther, Buschauer, Armin and König, Burkhard
(2011)
Synthesis and characterization of DMAP-Modified NPY Y1 receptor antagonists as acyl-transfer catalysts.
Collection of Czechoslovak chemical communications 76 (6), 763 -780.
Fulltext not available.
(2011)
Synthesis and characterization of DMAP-Modified NPY Y1 receptor antagonists as acyl-transfer catalysts.
Collection of Czechoslovak chemical communications 76 (6), 763 -780.
Fulltext not available.
Weiss, Stefan, Keller, Max, Bernhardt, G., Buschauer, Armin and König, Burkhard
(2010)
N(G)-Acyl-argininamides as NPY Y (1) receptor antagonists: Influence of structurally diverse acyl substituents on stability and affinity.
Bioorganic & Medicinal Chemistry (18), pp. 6292-6304.
Fulltext not available.
(2010)
N(G)-Acyl-argininamides as NPY Y (1) receptor antagonists: Influence of structurally diverse acyl substituents on stability and affinity.
Bioorganic & Medicinal Chemistry (18), pp. 6292-6304.
Fulltext not available.
Weiss, Stefan, Keller, Max, Bernhardt, Günther, Buschauer, Armin and König, Burkhard
(2008)
Modular synthesis of non-peptidic bivalent NPY Y(1) receptor antagonists.
Bioorganic & Medicinal Chemistry 16 (22), pp. 9858-9866.
Fulltext not available.
(2008)
Modular synthesis of non-peptidic bivalent NPY Y(1) receptor antagonists.
Bioorganic & Medicinal Chemistry 16 (22), pp. 9858-9866.
Fulltext not available.
Wabnitz, Tobias C., Rizzo, Simona , Götte, Carsten, Buschauer, Armin, Benincori, Tiziana and Reiser, Oliver
(2006)
Enantioselective hydrogenation of diaryl-substituted a,b-unsaturated nitriles.
Tetrahedron Letters 47 (22), pp. 3733-3736.
Fulltext not available.
, Götte, Carsten, Buschauer, Armin, Benincori, Tiziana and Reiser, Oliver
(2006)
Enantioselective hydrogenation of diaryl-substituted a,b-unsaturated nitriles.
Tetrahedron Letters 47 (22), pp. 3733-3736.
Fulltext not available.
Wiest, O., Harrison, C. B., Saettel, N. J. , Cibulka, R. , Sax, M. and König, B.
(2004)
Design, Synthesis, and Evaluation of a Biomimetic Artificial Photolyase Model.
J. Org. Chem. 69, 8183 – 8185.
Fulltext not available.
, Cibulka, R. , Sax, M. and König, B.
(2004)
Design, Synthesis, and Evaluation of a Biomimetic Artificial Photolyase Model.
J. Org. Chem. 69, 8183 – 8185.
Fulltext not available.
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Xie, Sheng-Xue, Schalkhausser, Fabian, Ye, Qi-Zhuang, Seifert, Roland and Buschauer, Armin
(2007)
Effects of Impromidine- and Arpromidine-Derived Guanidines on Recombinant Human and Guinea Pig Histamine H₁ and H₂ Receptors.
Archiv der Pharmazie 340 (1), pp. 9-16.
Xie, Sheng-Xue, Kraus, Anja, Ghorai, Prasanta, Ye, Qi-Zhuang, Elz, Sigurd, Buschauer, Armin and Seifert, Roland
(2006)
N1-(3-Cyclohexylbutanoyl)-N2-[3-(1H-imidazol-4-
yl)propyl]guanidine (UR-AK57), a Potent Partial Agonist for the Human Histamine H1- and H2- Receptors. Journal of Pharmacology and Experimental Therapeutics 317 (3), pp. 1262-1268. Fulltext restricted.
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Xie, Sheng-Xue, Ghorai, Prasanta, Ye, Qi-Zhuang, Buschauer, Armin and Seifert, Roland
(2006)
Probing Ligand-Specific Histamine H1- and H2-Receptor
Conformations with NG-Acylated Imidazolylpropylguanidines. The Journal of Pharmacology and Experimental Therapeutics 317 (1), pp. 139-146. Fulltext restricted.
Conformations with NG-Acylated Imidazolylpropylguanidines. The Journal of Pharmacology and Experimental Therapeutics 317 (1), pp. 139-146. Fulltext restricted.
Xie, Sheng-Xue, Petrache, Georgiana, Schneider, Erich , Ye, Qi-Zhuang, Bernhardt, Günther, Seifert, Roland and Buschauer, Armin
(2006)
Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine.
Bioorganic & Medicinal Chemistry Letters 16 (15), pp. 3886-3890.
Fulltext not available.
, Ye, Qi-Zhuang, Bernhardt, Günther, Seifert, Roland and Buschauer, Armin
(2006)
Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine.
Bioorganic & Medicinal Chemistry Letters 16 (15), pp. 3886-3890.
Fulltext not available.
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Ziemek, Ralf, Schneider, Erich , Kraus, Anja, Cabrele, Chiara , Beck-Sickinger, Annette G., Bernhardt, Günther and Buschauer, Armin
(2007)
Determination of affinity and activity of ligands at the human neuropeptide Y Y4 receptor by flow cytometry and aequorin luminescence.
Journal of Receptors and Signal Transduction 27 (4), pp. 217-233.
Fulltext not available.
, Kraus, Anja, Cabrele, Chiara , Beck-Sickinger, Annette G., Bernhardt, Günther and Buschauer, Armin
(2007)
Determination of affinity and activity of ligands at the human neuropeptide Y Y4 receptor by flow cytometry and aequorin luminescence.
Journal of Receptors and Signal Transduction 27 (4), pp. 217-233.
Fulltext not available.
Zimmermann, Jochen and Angerer, Erwin von
(2007)
Estrogenic and antiestrogenic activities of 2,4-diphenylfuran-based ligands of estrogen receptors α and β.
The Journal of Steroid Biochemistry and Molecular Biology 104 (3-5), pp. 259-268.
Fulltext not available.
Ziemek, Ralf, Brennauer, Albert, Schneider, Erich, Cabrele, Chiara, Beck-Sickinger, Annette G., Bernhardt, Günther and Buschauer, Armin
(2006)
Fluorescence- and luminescence-based methods for the determination of affinity and activity of neuropeptide Y(2) receptor ligands.
European Journal of Pharmacology 551 (1-3), pp. 10-8.
Fulltext not available.
Zimmermann, Jochen, Liebl, Renate and Angerer, Erwin von
(2005)
2,5-Diphenylfuran-based pure antiestrogens with selectivity for the estrogen receptor alpha.
The Journal of Steroid Biochemistry and Molecular Biology 94 (1-3), pp. 57-66.
Fulltext not available.
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Černovská, K., Kemter, M., Gallmeier, H.-C., Rzepecki, P., Schrader, T. and König, B.
(2004)
PEG-supported Synthesis of Pyrazole Oligoamides with Peptide β-Sheet Affinity.
Org. Biomol. Chem. 2, 1603 - 1611.
Fulltext not available.