Anzahl der Einträge in dieser Kategorie: 152.
Artikel
Ertl, Fabian J.,
Kopanchuk, Sergei ,
Dijon, Nicola C.,
Veikšina, Santa,
Tahk, Maris-Johanna ,
Laasfeld, Tõnis,
Schettler, Franziska,
Gattor, Albert O.,
Hübner, Harald,
Archipowa, Nataliya ,
Köckenberger, Johannes,
Heinrich, Markus R.,
Gmeiner, Peter ,
Kutta, Roger Jan ,
Holliday, Nicholas D. ,
Rinken, Ago und
Keller, Max
(2024)
Dually Labeled Neurotensin NTS1R Ligands for Probing Radiochemical and Fluorescence-Based Binding Assays.
Journal of Medicinal Chemistry 67 (18), S. 16664-16691.
Kuck, Katrin,
Unterholzner, Anna,
Lipowicz, Bartosz,
Schwindl, Sebastian,
Jürgenliemk, Guido,
Schmidt, Thomas J. und
Heilmann, Jörg
(2023)
Terpenoids from Myrrh and Their Cytotoxic Activity against HeLa Cells.
Molecules 28 (4), S. 1637.
Bresinsky, Merlin,
Strasser, Jessica M.,
Hubmann, Alexander,
Vallaster, Bernadette,
McCue, William M.,
Fuller, Jessica,
Singh, Gurpreet,
Nelson, Kathryn M.,
Cuellar, Matthew E.,
Finzel, Barry C.,
Ashe, Karen H.,
Walters, Michael A. und
Pockes, Steffen
(2022)
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis.
Archiv der Pharmazie 355 (9), S. 2200095.
Tahk, Maris-Johanna ,
Torp, Jane ,
Ali, Mohammed A. S. ,
Fishman, Dmytro,
Parts, Leopold ,
Grätz, Lukas ,
Müller, Christoph ,
Keller, Max ,
Veiksina, Santa ,
Laasfeld, Tõnis und
Rinken, Ago
(2022)
Live-cell microscopy or fluorescence anisotropy with budded baculoviruses—which way to go with measuring ligand binding to M 4 muscarinic receptors?
Open Biology 12 (6).
Volltext nicht vorhanden.
Lier, Svenja,
Sellmer, Andreas,
Orben, Felix ,
Heinzlmeir, Stephanie,
Krauß, Lukas ,
Schneeweis, Christian,
Hassan, Zonera ,
Schneider, Carolin ,
Patricia Gloria Schäfer, Arlett,
Pongratz, Herwig,
Engleitner, Thomas,
Öllinger, Rupert,
Kuisl, Anna,
Bassermann, Florian,
Schlag, Christoph,
Kong, Bo,
Dove, Stefan,
Kuster, Bernhard,
Rad, Roland,
Reichert, Maximilian,
Wirth, Matthias ,
Saur, Dieter ,
Mahboobi, Siavosh und
Schneider, Günter
(2022)
A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer.
Bioorganic Chemistry 119, S. 105505.
Volltext nicht vorhanden.
Schihada, Hannes,
Klompstra, Thomas M. ,
Humphrys, Laura J. ,
Cervenka, Igor,
Dadvar, Shamim ,
Kolb, Peter ,
Ruas, Jorge L. und
Schulte, Gunnar
(2022)
Isoforms of GPR35 have distinct extracellular N-termini that allosterically modify receptor-transducer coupling and mediate intracellular pathway bias.
Journal of Biological Chemistry 298 (9), S. 102328.
Volltext nicht vorhanden.
Shcherbina, Nadezhda A.,
Kazakov, Igor V.,
Lisovenko, Anna S.,
Kryukova, Mariya A.,
Krasnova, Irina S. ,
Bodensteiner, Michael und
Timoshkin, Alexey Y.
(2022)
Molecular complexes of non-chelating polydentate Lewis bases with group 13 Lewis acids: crystal structure and computed energy of stepwise donor–acceptor bond formation.
Mendeleev Communications 32 (1), S. 74-77.
Volltext nicht vorhanden.
Schindler, Lisa,
Wohlfahrt, Katrin,
Gluhacevic von Krüchten, Lara,
Prante, Olaf,
Keller, Max und
Maschauer, Simone
(2022)
Neurotensin analogs by fluoroglycosylation at Nω-carbamoylated arginines for PET imaging of NTS1-positive tumors.
Scientific Reports 12 (1).
Volltext nicht vorhanden.
Tang, Tingting,
Tan, Qiuxiang,
Han, Shuo,
Diemar, Anne,
Löbner, Kristin,
Wang, Hongyu,
Schüß, Corinna,
Behr, Victoria,
Mörl, Karin,
Wang, Mu,
Chu, Xiaojing,
Yi, Cuiying,
Keller, Max,
Kofoed, Jacob,
Reedtz-Runge, Steffen,
Kaiser, Anette,
Beck-Sickinger, Annette G.,
Zhao, Qiang und
Wu, Beili
(2022)
Receptor-specific recognition of NPY peptides revealed by structures of NPY receptors.
Science Advances 8 (18).
Volltext nicht vorhanden.
Müller, Christoph,
Gleixner, Jakob ,
Tahk, Maris-Johanna ,
Kopanchuk, Sergei ,
Laasfeld, Tõnis,
Weinhart, Michael,
Schollmeyer, Dieter,
Betschart, Martin U.,
Lüdeke, Steffen,
Koch, Pierre,
Rinken, Ago und
Keller, Max
(2022)
Structure-Based Design of High-Affinity Fluorescent Probes for the Neuropeptide Y Y1 Receptor.
Journal of Medicinal Chemistry 65 (6), S. 4832-4853.
Volltext nicht vorhanden.
Rösch, G.,
El Bagdadi, K.,
Muschter, D.,
Taheri, S. ,
Dorn, C.,
Meurer, A.,
Straub, R.H.,
Zaucke, F. ,
Schilling, A.F.,
Grässel, S. und
Jenei-Lanzl, Z.
(2022)
Sympathectomy aggravates subchondral bone changes during osteoarthritis progression in mice without affecting cartilage degeneration or synovial inflammation.
Osteoarthritis and Cartilage 30 (3), S. 461-474.
Volltext nicht vorhanden.
Rosier, Niklas,
Grätz, Lukas,
Schihada, Hannes ,
Möller, Jan,
Işbilir, Ali ,
Humphrys, Laura J. ,
Nagl, Martin,
Seibel, Ulla,
Lohse, Martin J. und
Pockes, Steffen
(2021)
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor.
Journal of Medicinal Chemistry 64 (15), S. 11695-11708.
Volltext nicht vorhanden.
Eap, C. B. ,
Gründer, G. ,
Baumann, P. ,
Ansermot, N.,
Conca, A.,
Corruble, E.,
Crettol, S.,
Dahl, M. L.,
de Leon, J. ,
Greiner, C.,
Howes, O.,
Kim, E.,
Lanzenberger, R.,
Meyer, J. H.,
Moessner, R.,
Mulder, H.,
Müller, D. J.,
Reis, M.,
Riederer, P.,
Ruhe, H. G.,
Spigset, O.,
Spina, E.,
Stegman, B.,
Steimer, W.,
Stingl, J. ,
Suzen, S.,
Uchida, H.,
Unterecker, S.,
Vandenberghe, F. und
Hiemke, C.
(2021)
Tools for optimising pharmacotherapy in psychiatry (therapeutic drug monitoring, molecular brain imaging and pharmacogenetic tests): focus on antidepressants.
The World Journal of Biological Psychiatry 22 (8), S. 561-628.
Volltext nicht vorhanden.
Höring, Carina ,
Seibel, Ulla ,
Tropmann, Katharina,
Grätz, Lukas ,
Mönnich, Denise ,
Pitzl, Sebastian,
Bernhardt, Günther ,
Pockes, Steffen und
Strasser, Andrea
(2020)
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.
International Journal of Molecular Sciences 21 (22), S. 8440.
Grätz, Lukas,
Tropmann, Katharina,
Bresinsky, Merlin,
Müller, Christoph,
Bernhardt, Günther und
Pockes, Steffen
(2020)
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells.
Scientific Reports 10, S. 13288.
Bartole, Edith,
Grätz, Lukas,
Littmann, Timo,
Wifling, David ,
Seibel, Ulla,
Buschauer, Armin und
Bernhardt, Günther
(2020)
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors.
Journal of Medicinal Chemistry 63 (10), S. 5297-5311.
Volltext nicht vorhanden.
Maslanka Figueroa, Sara ,
Fleischmann, Daniel,
Beck, Sebastian,
Tauber, Philipp,
Witzgall, Ralph,
Schweda, Frank und
Goepferich, Achim
(2020)
Nanoparticles Mimicking Viral Cell Recognition Strategies Are Superior Transporters into Mesangial Cells.
Advanced Science 7 (11), S. 1903204.
Dorn, Christoph ,
Schießer, Selina,
Wulkersdorfer, Beatrix,
Hitzenbichler, Florian,
Kees, Martin G. und
Zeitlinger, Markus
(2020)
Determination of free clindamycin, flucloxacillin or tedizolid in plasma: Keep attention to physiological conditions when using ultrafiltration.
Biomedical Chromatography 34, e4820.
Fleischmann, Daniel,
Maslanka-Figueroa, Sara,
Beck, Sebastian,
Abstiens, Kathrin,
Witzgall, Ralph,
Schweda, Frank,
Tauber, Philipp und
Goepferich, Achim
(2020)
Adenovirus-Mimetic Nanoparticles: Sequential Ligand-Receptor Interplay as a Universal Tool for Enhanced In Vitro/In Vivo Cell Identification.
ACS Applied Materials & Interfaces 12 (31), S. 34689-34702.
Volltext nicht vorhanden.
Spinnler, Katrin,
von Krüchten, Lara,
Konieczny, Adam,
Schindler, Lisa,
Bernhardt, Günther und
Keller, Max
(2020)
An Alkyne-functionalized Arginine for Solid-Phase Synthesis Enabling “Bioorthogonal” Peptide Conjugation.
ACS Medicinal Chemistry Letters 11 (3), S. 334-339.
Volltext nicht vorhanden.
Weber, Laura,
Kuck, Katrin,
Jürgenliemk, Guido,
Heilmann, Jörg,
Lipowicz, Bartosz und
Vissiennon, Cica
(2020)
Anti-Inflammatory and Barrier-Stabilising Effects of Myrrh, Coffee Charcoal and Chamomile Flower Extract in a Co-Culture Cell Model of the Intestinal Mucosa.
Biomolecules 10 (7), S. 1033.
Volltext nicht vorhanden.
Ullah, Sami,
Beer, Ronny,
Fuhr, Uwe,
Taubert, Max ,
Zeitlinger, Markus,
Kratzer, Alexander,
Dorn, Christoph,
Arshad, Usman,
Kofler, Mario und
Helbok, Raimund
(2020)
Brain Exposure to Piperacillin in Acute Hemorrhagic Stroke Patients Assessed by Cerebral Microdialysis and Population Pharmacokinetics.
Neurocritical Care.
Bohley, Marilena S.,
Birch, Emily,
Baumann, Felix J.,
Dillinger, Andrea E.,
Tamm, Ernst R. und
Goepferich, Achim M.
(2020)
Design of dye and superparamagnetic iron oxide nanoparticle loaded lipid nanocapsules with dual detectability in vitro and in vivo.
International Journal of Pharmaceutics 585, S. 119433.
Volltext nicht vorhanden.
Gruber, Corinna G.,
Pegoli, Andrea,
Müller, Christoph,
Grätz, Lukas,
She, Xueke und
Keller, Max
(2020)
Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity.
RSC Medicinal Chemistry 11 (7), S. 823-832.
Volltext nicht vorhanden.
Keller, Max,
Mahuroof, Shahani A.,
Hong Yee, Vivyanne,
Carpenter, Jessica,
Schindler, Lisa,
Littmann, Timo,
Pegoli, Andrea,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter und
Holliday, Nicholas D.
(2020)
Fluorescence Labeling of Neurotensin(8–13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
ACS Medicinal Chemistry Letters 11 (1), S. 16-22.
Volltext nicht vorhanden.
Biselli, Sabrina,
Alencastre, Inês,
Tropmann, Katharina,
Erdmann, Daniela,
Chen, Mengya,
Littmann, Timo,
Maia, André F. ,
Gomez-Lazaro, Maria,
Tanaka, Miho,
Ozawa, Takeaki,
Keller, Max,
Lamghari, Meriem,
Buschauer, Armin und
Bernhardt, Günther
(2020)
Fluorescent H2 Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications.
ACS Medicinal Chemistry Letters 11 (8), S. 1521-1528.
Volltext nicht vorhanden.
Abdellatif, Ahmed ,
Hennig, Robert,
Pollinger, Klaus,
Tawfeek, Hesham,
Goepferich, Achim und
make_name_string expected hash reference
(2020)
Fluorescent Nanoparticles Coated with a Somatostatin Analogue Target Blood Monocyte for Efficient Leukaemia Treatment.
Pharmaceutical Research 37 (11), S. 2017.
Sommer, Judith,
Dorn, Christoph ,
Gäbele, Erwin,
Bataille, Frauke,
Freese, Kim,
Seitz, Tatjana,
Thasler, Wolfgang E.,
Büttner, Reinhard,
Weiskirchen, Ralf ,
Bosserhoff, Anja und
Hellerbrand, Claus
(2020)
Four-And-A-Half LIM-Domain Protein 2 (FHL2) Deficiency Aggravates Cholestatic Liver Injury.
Cells 9 (1), S. 248.
Apaolaza, P.S. ,
Busch, M.,
Asin-Prieto, E. ,
Peynshaert, K. ,
Rathod, R.,
Remaut, K.,
Dünker, N. und
Göpferich, A.
(2020)
Hyaluronic acid coating of gold nanoparticles for intraocular drug delivery: Evaluation of the surface properties and effect on their distribution.
Experimental Eye Research 198, S. 108151.
Volltext nicht vorhanden.
Biswas, Siladitta,
Kojonazarov, Baktybek,
Hadzic, Stefan,
Majer, Michael,
Bajraktari, Ganimete,
Novoyatleva, Tatyana,
Ghofrani, Hossein Ardeschir,
Grimminger, Friedrich,
Seeger, Werner,
Weissmann, Norbert,
Schlossmann, Jens und
Schermuly, Ralph Theo
(2020)
IRAG1 Deficient Mice Develop PKG1β Dependent Pulmonary Hypertension.
Cells 9 (10), S. 2280.
Volltext nicht vorhanden.
Yagati, Ajay Kumar ,
Behrent, Arne,
Beck, Sebastian,
Rink, Simone,
Goepferich, Achim M.,
Min, Junhong ,
Lee, Min-Ho und
Baeumner, Antje J.
(2020)
Laser-induced graphene interdigitated electrodes for label-free or nanolabel-enhanced highly sensitive capacitive aptamer-based biosensors.
Biosensors and Bioelectronics 164, S. 112272.
Volltext nicht vorhanden.
Pontes de Sousa, Ingrid,
Ferreira, Antônio Gilberto ,
Miller Crotti, Antônio Eduardo,
Alves dos Santos, Raquel,
Kiermaier, Josef,
Kraus, Birgit,
Heilmann, Jörg und
Jacometti Cardoso Furtado, Niege Araçari
(2020)
New antifungal ent-labdane diterpenes against Candida glabrata produced by microbial transformation of ent-polyalthic acid.
Bioorganic Chemistry 95, S. 103560.
Volltext nicht vorhanden.
Ehmann, L.,
Simon, P.,
Busse, D.,
Petroff, D.,
Dorn, Christoph ,
Huisinga, W.,
Dietrich, A.,
Zeitlinger, M.,
Wrigge, H. und
Kloft, C.
(2020)
Risk of target non-attainment In obese compared to non-obese patients In Calculated linezolid therapy.
Clinical Microbiology and Infection.
Volltext nicht vorhanden.
Stolwijk, Judith A.,
Mildner, Anne-Kathrin,
Kade, Christian,
Skiba, Michael,
Bernhardt, Guenther,
Buschauer, Armin,
Huebner, Harald,
Gmeiner, Peter und
Wegener, Joachim
(2020)
Stepwise Dosing Protocol for Increased Throughput in Label-Free Impedance-Based GPCR Assays.
Journal of Visualized Experiments (156).
Volltext nicht vorhanden.
Maschauer, Simone,
Ott, Julian J. ,
Bernhardt, Günther,
Kuwert, Torsten,
Keller, Max und
Prante, Olaf
(2019)
18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET Imaging of mammary carcinoma.
Scientific Reports 9, S. 12990.
Schramm, Andrea,
Schweda, Frank,
Sequeira-Lopez, Maria Luisa S.,
Hofmann, Franz,
Sandner, Peter und
Schlossmann, Jens
(2019)
Protein Kinase G Is Involved in Acute but Not in Long-Term Regulation of Renin Secretion.
Frontiers in Pharmacology 2019 (10), S. 800.
Dorn, Christoph,
Petroff, David,
Neumann, Nancy,
Kratzer, Alexander,
El-Najjar, Nahed ,
Dietrich, Arne,
Kloft, Charlotte,
Zeitlinger, Markus ,
Kees, Martin,
Kees, Frieder,
Wrigge, Hermann und
Simon, Philipp
(2019)
Plasma and tissue pharmacokinetics of fosfomycin in morbidly obese and non-obese surgical patients: a controlled clinical trial.
Journal of Antimicrobial Chemotherapy.
Volltext nicht vorhanden.
Pegoli, Andrea,
Wifling, David ,
Gruber, Corinna G.,
Xueke, She,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter und
Keller, Max
(2019)
Conjugation of Short Peptides to Dibenzodiazepinone-Type
Muscarinic Acetylcholine Receptor Ligands Determines M2R
Selectivity.
Journal of Medicinal Chemistry 62, S. 5358-5369.
Volltext nicht vorhanden.
Schramm, Simon,
Agnetta, Luca,
Bermudez, Marcel,
Gerwe, Hubert,
Irmen, Matthias,
Holze, Janine,
Littmann, Timo,
Wolber, Gerhard ,
Tränkle, Christian und
Decker, Michael
(2019)
Novel BQCA‐ and TBPB‐Derived M 1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.
ChemMedChem 14 (14), S. 1349-1358.
Volltext nicht vorhanden.
Łażewska, Dorota ,
Mogilski, Szczepan,
Hagenow, Stefanie ,
Kuder, Kamil,
Głuch-Lutwin, Monika ,
Siwek, Agata ,
Więcek, Małgorzata,
Kaleta, Maria,
Seibel, Ulla,
Buschauer, Armin,
Filipek, Barbara,
Stark, Holger und
Kieć-Kononowicz, Katarzyna
(2019)
Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands.
Bioorganic & Medicinal Chemistry 27 (7), S. 1254-1262.
Volltext nicht vorhanden.
Polykandriotis, Elias,
Horch, Raymund E.,
Jost, Matthias,
Arkudas, Andreas,
Kees, Frieder und
Schmitz, Marweh
(2019)
Can systemically administered antibiotics be detected in wound tissues and surfaces under negative pressure wound therapy?
International Wound Journal 16 (2), S. 503-510.
Volltext nicht vorhanden.
Kowalewski, Christoph,
Haen, Ekkehard,
Hiemke, Christoph,
Ridders, Florian,
Endres, Katharina,
Gründer, Gerhard,
Paulzen, Michael und
Schoretsanitis, Georgios
(2019)
Cytochrome P450-mediated inhibition of venlafaxine metabolism by trimipramine.
International Clinical Psychopharmacology 34 (5), S. 241-246.
Volltext nicht vorhanden.
Dorn, Christoph ,
Kratzer, Alexander Ludwig,
Schießer, Selina,
Kees, Frieder ,
Wrigge, Hermann und
Simon, Philipp
(2019)
Determination of total or free cefazolin and metronidazole in human plasma or interstitial fluid by HPLC-UV for pharmacokinetic studies in man.
Journal of Chromatography B.
Volltext nicht vorhanden.
Agnetta, Luca,
Bermudez, Marcel ,
Riefolo, Fabio ,
Matera, Carlo ,
Claro, Enrique ,
Messerer, Regina,
Littmann, Timo,
Wolber, Gerhard ,
Holzgrabe, Ulrike und
Decker, Michael
(2019)
Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties.
Journal of Medicinal Chemistry 62 (6), S. 3009-3020.
Volltext nicht vorhanden.
Walz, Johanna M.,
Wecker, Thomas ,
Zhang, Pei Pei,
Cakir, Bertan,
Gruening, Bjoern,
Agostini, Hansjuergen,
Reuer, Tristan,
Ludwig, Franziska,
Boneva, Stefaniya ,
Faerber, Lothar,
Lange, Clemens,
Schlunck, Guenther R. und
Stahl, Andreas
(2019)
Impact of angiogenic activation and inhibition on miRNA profiles of human retinal endothelial cells.
Experimental Eye Research 181, S. 98-104.
Volltext nicht vorhanden.
Stolwijk, J. A.,
Skiba, M.,
Kade, C.,
Bernhardt, G.,
Buschauer, Armin ,
Hübner, H.,
Gmeiner, P. und
Wegener, Joachim
(2019)
Increasing the throughput of label-free cell assays to study the activation of G-protein-coupled receptors by using a serial agonist exposure protocol.
Integrative Biology 11 (3), S. 99-108.
Volltext nicht vorhanden.
Gergs, U. ,
Bernhardt, Günther,
Buchwalow, I. B.,
Edler, H.,
Fröba, J.,
Keller, Max,
Kirchhefer, U.,
Köhler, F.,
Mißlinger, N.,
Wache, H. und
Neumann, J.
(2019)
Initial Characterization of Transgenic Mice Overexpressing Human Histamine H2 Receptors.
Journal of Pharmacology and Experimental Therapeutics 369 (1), S. 129-141.
Volltext nicht vorhanden.
Schoretsanitis, Georgios ,
Haen, Ekkehard,
Hiemke, Christoph,
Endres, Katharina,
Ridders, Florian,
Veselinovic, Tanja,
Gründer, Gerhard und
Paulzen, Michael
(2019)
Pharmacokinetic correlates of venlafaxine: associated adverse reactions.
European Archives of Psychiatry and Clinical Neuroscience 269 (7), S. 851-857.
Volltext nicht vorhanden.
Heider, Fabian ,
Ansideri, Francesco,
Tesch, Roberta,
Pantsar, Tatu,
Haun, Urs,
Döring, Eva,
Kudolo, Mark,
Poso, Antti ,
Albrecht, Wolfgang,
Laufer, Stefan A. und
Koch, Pierre
(2019)
Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors.
European Journal of Medicinal Chemistry 175, S. 309-329.
Volltext nicht vorhanden.
Nowak, Hartmuth,
Weidemann, Caroline,
Martini, Stefan,
Oesterreicher, Zoe Anne,
Dorn, Christoph,
Adamzik, Michael,
Kees, Frieder,
Zeitlinger, Markus und
Rahmel, Tim
(2019)
Repeated determination of moxifloxacin concentrations in interstitial space fluid of muscle and subcutis in septic patients.
Journal of Antimicrobial Chemotherapy.
Volltext nicht vorhanden.
Kratzer, Alexander,
Schießer, Selina,
Matzneller, Peter,
Wulkersdorfer, Beatrix,
Zeitlinger, Markus ,
Schlossmann, Jens ,
Kees, Frieder und
Dorn, Christoph
(2018)
Determination of Total and Free Ceftolozane and Tazobactam in Human Plasma and Interstitial Fluid by HPLC-UV.
Journal of Pharmaceutical and Biomedical Analysis.
Volltext nicht vorhanden.
Walz, J. M.,
Bemme, S.,
Reichl, S.,
Akman, S.,
Breuß, H.,
Süsskind, D.,
Glitz, B.,
Müller, V. C.,
Wagenfeld, L.,
Gabel-Pfisterer, A.,
Aisenbrey, S.,
Engelmann, K.,
Koutsonas, A.,
Krohne, T. U. und
Stahl, A.
(2018)
Behandelte Frühgeborenenretinopathie in Deutschland.
Der Ophthalmologe 115 (6), S. 476-488.
Volltext nicht vorhanden.
Leonhardt, Michel,
Sellmer, Andreas ,
Krämer, Oliver H.,
Dove, Stefan,
Elz, Sigurd,
Kraus, Birgit,
Beyer, Mandy und
Mahboobi, Siavosh
(2018)
Design and biological evaluation of tetrahydro-β-carboline derivatives as highly potent histone deacetylase 6 (HDAC6) inhibitors.
European Journal of Medicinal Chemistry 152, S. 329-357.
Volltext nicht vorhanden.
Ridinger, Johannes,
Koeneke, Emily,
Kolbinger, Fiona R.,
Koerholz, Katharina,
Mahboobi, Siavosh,
Hellweg, Lars,
Gunkel, Nikolas,
Miller, Aubry K.,
Peterziel, Heike,
Schmezer, Peter,
Hamacher-Brady, Anne ,
Witt, Olaf und
Oehme, Ina
(2018)
Dual role of HDAC10 in lysosomal exocytosis and DNA repair promotes neuroblastoma chemoresistance.
Scientific Reports 8 (1).
Volltext nicht vorhanden.
Dorn, Christoph,
Kratzer, Alexander,
Liebchen, Uwe,
Schleibinger, Michael,
Murschhauser, Alexandra,
Schlossmann, Jens ,
Kees, Frieder,
Simon, Philipp und
Kees, Martin G.
(2018)
Impact of Experimental Variables on the Protein Binding of Tigecycline in Human Plasma as Determined by Ultrafiltration.
Journal of Pharmaceutical Sciences 107 (2), S. 739-744.
Volltext nicht vorhanden.
Sellmer, Andreas,
Stangl, Hubert,
Beyer, Mandy,
Grünstein, Elisabeth,
Leonhardt, Michel,
Pongratz, Herwig,
Eichhorn, Emerich,
Elz, Sigurd,
Striegl, Birgit,
Jenei-Lanzl, Zsuzsa,
Dove, Stefan,
Straub, Rainer H.,
Krämer, Oliver H. und
Mahboobi, Siavosh
(2018)
Marbostat-100 Defines a New Class of Potent and Selective Antiinflammatory and Antirheumatic Histone Deacetylase 6 Inhibitors.
Journal of Medicinal Chemistry 61 (8), S. 3454-3477.
Volltext nicht vorhanden.
Schoretsanitis, Georgios,
de Leon, Jose,
Haen, Ekkehard,
Stegmann, Benedikt,
Hiemke, Christoph,
Gründer, Gerhard und
Paulzen, Michael
(2018)
Pharmacokinetics of risperidone in different application forms – Comparing long-acting injectable and oral formulations.
European Neuropsychopharmacology 28 (1), S. 130-137.
Volltext nicht vorhanden.
Mathioudaki, Angeliki,
Berzesta, Ariola,
Kypriotakis, Zacharias,
Skaltsa, Helen und
Heilmann, Jörg
(2018)
Phenolic metabolites from Hypericum kelleri Bald., an endemic species of Crete (Greece).
Phytochemistry 146, S. 1-7.
Volltext nicht vorhanden.
Peña-Solórzano, Diana,
Scholler, Matthias,
Bernhardt, Günther,
Buschauer, Armin ,
König, Burkhard und
Ochoa-Puentes, Cristian
(2018)
Tariquidar-Related Chalcones and Ketones as ABCG2 Modulators.
ACS Medicinal Chemistry Letters 9, S. 854-859.
Volltext nicht vorhanden.
She, Xueke,
Pegoli, Andrea,
Mayr, Judith,
Hübner, Harald,
Bernhardt, Günther ,
Gmeiner, Peter und
Keller, Max
(2017)
Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity.
ACS Omega 2 (10), S. 6741-6754.
Dukorn, Stefanie,
Littmann, Timo,
Keller, Max,
Kuhn, Kilian K.,
Cabrele, Chiara ,
Baumeister, Paul,
Bernhardt, Günther und
Buschauer, Armin
(2017)
Fluorescence- and radio-labeling of Lys4,Nle17,30hPP yields molecular tools for the NPY Y4 receptor.
Bioconjugate Chemistry.
Volltext nicht vorhanden.
Noack, Katrin,
Mahendrarajah, Nisintha,
Hennig, Dorle,
Schmidt, Luisa,
Grebien, Florian ,
Hildebrand, Dagmar,
Christmann, Markus,
Kaina, Bernd,
Sellmer, Andreas,
Mahboobi, Siavosh,
Kubatzky, Katharina,
Heinzel, Thorsten und
Krämer, Oliver H.
(2017)
Analysis of the interplay between all-trans retinoic acid and histone deacetylase inhibitors in leukemic cells.
Archives of Toxicology 91 (5), S. 2191-2208.
Volltext nicht vorhanden.
Schäfer, Claudia,
Göder, Anja,
Beyer, Mandy,
Kiweler, Nicole,
Mahendrarajah, Nisintha,
Rauch, Anke,
Nikolova, Teodora,
Stojanovic, Natasa,
Wieczorek, Martin,
Reich, Thomas R.,
Tomicic, Maja T.,
Linnebacher, Michael,
Sonnemann, Jürgen,
Dietrich, Sascha,
Sellmer, Andreas,
Mahboobi, Siavosh,
Heinzel, Thorsten,
Schneider, Günter und
Krämer, Oliver H.
(2017)
Class I histone deacetylases regulate p53/NF-κB crosstalk in cancer cells.
Cellular Signalling 29, S. 218-225.
Volltext nicht vorhanden.
Schoretsanitis, Georgios ,
Haen, Ekkehard,
Stegmann, Benedikt,
Hiemke, Christoph,
Gründer, Gerhard und
Paulzen, Michael
(2017)
Effect of smoking on risperidone pharmacokinetics – A multifactorial approach to better predict the influence on drug metabolism.
Schizophrenia Research 185, S. 51-57.
Volltext nicht vorhanden.
Mahendrarajah, Nisintha,
Borisova, Marina E.,
Reichardt, Sigrid,
Godmann, Maren,
Sellmer, Andreas,
Mahboobi, Siavosh,
Haitel, Andrea,
Schmid, Katharina,
Kenner, Lukas ,
Heinzel, Thorsten,
Beli, Petra und
Krämer, Oliver H.
(2017)
HSP90 is necessary for the ACK1-dependent phosphorylation of STAT1 and STAT3.
Cellular Signalling 39, S. 9-17.
Volltext nicht vorhanden.
Kuhn, Kilian K.,
Littmann, Timo,
Dukorn, Stefanie,
Tanaka, Miho,
Keller, Max,
Ozawa, Takeaki,
Bernhardt, Günther und
Buschauer, Armin
(2017)
In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists.
ACS Omega 2 (7), S. 3616-3631.
Pegoli, Andrea ,
She, Xueke,
Wifling, David ,
Hübner, Harald,
Bernhardt, Günther,
Gmeiner, Peter und
Keller, Max
(2017)
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.
Journal of Medicinal Chemistry 60 (8), S. 3314-3334.
Volltext nicht vorhanden.
Lieb, Sebastian,
Littmann, Timo,
Plank, Nicole,
Felixberger, Johannes,
Tanaka, Miho,
Schäfer, Thorsten,
Krief, Stéphane,
Elz, Sigurd,
Friedland, Kristina,
Bernhardt, Günther,
Wegener, Joachim,
Ozawa, Takeaki und
Buschauer, Armin
(2016)
Label-free versus conventional cellular assays: functional investigations on the human histamine H1 receptor.
Pharmacological Research 114, S. 13-26.
Volltext nicht vorhanden.
Töpper, Christoph,
Steinbach, Cathérine Louise,
Dorn, Christoph ,
Kratzer, Alexander,
Wicha, Sebastian G.,
Schleibinger, Michael,
Liebchen, Uwe,
Kees, Frieder,
Salzberger, Bernd und
Kees, Martin G.
(2016)
Variable linezolid exposure in ICU patients—possible role of drug-drug interactions.
Therapeutic Drug Monitoring 38 (5), S. 573-578.
Volltext nicht vorhanden.
Schlossmann, Jens,
Wetzl, Veronika,
Schinner, Elisabeth,
Kees, Frieder K.,
Hofmann, Franz und
Faerber, Lothar
(2016)
Involvement of cyclic guanosine monophosphate-dependent protein kinase I in renal antifibrotic effects of serelaxin.
Frontiers in Pharmacology 7 (195), S. 1-27.
Kuhn, Kilian K.,
Ertl, Thomas,
Dukorn, Stefanie,
Keller, Max,
Bernhardt, Günther,
Reiser, Oliver und
Buschauer, Armin
(2016)
High affinity agonists of the neuropeptide Y (NPY) Y4 receptor derived from the C-terminal pentapeptide of human pancreatic polypeptide (hPP): synthesis, stereochemical discrimination and radiolabeling.
Journal of Medicinal Chemistry 59 (13), S. 6045-6058.
Volltext nicht vorhanden.
Lorenz, Peter,
Knittel, Diana N.,
Conrad, Jürgen,
Lotter, Eva M.,
Heilmann, Jörg,
Stintzing, Florian C. und
Kammerer, Dietmar R.
(2016)
1-Acetyl-3-[(3R)-hydroxyfatty acyl]glycerols: Lipid Compounds fromEuphrasia rostkovianaHayneandE. tetraquetra(Bréb.)Arrond.
Chemistry & Biodiversity 13 (5), S. 602-612.
Volltext nicht vorhanden.
Hammer, Sebastian,
Gobleder, Susanne,
Naporra, Franziska,
Wittmann, Hans-Joachim,
Elz, Sigurd,
Heinrich, Markus und
Strasser, Andrea
(2016)
2,4-Diaminopyrimidines as dual ligands at the histamine H1 and H4 receptor - H1/H4-receptor selectivity.
Bioorganic & Medicinal Chemistry Letters 26, S. 292-300.
Volltext nicht vorhanden.
Sawatzky, Edgar,
Wehle, Sarah,
Kling, Beata,
Wendrich, Jan,
Bringmann, Gerhard,
Sotriffer, Christoph A.,
Heilmann, Jörg und
Decker, Michael
(2016)
Discovery of Highly Selective and Nanomolar Carbamate-Based Butyrylcholinesterase Inhibitors by Rational Investigation into Their Inhibition Mode.
Journal of Medicinal Chemistry 59 (5), S. 2067-2082.
Volltext nicht vorhanden.
Keller, Max,
Kuhn, Kilian K.,
Einsiedel, Jürgen,
Hübner, Harald,
Biselli, Sabrina,
Mollereau, Catherine ,
Wifling, David,
Svobodova, Jaroslava,
Bernhardt, Günther,
Cabrele, Chiara ,
Vanderheyden, Patrick,
Gmeiner, Peter und
Buschauer, Armin
(2016)
Mimicking of arginine by functionalized Nω-carbamoylated arginine as a new broadly applicable approach to labeled bioactive peptides: high affinity angiotensin, neuropeptide Y, neuropeptide FF and neurotensin receptor ligands as examples.
Journal of Medicinal Chemistry 59 (5), S. 1925-1945.
Volltext nicht vorhanden.
Khan, Nadia,
Saad, Ali,
Nurulain, Syed M.,
Darras, Fouad H.,
Decker, Michael und
Sadek, Bassem
(2016)
The dual-acting H3 receptor antagonist and AChE inhibitor UW-MD-71 dose-dependently enhances memory retrieval and reverses dizocilpine-induced memory impairment in rats.
Behavioural Brain Research 297, S. 155-164.
Volltext nicht vorhanden.
Huang, Guozheng ,
Schramm, Simon,
Heilmann, Jörg,
Biedermann, David,
Křen, Vladimír und
Decker, Michael
(2016)
Unconventional application of the Mitsunobu reaction: Selective flavonolignan dehydration yielding hydnocarpins.
Beilstein Journal of Organic Chemistry 12, S. 662-669.
Volltext nicht vorhanden.
Dolles, Dominik,
Nimczick, Martin,
Scheiner, Matthias,
Ramler, Jacqueline,
Stadtmüller, Patricia,
Sawatzky, Edgar,
Drakopoulos, Antonios ,
Sotriffer, Christoph,
Wittmann, Hans-Joachim,
Strasser, Andrea und
Decker, Michael
(2015)
Aminobenzimidazoles and Structural Isomers as Templates for Dual-Acting Butyrylcholinesterase Inhibitors andhCB2R Ligands To Combat Neurodegenerative Disorders.
ChemMedChem 11 (12), S. 1270-1283.
Volltext nicht vorhanden.
Egger, M.,
Pellett, P.,
Nickl, K.,
Geiger, S.,
Graetz, S.,
Seifert, R.,
Heilmann, J. und
König, B.
(2008)
Synthesis and Cannabinoid Receptor Activity of Ketoalkenes from Echinacea pallida and Non-natural Analogues.
Chem. Eur. J. 14, 10978 - 10984.
Volltext nicht vorhanden.
Schlegel, Birgit,
Laggner, Christian,
Meier, Rene,
Langer, Thierry,
Schnell, David,
Seifert, Roland,
Stark, Holger,
Höltje, Hans-Dieter und
Sippl, Wolfgang
(2007)
Generation of a homology model of the human histamine H₃ receptor for ligand docking and pharmacophore-based screening.
Journal of Computer-Aided Molecular Design.
Monographie
Hochschulschrift der Universität Regensburg
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